Actively Recruiting

Phase 1
Age: 18Years +
MALE
NCT07145177

177Lu-PSMA-617 With Liver Directed Therapy in Metastatic Castration Resistant Prostate Cancer

Led by University of California, San Francisco · Updated on 2026-03-23

30

Participants Needed

1

Research Sites

241 weeks

Total Duration

On this page

Sponsors

U

University of California, San Francisco

Lead Sponsor

N

Novartis

Collaborating Sponsor

AI-Summary

What this Trial Is About

This is an open label, single arm, phase 1b study to determine the safety of combining sequential Prostate-Specific Membrane Antigen (PSMA)-targeted 177Lu-PSMA-617 radionuclide therapy with liver-directed therapy in metastatic castrate-resistant prostate cancer (mCRPC) patients with liver metastases amenable to liver-directed therapy who have progressed on at least one prior androgen pathway inhibitor.

CONDITIONS

Official Title

177Lu-PSMA-617 With Liver Directed Therapy in Metastatic Castration Resistant Prostate Cancer

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Histologically confirmed prostate cancer.
  • Progressive disease by PCWG3 criteria at study entry.
  • Male participants who are at least 18 years of age on the day of signing informed consent.
  • Castrate level of serum testosterone at study entry (< 50 ng/dL). Participants without prior bilateral orchiectomy must remain on LHRH analogue treatment during the study.
  • Prior progression on at least one second generation androgen signaling inhibitor (abiraterone, apalutamide, darolutamide, and/or enzalutamide).
  • Recovery from adverse events related to prior anti-cancer treatment to Grade ≤ 1 (except alopecia and Grade ≤ 2 neuropathy).
  • Prior external beam radiotherapy allowed if last treatment was > 2 weeks before study treatment start and participant recovered from radiation toxicities.
  • At least one PSMA-avid extrahepatic lesion on screening PSMA PET; liver lesions may be PSMA PET-negative or positive.
  • Availability of archival mCRPC tissue or willingness to undergo biopsy if no archival tissue available.
  • Presence of one or more liver metastases amenable to liver-directed therapy.
  • ECOG performance status ≤ 2 or Karnofsky score ≥ 50%.
  • Adequate organ function as defined by specific blood counts, liver and kidney function tests.
  • Participants with treated brain metastases eligible if last treatment > 28 days prior and no new/progressive brain metastases on MRI.
  • Use of appropriate contraception during and for 6 months after study treatment.
  • Ability to understand and willingness to sign informed consent.
Not Eligible

You will not qualify if you...

  • De novo small cell neuroendocrine prostate cancer.
  • One or more extrahepatic soft tissue lesions > lymph nodes 1.5 cm or visceral/soft tissue lesions > 1 cm on CT that are PSMA PET-negative; non-PSMA avid liver lesions allowed.
  • Receipt of other systemic anti-cancer therapies within 14 days or 5 half-lives before study treatment, except LHRH analogues.
  • Prior PSMA-directed radioligand treatment.
  • More than 2 prior lines of taxane-based chemotherapy in the castration-resistant setting.
  • Previous bilio-enteric anastomosis, ampulla of Vater sphincterotomy, biliary stent, or biliary drain through ampulla.
  • Participation in another investigational study within 4 weeks prior to first dose.
  • Clinically significant cardiovascular disease including uncontrolled heart failure, recent myocardial infarction, unstable angina, stroke within 6 months, or uncontrolled arrhythmias.
  • Major surgery within 28 days before study treatment without adequate recovery.
  • Secondary malignancy requiring active treatment except certain low-risk cancers.
  • Active infection requiring intravenous antibiotics within 7 days before study treatment.
  • Known active Hepatitis B or C infections unless controlled with antiviral therapy.
  • Not a candidate for liver-directed therapy due to bleeding disorders, anticoagulation, or significant ascites.
  • Unable or unwilling to follow radiation safety precautions.
  • Any condition impairing ability to comply with study procedures as judged by investigator.

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 1 location

1

University of California, San Francisco

San Francisco, California, United States, 94143

Actively Recruiting

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Research Team

M

Maya Aslam

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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