Actively Recruiting

Phase 1
Age: 18Years - 100Years
All Genders
NCT05870579

[177Lu]Lu-NeoB in Combination With Ribociclib and Fulvestrant in Participants With ER+, HER2- and GRPR+ Advanced Breast Cancer

Led by Novartis Pharmaceuticals · Updated on 2026-04-30

48

Participants Needed

25

Research Sites

428 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The purpose of this trial is to estimate the recommended dose (RD) of \[177Lu\]Lu-NeoB in combination with ribociclib and fulvestrant in participants with estrogen receptor (ER) positive (ER+), human epidermal growth factor receptor-2 (HER2) negative (HER2-) and gastrin releasing peptide receptor (GRPR) positive (GRPR+) advanced breast cancer experiencing early relapse from (neo)adjuvant endocrine therapy or who have progressed on endocrine therapy in combination with a CDK4/6 inhibitor for advanced disease.

CONDITIONS

Official Title

[177Lu]Lu-NeoB in Combination With Ribociclib and Fulvestrant in Participants With ER+, HER2- and GRPR+ Advanced Breast Cancer

Who Can Participate

Age: 18Years - 100Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Adult female or male 18 years of age or older at the time of informed consent
  • Confirmed diagnosis of estrogen receptor positive breast cancer with ER >10%
  • HER2 negative breast cancer verified by local laboratory testing
  • Advanced breast cancer that is locoregionally recurrent or metastatic
  • Relapsed within 12 months from (neo)adjuvant endocrine therapy without advanced disease treatment, or relapsed >12 months and progressed after one line of endocrine therapy (except fulvestrant), or advanced breast cancer at diagnosis progressed after one line of endocrine therapy (except fulvestrant)
  • At least one measurable target lesion showing uptake on PET imaging using [68Ga]Ga-NeoB
  • Adequate bone marrow and organ function
  • QTcF interval less than 450 msec and resting heart rate between 50-90 bpm
  • ECOG performance status of 0 or 1
Not Eligible

You will not qualify if you...

  • More than one prior treatment line for advanced/metastatic breast cancer
  • Prior treatment with fulvestrant
  • Previous ribociclib dose reduction due to safety concerns
  • Relapse or progression within 6 months after CDK4/6 inhibitor therapy
  • Symptomatic visceral disease or disease burden unsuitable for ribociclib plus endocrine therapy
  • Central nervous system involvement unless stable and off steroids or enzyme-inducing anti-epileptics for at least 4 weeks
  • Current use of warfarin or Coumadin anticoagulants
  • Diagnosis of inflammatory breast cancer
  • Child Pugh score B or C
  • History or current significant cardiac disease or ECG abnormalities
  • Known allergy to study drugs or their components
  • Recent radiopharmaceutical treatment without sufficient clearance time
  • Recent radiotherapy with unresolved side effects affecting safety
  • Recent systemic corticosteroid use without recovery
  • History of acute pancreatitis within 1 year
  • Current use of medications or supplements affecting cytochrome P450 3A4 metabolism or prolonging QT interval that cannot be discontinued
  • Current use of NEP inhibitors preventing dosimetry imaging
  • Other protocol-specified criteria may apply

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 25 locations

1

UCLA Jonsson Comp Cancer Center

Los Angeles, California, United States, 90095

Actively Recruiting

2

Hoag Memorial Hospital Presbyterian

Newport Beach, California, United States, 92663

Actively Recruiting

3

University of Kansas Medical Center

Westwood, Kansas, United States, 66205

Actively Recruiting

4

University of Pennsylvania

Philadelphia, Pennsylvania, United States, 19104

Actively Recruiting

5

MD Anderson Cancer Center

Houston, Texas, United States, 77030

Actively Recruiting

6

Utah Intermountain Medical Center

Murray, Utah, United States, 84107

Actively Recruiting

7

Novartis Investigative Site

Guangzhou, China, 510060

Actively Recruiting

8

Novartis Investigative Site

Shanghai, China, 200032

Actively Recruiting

9

Novartis Investigative Site

Tianjin, China, 300300

Actively Recruiting

10

Novartis Investigative Site

Saint-Cloud, Hauts De Seine, France, 92210

Actively Recruiting

11

Novartis Investigative Site

Bordeaux, France, 33076

Actively Recruiting

12

Novartis Investigative Site

Clermont-Ferrand, France, 63011

Actively Recruiting

13

Novartis Investigative Site

Saint-Herblain, France, 44805

Actively Recruiting

14

Novartis Investigative Site

Strasbourg, France, F 67085

Actively Recruiting

15

Novartis Investigative Site

Cologne, North Rhine-Westphalia, Germany, 50937

Actively Recruiting

16

Novartis Investigative Site

Erlangen, Germany, 91054

Actively Recruiting

17

Novartis Investigative Site

Essen, Germany, 45147

Actively Recruiting

18

Novartis Investigative Site

München, Germany, 80377

Actively Recruiting

19

Novartis Investigative Site

Gliwice, Poland, 44 101

Actively Recruiting

20

Novartis Investigative Site

Porto, Portugal, 4200-072

Actively Recruiting

21

Novartis Investigative Site

L'Hospitalet de Llobregat, Barcelona, Spain, 08907

Actively Recruiting

22

Novartis Investigative Site

Barcelona, Spain, 08035

Actively Recruiting

23

Novartis Investigative Site

Barcelona, Spain, 08036

Actively Recruiting

24

Novartis Investigative Site

Madrid, Spain, 28034

Actively Recruiting

25

Novartis Investigative Site

Madrid, Spain, 28040

Actively Recruiting

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Research Team

N

Novartis Pharmaceuticals

CONTACT

N

Novartis Pharmaceuticals

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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