Status:

COMPLETED

A Study of ARRY-438162 (MEK162) in Patients With Advanced Cancer

Lead Sponsor:

Array Biopharma, now a wholly owned subsidiary of Pfizer

Conditions:

Advanced Solid Tumors

Advanced or Metastatic Biliary Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

This is a Phase 1 study during which patients with advanced solid tumors will receive investigational study drug ARRY-438162 (MEK162). This study has 3 parts. In the first part, patients with advance...

Eligibility Criteria

Inclusion

  • Key Inclusion Criteria (for Part 3):
  • A histologically or cytologically confirmed diagnosis of colorectal adenocarcinoma which is metastatic (measurable disease).
  • Documented KRAS- or BRAF- tumor mutation.
  • Previously treated with or unsuitable for treatment with 5-Fluorouracil (5-FU), oxaliplatin, irinotecan and, if available, bevacizumab.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0, 1 or 2.
  • Additional criteria exist.
  • Key Exclusion Criteria (for Part 3):
  • Uncontrolled or symptomatic brain metastases (if the patient has brain metastases and is on steroids, the steroid dose must have been stable for at least 30 days).
  • History of central serous retinopathy, retinopathy visible at baseline that would be considered a risk factor for central serous retinopathy or retinal vein occlusion.
  • Concomitant malignancies or previous malignancies with less than a 2-year disease free interval at the time of enrollment; patients with adequately resected basal or squamous cell carcinoma of the skin, carcinoma in situ of the cervix, or stage A low grade prostate cancer may enroll irrespective of the time of diagnosis.
  • Prior treatment with a MEK inhibitor.
  • Treatment with prior chemotherapy, anticancer immunotherapy, monoclonal antibodies or other protein or peptide therapeutics within 21 days of the first dose of study drug.
  • Treatment with a small molecule targeted agent or anticancer hormonal therapy within 14 days of the first dose of study drug.
  • Treatment with prior radiotherapy within 28 days of initiating study drug (if the radiation portal covered ≤ 10% of the bone marrow reserve, the patient may be enrolled irrespective of the end date of radiotherapy).
  • Major surgery within 4 weeks or minor surgery within 7 days prior to the first dose of study drug.
  • Known positive serology for the human immunodeficiency virus (HIV), hepatitis C, and/or active hepatitis B.
  • Additional criteria exist.

Exclusion

    Key Trial Info

    Start Date :

    August 1 2009

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    January 1 2013

    Estimated Enrollment :

    93 Patients enrolled

    Trial Details

    Trial ID

    NCT00959127

    Start Date

    August 1 2009

    End Date

    January 1 2013

    Last Update

    September 16 2020

    Active Locations (10)

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    Page 1 of 3 (10 locations)

    1

    University of California, Los Angeles

    Los Angeles, California, United States, 90095

    2

    University of Colorado Cancer Center

    Aurora, Colorado, United States, 80045

    3

    The Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins

    Baltimore, Maryland, United States, 21231-1000

    4

    Dana-Farber/Harvard Cancer Center

    Boston, Massachusetts, United States, 02114

    A Study of ARRY-438162 (MEK162) in Patients With Advanced Cancer | DecenTrialz