Status:

COMPLETED

Efficacy and Safety of All-Oral Combination of Narlaprevir/Ritonavir and Daclatasvir in Treatment-Naїve Patients With Chronic Hepatitis C Genotype 1b

Lead Sponsor:

R-Pharm

Collaborating Sponsors:

Almedis

Conditions:

Chronic Hepatitis C Genotype 1b

Eligibility:

All Genders

18-70 years

Phase:

PHASE2

Brief Summary

The purpose of this study is to confirm that combination of Narlaprevir, Ritonavir and Daclatasvir is safe and highly effective regimen in treatment-naїve patients with chronic hepatitis C (HCV) genot...

Detailed Description

To evaluate effectiveness and safety of treatment with Narlaprevir, Ritonavir and Daclatasvir combination will be selected 105 treatment-naїve patients with chronic HCV genotype 1b without genetic var...

Eligibility Criteria

Inclusion

  • Inclusion Criteria -
  • Subjects who meet all of the following criteria are eligible for participation in the study:
  • Are willing and able to provide written informed consent.
  • Have confirmed chronic HCV infection as documented by:
  • positive anti-HCV antibody (Ab) test or
  • positive HCV RNA or
  • positive HCV genotyping test at least 6 months prior to the Baseline/Day 1 visit.
  • Have HCV genotype 1b at screening as determined by the Central Laboratory. Any non definitive results must exclude the subject from study participation.
  • Minimum HCV-RNA level of ≥10,000 IU at baseline.
  • No evidence of cirrhosis; availability at Baseline of at least one of the following tests, negative results:
  • Liver biopsy within 2 years of screening showing absence of cirrhosis;
  • Fibroscan with a result of ≤ 12.5 kPa within 6 months of baseline/Day1;
  • FibroTest score of ≤ 0.48 AND APRI of ≤ 1 performed during screening. In the absence of a definitive diagnosis of the presence or absence of cirrhosis by the above criteria, a liver biopsy was required. Liver biopsy results supersede the results obtained by Fibroscan or FibroTest.
  • Have a screening electrocardiogram (ECG) without clinically significant abnormalities (P wave \< 0.1 s; PQ interval 0,12-0,2 s; QRS complex 0,06-0,1 s; QT interval 0,35-0,49 s).
  • Must have the following laboratory parameters at screening:
  • alanine aminotransferase (ALT) ≤ 10 x the upper limit of normal (ULN);
  • aspartate aminotransferase (AST) ≤ 10 x ULN;
  • Hemoglobin ≥ 12g/dL for male, ≥ 11g/dL for female subjects;
  • Platelets ≥ 50,000cells/mm3;
  • International normalized ratio (INR) ≤ 1.5 x ULN unless subject has known hemophilia or is stable on an anticoagulant regimen affecting INR;
  • Albumin ≥ 3g/dL;
  • Direct bilirubin ≤ 1.5 x ULN;
  • Hemoglobin A1c (HbA1c) ≤ 10%;
  • Creatinine clearance (CLcr) ≥ 60 mL/min, as calculated by the Cockcroft-Gault equation;
  • Have not been treated with any investigational drug or device within 30 days of the screening visit.
  • A female subject is eligible to enter the study if it is confirmed that she is:
  • Not pregnant or nursing;
  • Of non-childbearing potential (i.e., women who have had a hysterectomy, both ovaries removed, or medically documented ovarian failure, or are postmenopausal women \>50 years of age with cessation \[for ≥12 months\] of previously occurring menses), or
  • Of childbearing potential (i.e., women who had not had a hysterectomy, both ovaries removed, or medically documented ovarian failure). Women ≤ 50 years of age with amenorrhea are considered to be of childbearing potential. These women must have a negative serum pregnancy test at screening and a negative urine pregnancy test on the baseline/Day 1 visit prior to enrollment. They must also agree to one of the following from 3 weeks prior to baseline/Day 1 until 6 months after last dose of the investigational drugs:
  • Complete abstinence from intercourse. Periodic abstinence from intercourse (e.g., calendar, ovulation, sympto thermal, post-ovulation methods) is not permitted Or
  • Consistent and correct use of 1 of the following methods of birth control listed below in addition to a male partner who correctly uses a condom from the date of screening until 6 months after the last dose of the investigational drugs:
  • intrauterine device (IUD) with a failure rate of \< 1% per year;
  • female barrier method: cervical cap or diaphragm with spermicidal agent;
  • tubal sterilization;
