Status:

ACTIVE_NOT_RECRUITING

Study of LEE011, BYL719 and Letrozole in Advanced ER+ Breast Cancer

Lead Sponsor:

Novartis Pharmaceuticals

Conditions:

Breast Cancer

Eligibility:

FEMALE

18-100 years

Phase:

PHASE1

PHASE2

Brief Summary

The purpose of this trial is to inform the future clinical development of the two investigational agents in ER+ breast cancer, LEE011 (CDK4/6 inhibitor) and BYL719 (PI3K-alpha inhibitor). This is a m...

Eligibility Criteria

Inclusion

  • Postmenopausal, Estrogen-receptor positive and/or Progesterone-receptor positive breast cancer
  • Phase Ib dose escalation only: Any number of prior lines of endocrine therapy is allowed with the exception of cytotoxic therapy which is limited to one prior line administered in the advanced (metastatic or locally advanced) setting.
  • Phase Ib dose expansions Arms 1, 2 and 3
  • No prior systemic treatment in the advanced (metastatic or locally advanced) setting with the exception of treatment with letrozole for a maximum of one month prior to starting study treatment.
  • Patients who received (neo)adjuvant therapy for breast cancer are eligible. Prior therapy with letrozole or anastrozole in the (neo)adjuvant setting is permitted if the disease-free interval is greater than 12 months from the completion of treatment.

Exclusion

  • HER2-overexpression in the patient's tumor tissue
  • Patients with active CNS or other brain metastases
  • Major surgery within 2 weeks
  • Acute or chronic pancreatitis
  • Bilateral diffuse lymphangitic carcinomatosis
  • Another malignancy within 3 years
  • Receiving hormone replacement therapy that cannot be discontinued
  • Impaired cardiac function
  • Patients with clinically manifest diabetes mellitus (treated and/or clinical signs or with fasting glucose ≥ 126 mg/dL / 7.0 mmol/L or hemoglobin A1c \>6.5%), history of gestational diabetes mellitus or documented steroid-induced diabetes mellitus.
  • Other protocol-defined inclusion/exclusion criteria may apply

Key Trial Info

Start Date :

October 22 2013

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

February 26 2027

Estimated Enrollment :

255 Patients enrolled

Trial Details

Trial ID

NCT01872260

Start Date

October 22 2013

End Date

February 26 2027

Last Update

October 29 2025

Active Locations (25)

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Page 1 of 7 (25 locations)

1

Univ of California at San Diego Moores Cancer Ctr

San Diego, California, United States, 92103

2

UCSF Medical Center

San Francisco, California, United States, 94143

3

H Lee Moffitt Cancer Center and Research Institute

Tampa, Florida, United States, 33612

4

Massachusetts General Hospital SC-5

Boston, Massachusetts, United States, 02114

Study of LEE011, BYL719 and Letrozole in Advanced ER+ Breast Cancer | DecenTrialz