Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
NCT05608252

VS-6766+Abema+Fulv in Met HR+/HER- BC

Led by Adrienne G. Waks · Updated on 2026-04-30

63

Participants Needed

3

Research Sites

305 weeks

Total Duration

On this page

Sponsors

A

Adrienne G. Waks

Lead Sponsor

V

Verastem, Inc.

Collaborating Sponsor

AI-Summary

What this Trial Is About

This research is being done to evaluate the safety and effectiveness of a drug currently known as VS-6766 in combination with the drugs abemaciclib and fulvestrant in HR+/HER2-negative breast cancer. The names of the study drugs involved in this study are: * VS-6766 * Abemaciclib * Fulvestrant

CONDITIONS

Official Title

VS-6766+Abema+Fulv in Met HR+/HER- BC

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Histologically or cytologically confirmed HR+, HER2-negative metastatic or locally recurrent unresectable invasive breast cancer
  • Measurable or non-measurable disease per RECIST v1.1
  • Men and pre- or postmenopausal women eligible; premenopausal women and men must have ongoing monthly GNRH agonist treatment for at least 4 weeks prior to study entry
  • Radiological or objective evidence of progression on any CDK4/6 inhibitor regimen in metastatic setting or relapse/progression during or within 12 months after adjuvant CDK4/6 inhibitor regimen
  • Radiological or objective evidence of progression on fulvestrant in metastatic setting
  • No more than two prior chemotherapy regimens in metastatic setting
  • No limit on prior endocrine therapy lines
  • Phase 2 participants willing to undergo pre- and on-treatment tumor biopsies unless contraindicated
  • ECOG performance status less than 2
  • Adequate organ and marrow function as defined in study criteria
  • Recovery from prior treatment toxicities to Grade 1 or better, except alopecia and peripheral neuropathy grade 2 or less
  • Age greater than 18 years
  • Women of childbearing potential, postmenopausal women via GNRH agonists, and men must agree to use adequate contraception during and after study treatment
  • Female participants of childbearing potential must have negative pregnancy test within 7 days before first dose
  • Ability to swallow and retain oral medication
  • Ability to understand and sign informed consent
Not Eligible

You will not qualify if you...

  • Active brain metastases or carcinomatous meningitis; stable, treated brain metastases allowed if meeting criteria
  • Discontinued prior abemaciclib for toxicity (phase I: any dose; phase II: at or above RP2 dose level)
  • Discontinued prior fulvestrant for toxicity
  • Prior treatment with any MEK inhibitor
  • Recent investigational agent use within 30 days or 5 half-lives
  • Chemotherapy or immunotherapy within 21 days before study drug
  • Endocrine or biologic agent within 14 days before study drug
  • Radiation therapy completed within 14 days before registration unless recovered from acute effects
  • Major surgery within 14 days before registration
  • Pre-existing ocular conditions including glaucoma, retinal vein occlusion risk factors, corneal diseases
  • History of rhabdomyolysis or neuromuscular disorders with elevated creatine kinase
  • Uncontrolled serious illnesses including certain cardiac, pulmonary, hepatic, renal, or metabolic conditions
  • History of recent second malignancy unless disease-free or low recurrence risk as specified
  • Allergic reactions to study drugs or their components
  • HIV positive with recent AIDS-defining infection or requiring certain antiretroviral therapies
  • Active hepatitis B or C infections without appropriate management
  • Recent use of strong CYP3A4 inhibitors or inducers
  • Pregnant or breastfeeding women
  • Inability to swallow oral medications or gastrointestinal conditions affecting absorption
  • Active systemic bacterial, fungal infections, or recent severe COVID-19
  • Current treatment with warfarin without appropriate anticoagulation switch
  • Other serious uncontrolled medical conditions posing high risk for toxicity per investigator judgment

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 3 locations

1

Massachusetts General Hospital Cancer Center

Boston, Massachusetts, United States, 02114

Withdrawn

2

Brigham and Women's Hospital

Boston, Massachusetts, United States, 02115

Actively Recruiting

3

Dana Farber Cancer Institite

Boston, Massachusetts, United States, 02115

Actively Recruiting

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Research Team

A

Adrienne G Waks, MD

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

2

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