Status:

TERMINATED

A Trial of 18F-AV-133 Positron Emission Tomography (PET)

Lead Sponsor:

Avid Radiopharmaceuticals

Conditions:

Type 1 Diabetes

Type 2 Diabetes

Eligibility:

All Genders

18-70 years

Phase:

PHASE1

Brief Summary

The purpose of this study is to evaluate the safety and pancreas imaging properties of 18F-AV-133.

Detailed Description

The primary objective of this protocol is to address the feasibility for further development of the VMAT2-binding compound 18F-AV-133 as a diagnostic radiopharmaceutical in the field of diabetes. Spec...

Eligibility Criteria

Inclusion

  • Patients with type 1 diabetes may be enrolled if they meet all of the following criteria:
  • Are males or females between 18 and 70 years of age, inclusive;
  • Have a diagnosis of type 1 diabetes mellitus as defined by ADA criteria; diabetes onset younger than age 21, duration \>5 years; Insulin dose requirements ≤ 0.8 units/kg/day;
  • HbA1c level ≥ 5% and ≤ 8%;
  • Have fasting C-Peptide \< 0.1 ng/ml;
  • Have a BMI between 18 and 32 kg/m2;
  • Able to tolerate PET imaging;
  • In the judgment of the physician, are capable of fasting 4-6 hours prior to screening and Day 1 imaging procedures; and
  • Give informed consent.
  • Patients with type 2 diabetes may be enrolled if they meet all of the following criteria:
  • Are males or females between 18 and 70 years of age, inclusive;
  • Must have been diagnosed with type 2 diabetes for more than five years;
  • HbA1c level ≥ 5% and ≤ 8%;
  • Have a BMI between 18 and 32 kg/m2;
  • Glucose \> 200 mg/dl on Mixed Meal Tolerance Test at screening visit;
  • Able to tolerate PET imaging;
  • In the judgment of the physician, are capable of fasting 4-6 hours prior to screening and Day 1 imaging procedures; and
  • Give informed consent.
  • Healthy volunteers may be enrolled if they meet all of the following criteria:
  • Are males or females between 18 and 70 years of age, inclusive;
  • Have no history of type 1 or type 2 diabetes in a first degree relative;
  • Fasting blood glucose ≤ 100 mg/dL;
  • HbA1c level ≤ 6%;
  • Normal Mixed Meal Tolerance test at screening visit;
  • BMI between 18 and 32 kg/m2;
  • Able to tolerate PET imaging;
  • In the judgment of the physician, are capable of fasting 4-6 hours prior to screening and Day 1 imaging procedures; and
  • Give informed consent.
  • Subjects will be excluded from enrollment if they meet any of the following criteria:
  • Clinically significant renal dysfunction;
  • Clinically significant liver dysfunction as determined by history, physical examination, and standard liver function testing at screening (AST, ALT, Total/Direct Bilirubin, Alkaline Phosphatase);
  • Coagulopathy;
  • Use medications known to affect dopaminergic function, including MAO inhibitors, tetrabenazine, or levodopa;
  • Recent (within 3 months) or current treatment with drugs influencing beta cell function or insulin sensitivity (e.g. glucocorticoids, reserpine);
  • Have polycystic ovarian syndrome;
  • History of movement disorder such as Parkinson's Disease, Huntington's Disease;
  • Clinically significant psychiatric disease or history of psychiatric illness such as depression, bipolar disease, anxiety or schizophrenia;
  • Current use (within past year) of cocaine, methamphetamine, and/or ecstasy ( MDMA, 34- methylenedioxymethamphetamine;
  • Have a recent history of alcohol or substance abuse or dependence;
  • Clinically significant cardiovascular disease or clinically significant abnormalities on screening ECG (including but not limited to QTc\>450 msec);
  • Clinically significant pulmonary, renal or hepatic impairment, or cancer;
  • Have clinically significant infectious disease, including AIDS or HIV infection or previous positive test for hepatitis B, hepatitis C, HIV-1, or HIV-2;
  • Are women of childbearing potential who are not surgically sterile, not refraining from sexual activity or not using adequate contraception. Women must not be pregnant (negative serum β-HCG at the time of screen) or breastfeeding at screening, and must agree to take appropriate steps not to become pregnant for 30 days following the clinical trial;
  • Require medications with a narrow therapeutic window (e.g., warfarin), are receiving any investigational medications, or have participated in a trial with investigational medications within the last 30 days;
  • Weigh more than the manufacturer-recommended limit for the PET/CT camera being used;
  • Any prior participation in other research protocols within the past month that involved radiation, with the exception of plain radiography studies (i.e., chest x-rays); and
  • Have received a diagnostic or therapeutic radiopharmaceutical within the past week.

Exclusion

    Key Trial Info

    Start Date :

    June 1 2010

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    February 1 2013

    Estimated Enrollment :

    19 Patients enrolled

    Trial Details

    Trial ID

    NCT01515384

    Start Date

    June 1 2010

    End Date

    February 1 2013

    Last Update

    January 13 2020

    Active Locations (1)

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    Page 1 of 1 (1 locations)

    1

    Research Site

    New York, New York, United States, 10027