Status:

COMPLETED

Effects of Telbivudine and Tenofovir Disproxil Fumarate on the Kinetics of Hepatitis B Virus DNA in Chronic Hepatitis B (CHB)

Lead Sponsor:

The University of Hong Kong

Collaborating Sponsors:

Novartis Pharmaceuticals

Conditions:

Chronic Hepatitis B

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

The purpose of this study is to compare the safety, tolerability and effectiveness of 12 weeks of treatment with telbivudine 600 mg daily plus tenofovir DF 300 mg once daily (QD) taken together versus...

Detailed Description

The primary goal of therapy for chronic hepatitis B (CHB) is suppression of viral replication. Long-term suppression of serum HBV DNA is likely to reduce progression to cirrhosis and hepatic decompens...

Eligibility Criteria

Inclusion

  • Patients must meet all of the following inclusion criteria at screening to be eligible for participation in this study.
  • Chronic HBV infection, defined as positive serum HBsAg for at least 6 months, or HBsAg positive \> 3 months and negative for IgM anti-HBc and positive for IgG anti-HBc
  • Age \< 40 years old
  • HBeAg positive
  • HBV DNA ≥ 10\^7 copies/mL by Abbott real-time PCR
  • ALT ≤ 1 ULN
  • Willing and able to provide written informed consent
  • Negative serum β-HCG (for females of childbearing potential only)
  • Calculated creatinine clearance ≥ 70 mL/min by the following formula: (140 - age in years) x (body weight \[kg\]) / (72) x (serum creatinine \[mg/dl\]) \[Note: multiply estimated rate by 0.85 for women\]
  • Hemoglobin ≥ 10 g/dL
  • Neutrophils ≥ 1,500 /mm\^3
  • No prior oral HBV therapy (e.g., nucleotide and/or nucleoside therapy or other investigational agents for HBV infection)
  • Is willing and able to comply with the study drug regimen and all other study procedures and requirements
  • Is willing and able to provide written informed consent before any study assessment is perform.

Exclusion

  • Patients will be excluded from the study for any of the criteria:
  • Decompensated liver disease defined as direct (conjugated) bilirubin \> 1.2 × ULN, PT \> 1.2 × ULN, platelets \< 150,000/mm3, serum albumin \< 3.5 g/dL, or prior history of clinical hepatic decompensation (e.g. ascites, jaundice, encephalopathy, variceal hemorrhage).
  • Received interferon (pegylated or not) therapy within 6 months of the screening visit
  • α-fetoprotein \> 50 ng/mL
  • Evidence of hepatocellular carcinoma (HCC)
  • Co-infection with HCV (by serology), HIV, or HDV.
  • Significant renal, cardiovascular, pulmonary, or neurological disease.
  • Received solid organ or bone marrow transplantation.
  • Is currently receiving therapy with immunomodulators (e.g., corticosteroids, etc.), investigational agents, nephrotoxic agents, or agents susceptible of modifying renal excretion.
  • Has proximal tubulopathy.
  • Use of other investigational drugs at the time of enrollment, or within 30 days
  • History of hypersensitivity to any of the study drugs or to drugs of similar chemical classes
  • Is pregnant or breastfeeding. Women of childbearing potential must have a negative serum β - HCG during Screening.
  • Is a women of child-bearing potential (WOCBP), defined as all women physiologically capable of becoming pregnant, including women whose career, lifestyle, or sexual orientation precludes intercourse with a male partner and women whose partners have been sterilized by vasectomy or other means, UNLESS they meet the following definition of post-menopausal: 12 months of natural (spontaneous) amenorrhea or 6 months of spontaneous amenorrhea with serum FSH levels \>40 mIU/m or 6 weeks post surgical bilateral oophorectomy with or without hysterectomy OR are using one or more of the following acceptable methods of contraception: surgical sterilization (e.g., bilateral tubal ligation, vasectomy), hormonal contraception (implantable, patch, oral), and double-barrier methods (any double combination of: IUD, male or female condom with spermicidal gel, diaphragm, sponge, cervical cap).
  • Patient has any other concurrent medical or social condition likely to preclude compliance with the schedule of evaluations in the protocol, or likely to confound the efficacy or safety observations of the study.
  • Patient is currently abusing alcohol or illicit drugs, or has a history of alcohol abuse or illicit substance abuse within the preceding two years. Please refer to Appendix 3.
  • Patient has a medical condition that requires prolonged or frequent use of systemic acyclovir or famciclovir. Please refer to Appendix 1.

Key Trial Info

Start Date :

December 1 2008

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

March 1 2010

Estimated Enrollment :

15 Patients enrolled

Trial Details

Trial ID

NCT00804622

Start Date

December 1 2008

End Date

March 1 2010

Last Update

July 11 2012

Active Locations (1)

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1

Department of Medicine, Queen Mary Hospital

Hong Kong, China