Status:

COMPLETED

Pharmacokinetics of AP214 Acetate in Patients Undergoing Cardiac Surgery

Lead Sponsor:

Action Pharma A/S

Conditions:

Cardiac Surgery

Coronary Artery Bypass Grafting

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

The purpose of the present research study is to investigate the pharmacokinetics, as well as safety, tolerability and pharmacodynamics of different ascending dosing regimens of AP214 in patients under...

Eligibility Criteria

Inclusion

  • Has signed the trial-specific informed consent form.
  • Patients ≥ 18 years old, male or female, not of childbearing potential (postmenopausal or permanently sterilized, e.g. tubal ligation, hysterectomy, bilateral salpingectomy), regardless of ethnicity.
  • Patients undergoing CABG, valve(s), CABG/valve(s) and/or aortic root or ascending aortic aneurysm repair surgery.
  • Cleveland Clinic Renal Score ≥ 2 (higher than average risk for AKI).
  • EF ≥ 30%, evaluated within 2 months prior to screening visit.

Exclusion

  • Cardiac surgery to be performed "off pump" without cardiopulmonary bypass.
  • Circulatory arrest in connection with aortic root or ascending aortic aneurysm repair surgery.
  • Confirmed or suspected endocarditis.
  • Requiring a reoperation on one of the valves within 3 months following the original valve surgical procedure.
  • Receiving Aprotinin during the trial, from Screening to Day 90.
  • Having undergone cardiovascular catheterization ≤ 48 hours prior to scheduled surgery.
  • Active peptic ulcer disease and gastritis.
  • Hemoccult positive stools, hematological, bleeding, and coagulation disorders.
  • Receiving dopamine at renal doses (2-4 mcg/kg/min), from Screening to Day of surgery.
  • S-Creatinine greater than 2.1 mg/dl.
  • Known or suspected hypersensitivity to the investigational medicinal product.
  • Known or suspected hypersensitivity to Ondansetron or other selective 5-hydroxytryptamine 3 (5-HT3) receptor antagonists.
  • Current participation in any other interventional clinical trial.
  • Previously dosed with AP214.
  • Use of investigational medicinal products within the previous 6 months.
  • Body weight above 140 kg.
  • History of any organ transplant.
  • Women who are of childbearing potential, pregnant, or breast-feeding.
  • Current abuse of alcohol or substance, according to the investigator's medical judgment.
  • Has a mental incapacity or language barriers precluding adequate understanding of trial procedures.
  • Is considered by the Investigator unsuitable to participate in the trial for any other reason, for instance due to a significant serious underlying condition.

Key Trial Info

Start Date :

May 1 2009

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

June 1 2010

Estimated Enrollment :

42 Patients enrolled

Trial Details

Trial ID

NCT00903604

Start Date

May 1 2009

End Date

June 1 2010

Last Update

May 17 2011

Active Locations (2)

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Page 1 of 1 (2 locations)

1

Department of Cardiac and Thoracic Surgery, Copenhagen University Hospital, Rigshospitalet

Copenhagen, Denmark, 2100

2

Odense University Hospital, Department of Cardiac, Thoracic and Vascular Surgery

Odense, Denmark, 5000