Status:

COMPLETED

Study to Evaluate the Pharmacokinetics, Tolerability, and Safety of ACT-128800 in Japanese and Caucasian Healthy Male and Female Subjects

Lead Sponsor:

Actelion

Conditions:

Healthy

Eligibility:

All Genders

18-45 years

Phase:

PHASE1

Brief Summary

This is a study to evaluate the relative pharmacokinetic properties and the tolerability and safety of ACT-128800 in Japanese and Caucasian healthy male and female subjects after single-dose administr...

Detailed Description

10 Japanese and 10 Caucasian healthy male and female subjects in a one to one male to female ratio will be included in the study. Japanese and Caucasian subjects will be matched for body weight.

Eligibility Criteria

Inclusion

  • Signed informed consent prior to any study-mandated procedure.
  • Japanese or Caucasian. (Japanese subjects: both parents of the subject are Japanese \[born in Japan\]. Caucasian subjects: both parents of the subject are Caucasian).
  • Body mass index between 18 and 28 kg/m\^2, inclusive.
  • Women not of childbearing potential:
  • Women of childbearing potential must have a negative serum pregnancy test at screening and a negative urine pregnancy test prior to drug intake on Day 1; use a reliable method of contraception and continue this contraception for the duration of the study and for at least 2 months after study drug intake. In addition, her partner must use a condom.
  • Systolic blood pressure 100-145 mmHg, diastolic blood pressure 50-90 mmHg, and heart rate (HR) 50-95 beats per minute (inclusive).
  • 12-lead electrocardiogram without clinically relevant abnormalities at screening.
  • Hematology and clinical chemistry results not deviating from the normal range to a clinically relevant extent at screening.
  • Negative results from urine drug screen at screening.
  • Ability to communicate well with the Investigator (if necessary with the help of an interpreter) and to understand and comply with the requirements of the study.

Exclusion

  • Electrocardiograph PQ/PR interval (time interval from the beginning of the P wave to the beginning of the QRS complex) \> 200 milliseconds at screening.
  • Nursing woman.
  • History of asthma or chronic obstructive pulmonary disease.
  • Known hypersensitivity to any excipients of the drug formulation.
  • Treatment with another investigational drug within 3 months prior to screening.
  • Excessive caffeine consumption, defined as \> 800 mg per day at screening.
  • History or clinical evidence of any disease and/or existence of any surgical or medical condition that might interfere with the absorption, distribution, metabolism or excretion of the study drug.
  • Any cardiac condition or illness, including ECG abnormalities, with a potential to increase the cardiac risk of the subject.
  • Smoking within the last month prior to screening.
  • Any immunosuppressive treatment within 6 weeks before study drug administration.
  • Previous treatment with any prescribed or over-the-counter medications within 2 weeks prior to screening.
  • Loss of 250 mL or more of blood within 3 months prior to screening.
  • Lymphopenia (\< 1,000 lymphocytes/μL).
  • Viral, fungal, bacterial or protozoal infection within 4 weeks before study drug administration.
  • Positive results from the hepatitis serology, except for vaccinated subjects, at screening.
  • Positive results from human immunodeficiency vrus serology at screening.
  • Legal incapacity or limited legal capacity at screening.
  • History of alcoholism or drug abuse.
  • Any circumstances or conditions, which, in the opinion of the investigator, may affect full participation in the study or compliance with the protocol.

Key Trial Info

Start Date :

February 1 2009

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

April 1 2009

Estimated Enrollment :

20 Patients enrolled

Trial Details

Trial ID

NCT02223832

Start Date

February 1 2009

End Date

April 1 2009

Last Update

August 22 2014

Active Locations (1)

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Page 1 of 1 (1 locations)

1

Hawaii Clinical Research Center

Honolulu, Hawaii, United States, 96813