Status:

COMPLETED

Mass Balance Study of [14C]-Orvepitant Oral Solution in Healthy Male Subjects

Lead Sponsor:

Nerre Therapeutics Ltd.

Conditions:

Healthy

Eligibility:

MALE

30-65 years

Phase:

PHASE1

Brief Summary

This is a single centre, open-label, non-randomised study to assess the mass balance recovery, absorption, metabolism, and excretion of a single oral dose of \[14C\]-orvepitant in healthy male subject...

Eligibility Criteria

Inclusion

  • Key
  • Healthy males
  • Aged 30 to 65 years inclusive at the time of signing informed consent.
  • Body mass index (BMI) of 18.0 to 35.0 kg/m2 as measured at screening.
  • Must provide written informed consent.
  • Must agree to adhere to the contraception requirements
  • Key

Exclusion

  • History of any drug or alcohol abuse in the past 2 years.
  • Regular alcohol consumption \>21 units per week.
  • Current smokers and those who have smoked within the last 12 months.
  • Radiation exposure, including that from the present study, excluding background radiation but including diagnostic x-rays and other medical exposures, exceeding 5 mSv in the last 12 months or 10 mSv in the last 5 years.
  • Clinically significant abnormal clinical chemistry, haematology, or urinalysis as judged by the Investigator.
  • Subjects with a presence of any of the following at screening: bilirubin, alanine aminotransferase (ALT), or aspartate aminotransferase (AST) \>1.5 × the upper limit of normal.
  • Confirmed positive drugs of abuse test result.
  • Positive hepatitis B surface antigen (HBsAg), hepatitis C virus antibody (HCV Ab) or human immunodeficiency virus (HIV) results.
  • Evidence of renal impairment at screening, as indicated by an estimated creatinine clearance (CLcr) of \<80 mL/min using the Cockcroft-Gault equation.
  • History of clinically significant cardiovascular, renal, hepatic, chronic respiratory, or GI disease, neurological or psychiatric disorder, as judged by the Investigator.

Key Trial Info

Start Date :

June 1 2020

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

June 28 2020

Estimated Enrollment :

6 Patients enrolled

Trial Details

Trial ID

NCT04387981

Start Date

June 1 2020

End Date

June 28 2020

Last Update

August 7 2020

Active Locations (1)

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1

Quotient Sciences

Nottingham, United Kingdom