Status:

COMPLETED

A Study to Assess CH1504 in Patients With Active Rheumatoid Arthritis

Lead Sponsor:

Chelsea Therapeutics

Conditions:

Arthritis, Rheumatoid

Eligibility:

All Genders

18-80 years

Phase:

PHASE2

Brief Summary

The purpose of this trial is to assess the clinical effect of CH-1504 at doses of 0.25, 0.5 and 1.0 mg per day in patients with active rheumatoid arthritis by determining the proportion of patients ac...

Detailed Description

Rheumatoid Arthritis (RA) is a chronic inflammatory disease of unknown cause that leads to pain, stiffness, swelling and limitation of joint function. If left untreated, RA produces serious destructio...

Eligibility Criteria

Inclusion

  • Inclusion; To be eligible for inclusion, each patient must fulfill the following criteria:
  • Patients must be between the ages of 18 and 80;
  • Have been diagnosed with active rheumatoid arthritis according to ACR criteria;
  • Have at least 6 swollen joints (max = 66) and 6 tender joints (max = 68) at screening and baseline visits;
  • Patients must have at least one of the following:
  • C-reactive protein \> 1.0 mg/dl at screening;
  • erythrocyte sedimentation rate \> 20 mm/Hr;
  • Morning stiffness \> 45 min. at screening;
  • Patients must have blood test values per the following criteria:
  • ALT, AST \< 1.2 U/l x ULN
  • Albumin \> 2.5 g/dl
  • Prothrombin Time \< 1.2 INR
  • Hb \> 9.0 g/dl
  • Hct \> 35%
  • WBC \> 3000 μl (mm3)
  • Neutrophils \> 1000 μl (mm3)
  • Platelets \> 100000 μl
  • Creatinine \< 1.2 mg/dl
  • Patients must have voluntarily signed the informed consent
  • Exclusion; Patients are not eligible for this study if they fulfill one or more of the following criteria:
  • Patients who received previous methotrexate therapy;
  • Patients who received previous therapy with any biologic agent;
  • Previous biologic therapy for a disease other than RA is permitted so long as their last dose was more than 120 days prior to baseline;
  • Patients currently taking sulfasalazine;
  • Previous sulfasalazine therapy is permitted so long as their last dose was more than 30 days prior to baseline;
  • Patients currently taking hydroxychloroquine;
  • Previous hydroxychloroquine is permitted so long as their last dose was more than 120 days prior to baseline;
  • Female patients of child bearing potential who are pregnant or who are not using two methods of contraception (at least one barrier: i.e. condom) with their partner;
  • Male patients who are sexually active and not using two methods of contraception (at least one barrier: i.e. condom) with their partner;
  • Patients with any current active infection or infections requiring IV drug therapy within 30 days of baseline or oral therapy within 15 days of Baseline;
  • Patients that have had any surgical procedures within 30 days of baseline;
  • Patients with a history of HIV, Hepatitis B or C;
  • Patients who consume more than 7 units of alcohol per week (1 unit = 5 ounces/150 ml of wine = 1.5 ounces/45 ml spirits = 12 ounces/360 ml of beer);
  • Patients currently receiving any investigational drug or have received an investigational drug within 30 days of baseline or 5 half-lives of the investigational drug (whichever is longer);
  • Patients with a history of cancer within the past 5 years other than a successfully treated, non-metastatic cutaneous squamous cell or basal cell carcinoma or cervical cancer in situ;
  • Patients with a history of, or any, disease associated with an inflammatory arthritis other than RA;
  • Patients with a chest X-ray that indicates the presence of pulmonary fibrosis (Chest x-ray may be taken with in 28 days of screening);
  • Patients receiving Probenecid;
  • Patients who have received any steroid injections within 30 days of baseline;
  • Patients with concomitant diseases that are unstable (i.e. cardiac, pulmonary) or that may affect drug activity (i.e. absorption, reactions, change in kinetics);
  • Patients considered by the investigator to be an unsuitable candidate to receive CH-1504;
  • Wheelchair or bed-bound patients.

Exclusion

    Key Trial Info

    Start Date :

    April 1 2008

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    June 1 2009

    Estimated Enrollment :

    201 Patients enrolled

    Trial Details

    Trial ID

    NCT00658047

    Start Date

    April 1 2008

    End Date

    June 1 2009

    Last Update

    April 15 2013

    Active Locations (1)

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    Page 1 of 1 (1 locations)

    1

    The Rebecca MacDonald Centre for Arthritis and Autoimmune Disease

    Toronto, Ontario, Canada, M5G 1X5