Status:

COMPLETED

A First Time In Human Study to Evaluate the Safety, Tolerability and Pharmacokinetics of GSK1399686

Lead Sponsor:

GlaxoSmithKline

Conditions:

Inflammatory Bowel Diseases

Eligibility:

All Genders

18-65 years

Phase:

PHASE1

Brief Summary

A First-Time-in-Human Study to Evaluate the Safety, Tolerability and Pharmacokinetics of GSK1399686 After Single and Repeated Oral Dosing in Healthy Volunteers

Eligibility Criteria

Inclusion

  • Inclusion criteria:
  • Healthy as determined by a responsible physician
  • Male, or only for the RDF cohort female of non-childbearing potential, between 18 and 65 years of age.
  • Body weight greater than 50 kg (110 lbs) and BMI within the range 18.5-29.9 kg/m2 (inclusive).
  • QTcB or QTcF \< 450 msec
  • Capable of giving written informed consent
  • Exclusion criteria:
  • The subject has a positive pre-study drug/alcohol screen
  • History of regular alcohol consumption within 6 months of the study defined as an average weekly intake of greater than 21 units
  • Urinary cotinine levels indicative of active smoking or regular use of tobacco
  • A positive pre-study Hepatitis B surface antigen or positive Hepatitis C antibody
  • A positive test for HIV antibody
  • The subject has participated in a clinical trial and has received an investigational product within 30 days, 5 half-lives of the investigational product
  • Exposure to more than four new chemical entities within 12 months
  • Use of prescription or non-prescription drugs, including vitamins, herbal and dietary supplements (including St John's Wort) within 7 days
  • Consumption of red wine, seville oranges, grapefruit or grapefruit juice and/or pummelos, exotic citrus fruits, grapefruit hybrids or fruit juices within 7 days
  • Subject is receiving hormone replacement therapy
  • History of sensitivity to any of the study medications
  • History of sensitivity to heparin or heparin-induced thrombocytopenia

Exclusion

    Key Trial Info

    Start Date :

    September 25 2008

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    May 27 2009

    Estimated Enrollment :

    87 Patients enrolled

    Trial Details

    Trial ID

    NCT00721812

    Start Date

    September 25 2008

    End Date

    May 27 2009

    Last Update

    July 7 2017

    Active Locations (1)

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    Page 1 of 1 (1 locations)

    1

    GSK Investigational Site

    Harrow, Middlesex, United Kingdom, HA1 3UJ