Status:

TERMINATED

Orteronel in Treating Patients With Metastatic Hormone-Resistant Prostate Cancer

Lead Sponsor:

University of Southern California

Collaborating Sponsors:

National Cancer Institute (NCI)

Millennium Pharmaceuticals, Inc.

Conditions:

Adenocarcinoma of the Prostate

Hormone-resistant Prostate Cancer

Eligibility:

MALE

18+ years

Phase:

PHASE2

Brief Summary

This phase II trial studies how well orteronel works in treating patients with metastatic hormone-resistant prostate cancer. Orteronel may stop the growth of tumor cells by blocking some of the enzyme...

Detailed Description

PRIMARY OBJECTIVES: I. To assess the relationship between circulating tumor cell (CTC)-based androgen receptor (AR) expression level and \>=-50% prostate-specific antigen (PSA) decline following 12 w...

Eligibility Criteria

Inclusion

  • Histologically confirmed adenocarcinoma of the prostate
  • Voluntary written informed consent before performance of any study-related procedure not part of normal medical care, with the understanding that consent may be withdrawn by the subject at any time without prejudice to future medical care
  • Patients, even if surgically sterilized (i.e., status post vasectomy), who agree to practice effective barrier contraception during the entire study treatment period and for 4 months after the last dose of study drug, or
  • Agree to completely abstain from intercourse
  • Serum alanine aminotransferase (ALT) and aspartate aminotransferase (AST) must be =\< 2.5 x the upper limit of normal (ULN)
  • Total bilirubin =\< 1.5 x ULN
  • Estimated creatinine clearance using the Cockcroft-Gault formula must be \> 40 mL/minute
  • Absolute neutrophil count (ANC) \>= 1500 cells/microliter
  • Platelet count \>= 100,000 cells/microliter
  • Testosterone \< 50 ng/dL
  • Screening calculated ejection fraction of \>= 50% by multiple gated acquisition (MUGA) scan or echocardiogram; metastatic progression on primary androgen-deprivation therapy (medical or surgical castration)
  • Progression requiring a change in oncologic therapy defined by any of the following:
  • Radiographic progression: appearance or increase in measurable lesions on cross-sectional imaging or appearance of one or more new lesions on bone scan \* Rising PSA (\>= 2 ng/ml) which has risen on two occasions \>= 1 week apart
  • Clinical progression evidenced by increased pain or other cancer-related symptoms
  • Patients should have recovered from prior oncologic therapies to a Common Terminology Criteria (CTC) grade =\< 1 except stable neuropathy or alopecia at National Cancer Institute (NCI) Common Terminology Criteria for Adverse Events (CTCAE) grade =\< 2; if rapid clinical progression is documented by imaging, changes in PSA, or symptoms, then study treatment can begin \>= 2 weeks from prior therapy; otherwise, the following time periods between prior anti-cancer therapies and study treatment day 1 will apply:
  • \>= 3 weeks for prior cytotoxic therapies
  • \>= 4 weeks for flutamide or nilutamide
  • \>= 6 weeks for bicalutamide
  • \>= 6 weeks since bone targeted radiopharmaceutical (e.g. samarium-153, radium-223)
  • Gonadotropin-releasing hormone (GnRH) agonists (leuprolide acetate, goserelin, etc.) or antagonists (degarelix, etc.) should be continued in patients without surgically-induced castrate androgen levels
  • For chemotherapy naïve castration-resistant prostate cancer who are moderately symptomatic or who have hepatic metastasis: subjects must not be a candidate for docetaxel-based chemotherapy.

Exclusion

  • History of myocardial infarction, unstable symptomatic ischemic heart disease, ongoing arrhythmias of grade \> 2 (NCI CTCAE, version 4), thromboembolic events (e.g., deep vein thrombosis, pulmonary embolism, or symptomatic cerebrovascular events), or any other cardiac condition (e.g. pericardial effusion, restrictive cardiomyopathy) within 6 months prior to first dose of study drug; chronic stable atrial fibrillation on stable anticoagulant therapy is allowed
  • New York Heart Association class III or IV heart failure
  • Electrocardiogram (ECG) abnormalities of:
  • Q-wave infarction, unless identified 6 or more months prior to screening
  • Corrected QT (QTc) interval \> 460 msec
  • Patient has received other investigational drugs within 28 days before enrollment
  • Diagnosed or treated for another malignancy within 2 years of enrollment, with the exception of complete resection of basal cell carcinoma or squamous cell carcinoma of the skin, an in situ malignancy
  • Known hypersensitivity to compounds related to TAK-700 or to TAK-700 excipients
  • Uncontrolled hypertension despite appropriate medical therapy (blood pressure \[BP\] of greater than 160 mmHg systolic and 90 mmHg diastolic at 2 separate measurements no more than 60 minutes apart during the screening visit); Note: patients may be rescreened after adjustment of antihypertensive medications
  • Known active chronic hepatitis B or C, life-threatening illness unrelated to cancer, or any serious medical or psychiatric illness that could, in the investigator's opinion, potentially interfere with participation in this study
  • Likely inability to comply with the protocol or cooperate fully with the investigator and site personnel
  • Known gastrointestinal (GI) disease or GI procedure that could interfere with the GI absorption or tolerance of TAK-700, including difficulty swallowing tablets
  • Prior treatment with \>= 3 lines of cytotoxic chemotherapy for metastatic prostate cancer
  • Prior treatment with TAK-700

Key Trial Info

Start Date :

October 25 2013

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

July 26 2016

Estimated Enrollment :

4 Patients enrolled

Trial Details

Trial ID

NCT01866423

Start Date

October 25 2013

End Date

July 26 2016

Last Update

August 31 2017

Active Locations (1)

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USC Norris Comprehensive Cancer Center

Los Angeles, California, United States, 90033