Status:

TERMINATED

Trial of Dasatinib in Patients With Advanced Cancers Harboring DDR2 Mutation or Inactivating B-RAF Mutation

Lead Sponsor:

Bristol-Myers Squibb

Conditions:

Carcinoma, Non-small Cell Lung

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

The purpose of this study is to establish whether patients with malignancy harboring a discoidin domain receptor 2 mutation or an inactivating B-RAF mutation will respond to dasatinib.

Eligibility Criteria

Inclusion

  • For more information regarding BMS clinical trial participation, please visit www.BMSStudyConnect.com.
  • Inclusion Criteria
  • Diagnosis of advanced malignancy, nonsmall-cell lung cancer (NSCLC) only during stage 1 of accrual.
  • Nonsynonymous mutation of B-RAF or DDR2, defined as follows:.
  • i) NSCLC with inactivating B-RAF mutation.
  • ii) NSCLC with discoidin domain receptor 2 (DDR2) mutation.
  • iii) Malignancy of other histology with DDR2 mutation or inactivating B-RAF mutation, or NSCLC having a B-RAF mutation that is not functionally characterized.
  • At least 1 target lesion per Response Evaluation Criteria in Solid Tumors, vol 1.1, on baseline staging evaluation.
  • Disease progression after ≥ 1 prior treatment regimen.
  • Exclusion Criteria
  • Pleural or pericardial effusion, Grade \>1.
  • QTcF \>470 msec (Grade ≥2) or diagnosed congenital long QT syndrome.
  • Absolute granulocyte count \<1500/mm\^3.
  • Hemoglobin level \<10 g/dL.
  • Platelet count \< 75,000/mm\^3.
  • Serum calcium level \<institutional lower limit of normal.
  • Hypokalemia, hypophosphatemia, or hypomagnesemia, Grade \>1, despite supplementation.
  • Creatinine \>3\*institutional upper limit of normal (ULN).
  • Total bilirubin level \>1.5\*ULN.
  • Alanine transaminase level \>3\*ULN.
  • Other protocol-defined Inclusion/Exclusion criteria apply.

Exclusion

    Key Trial Info

    Start Date :

    May 31 2012

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    July 23 2014

    Estimated Enrollment :

    19 Patients enrolled

    Trial Details

    Trial ID

    NCT01514864

    Start Date

    May 31 2012

    End Date

    July 23 2014

    Last Update

    December 19 2023

    Active Locations (24)

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    Page 1 of 6 (24 locations)

    1

    H. Lee Moffitt Cancer & Research Institute

    Tampa, Florida, United States, 33612

    2

    Memorial Sloan Kettering Cancer Center

    New York, New York, United States, 10065

    3

    Memorial Sloan Kettering Nassau

    New York, New York, United States, 10065

    4

    Local Institution

    Barretos, São Paulo, Brazil, 14784-400

    Trial of Dasatinib in Patients With Advanced Cancers Harboring DDR2 Mutation or Inactivating B-RAF Mutation | DecenTrialz