Status:

COMPLETED

Safety/Effectiveness of Oral Chemokine Coreceptor 5 (CCR5) Antagonist INCB009471 in R5-tropic HIV Infected Patients

Lead Sponsor:

Incyte Corporation

Conditions:

HIV Infections

Eligibility:

All Genders

18-65 years

Phase:

PHASE2

Brief Summary

This study will evaluate the safety, pharmacokinetics and efficacy of the CCR5 antagonist INCB009471 in HIV-1 infected patients who are antiretroviral therapy naïve, or who are not currently on a HAAR...

Eligibility Criteria

Inclusion

  • Asymptomatic HIV-1 infected individuals that are treatmen naïve (ie less than 2 weeks prior ARV exposure) or treatment experienced subjects who are not currently on HAART and have not received any ARVs for 3 months prior to Screening.
  • Males between 18 years and 65 years of age, utilizing adequate contraceptive methods.
  • Post menopausal or surgically sterile females between 18 years and 65 years of age. Women of childbearing potential, utilizing adequate contraceptive methods.
  • CD4-lymphocyte count \>350 cells/mm3
  • HIV-1 RNA copies/ml \> 10,000.
  • HIV-1 is CCR5 tropic virus only.
  • CCR5 antagonist treatment naive.
  • BMI \> 16 to \< 32 kg/m2.
  • Have no clinically significant findings on screening evaluations, which in the opinion of the Investigator would interfere with the subject's ability to comply with the protocol.
  • Able to comprehend and willing to sign an Informed Consent Form.

Exclusion

  • Current or recent (\<30 days) opportunistic infection.
  • Presence of CXCR4- or dual-tropic HIV-1 virus at Screening or Baseline assessments.
  • Subjects with chronic renal insufficiency
  • Personal history of cardiac diseases.
  • History or presence of an abnormal ECG.
  • History of unstable ischemic heart disease or uncontrolled hypertension.
  • History of malignancy, with the exception of cured basal cell or squamous cell carcinoma of the skin.
  • Subjects who have received radiation therapy or cytotoxic chemotherapeutic agents and have not recovered from side effects.
  • Current treatment or treatment within 30 days or 5 half-lives with another investigational medication or current enrollment in another investigational drug protocol.
  • Subjects with unstable medical condition (s), which , in the opinion of the Investigator would compromise their participation in the trial

Key Trial Info

Start Date :

October 1 2006

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

September 1 2007

Estimated Enrollment :

45 Patients enrolled

Trial Details

Trial ID

NCT00393120

Start Date

October 1 2006

End Date

September 1 2007

Last Update

March 26 2018

Active Locations (6)

Enter a location and click search to find clinical trials sorted by distance.

Page 1 of 2 (6 locations)

1

Los Angeles, California, United States, 90069

2

Washington D.C., District of Columbia, United States, 20007

3

Orlando, Florida, United States, 32803

4

Vero Beach, Florida, United States, 32960