Status:

TERMINATED

TC-5214 as Augmentation Therapy in Patients With Refractory Hypertension

Lead Sponsor:

Targacept Inc.

Conditions:

Refractory Hypertension

Eligibility:

All Genders

18-65 years

Phase:

PHASE1

PHASE2

Brief Summary

A pilot study of subjects with refractory hypertension (on 3 concomitant agents with SBP \> 140 mmHg and a DBP \> 90 mmHg) randomized in a double-blind fashion to receive 4 single escalating doses of ...

Detailed Description

12 subjects with refractory hypertension will be randomized in a double-blind fashion to receive single escalating doses of study medication in-clinic: on Day 1 (1mg), Day 8 (2mg), Day 15 (4mg) and Da...

Eligibility Criteria

Inclusion

  • Refractory hypertension, defined as a SBP of \>140mmHg and a DBP \> 90mmHg, on stable doses of at least 3 concomitant antihypertensive treatment (which must include a diuretic and an ACEI, ARB or RA) for 8 weeks prior to Screening. All approved antihypertensive treatments are allowed except for alpha-adrenergic blockers, hydralazine, clonidine, guanethidine, guanadrel, and rauwolfia alkaloids.
  • Stable hypertension, as defined by: a. mean SBP on Day -7 that is within 20mmHg of the mean SBP on Day 1, with both mean SBPs \> 140mmHg; and b. mean DBP on Day -7 that is within 10mm of the mean DBP on Day 1, with both mean DBPs \> 90mmHg.
  • Outpatient with stable housing.
  • Subjects must be able to stay in the clinic for 8 hrs on Day 1, Day 8, Day 15, Day 22, and Day 36.
  • Able to give and to sign informed consent.

Exclusion

  • Any unstable medical condition other than hypertension;
  • Stage 3 hypertension (SBP \> 180mmHg and/or DBP \> 110mmHg);
  • Heart rate \> 100 beats per minute;
  • WOCBP who is pregnant or who is planning to become pregnant during the study;
  • History within past year of alcohol or illicit drug abuse;
  • Unable to comply with study procedures in opinion of investigator;
  • Concomitant medications for any medical condition that is uncontrolled for more than 2 weeks prior to study entry;
  • Current use of alpha-adrenergic blocker, hydralazine, clonidine, guanethidine, guanadrel, or rauwolfia alkaloids;
  • History of myocardial infarction or angina pectoris;
  • Current seizure disorder;
  • Renal insufficiency as defined by a serum creatinine \> 2.0;
  • Uncontrolled hypothyroidism, vitamin B12 or folic acid deficiency;
  • History of or concurrent ileus, glaucoma, or urinary retention;
  • Inability of subject to understand and sign the ICF;
  • Known systemic infection (HBV, HCV, HIV, TB);
  • Current use of smoking cessation therapy within 4 weeks of screening;
  • Use of herbal supplements;
  • Clinically significant finding on physical exam;
  • Clinically significant laboratory or ECG abnormality, including QTcF \> 460 msec;
  • Participation in another clinical trial in last month;
  • Body Mass Index (BMI) \> 35.
  • Body weight \< 100 pounds.
  • Site staff or family member of study site staff.

Key Trial Info

Start Date :

May 1 2009

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

December 1 2009

Estimated Enrollment :

1 Patients enrolled

Trial Details

Trial ID

NCT00899977

Start Date

May 1 2009

End Date

December 1 2009

Last Update

September 13 2013

Active Locations (1)

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Page 1 of 1 (1 locations)

1

Piedmont Medical Research

Winston-Salem, North Carolina, United States, 27101

TC-5214 as Augmentation Therapy in Patients With Refractory Hypertension | DecenTrialz