  • vasectomy in male partner; Women of childbearing potential must not rely on hormone-containing contraceptives as a form of birth control during the study. Female subjects using a hormone-containing contraceptive prior to screening must stop their contraceptive regimen use from the date of screening until 6 months after their last dose of investigational drugs.
  • All male study participants must agree to consistently and correctly use a condom, while their female partner agrees to use either 1 of the non hormonal methods of birth control listed above or a hormone-containing contraceptive listed below, from the date of screening until 6 months after their last dose of investigational drugs:
  • implants of levonorgestrel;
  • injectable progesterone;
  • oral contraceptives (either combined or progesterone only);
  • contraceptive vaginal ring;
  • transdermal contraceptive patch;
  • Male subjects must agree to refrain from sperm donation for at least 6 months after the last dose of investigational drugs.
  • Are in generally good health as determined by the investigator.
  • Are able to comply with the dosing instructions for study drug administration and are able to complete the study schedule of assessments.
  • Exclusion Criteria -
  • Subjects with any of the following are not eligible for participation in the study:
  • Had prior exposure to IFN, RBV, or other approved or experimental DAA targeting the HCV.
  • Had prior exposure to amiodarone within 24 months before the screening
  • Are pregnant or nursing female or male with pregnant female partner.
  • Сhronic liver disease of a non-HCV etiology (e.g., hemochromatosis, Wilson's disease, α1-antitrypsin deficiency, cholangitis).
  • Are infected with hepatitis B virus (HBV) or human immunodeficiency virus (HIV).
  • Have history of malignancy diagnosed or treated within 5 years; subjects under evaluation for malignancy are not eligible.
  • Have chronic use of systemically administered immunosuppressive agents (e.g., prednisone equivalent \> 10 mg/day).
  • Have clinically relevant drug or alcohol abuse within 12 months of screening. A positive drug screen must exclude subjects unless it can be explained by a prescribed medication; the diagnosis and prescription must be approved by the investigator.
  • Have excessive alcohol consumption, defined as more than 3 drinks on any single day and more than 7 drinks per week for females, and \> than 4 drinks on any single day and more than 14 drinks per week for males.
  • Have history of solid organ transplantation.
  • Have history of clinically significant illness or any other major medical disorder that may interfere with subject treatment, assessment, or compliance with the protocol by Investigators' opinion.
  • Have history of a gastrointestinal disorder (or postoperative condition) that can interfere with the absorption of the study drug.
  • Have history of difficulty with blood collection and/or poor venous access for the purposes of phlebotomy.
  • Usage of any prohibited concomitant medications as described in the protocol (list of drugs with expected drug-drug interactions due to concomitant ritonavir usage)
  • Have known hypersensitivity to the study investigational medicinal product, the metabolites, or formulation excipients.
  • Chronic HCV genotype 1b-infected participant who has the presence of genetic variants coding for the NS5A-Y93 С/H/N/S and/or L31 F/M/V/I amino acid substitutions at Screening.

Exclusion

    Key Trial Info

    Start Date :

    November 27 2017

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    November 21 2018

    Estimated Enrollment :

    105 Patients enrolled

    Trial Details

    Trial ID

    NCT03485846

    Start Date

    November 27 2017

    End Date

    November 21 2018

    Last Update

    December 19 2018

    Active Locations (4)

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    Page 1 of 1 (4 locations)

    1

    FBIS CSRI of Epidemiology of Federal Service on Customers

    Moscow, Russia

    2

    SBEI HPE Moscow State Medical and Dental University n.a. A.I. Evdokimov of Ministry of Health of Russia

    Moscow, Russia

    3

    SBHI of Moscow "City Clinical Hospital #24"

    Moscow, Russia

    4

    St. Petersburg SBHI Center of Prevention and Fight against AIDS and Infection Diseases

    Saint Petersburg, Russia