Status:

COMPLETED

A Single Ascending and Repeated Dose Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of TS-142 in Healthy Participants

Lead Sponsor:

Taisho Pharmaceutical R&D Inc.

Conditions:

Healthy Volunteers

Eligibility:

All Genders

18-55 years

Phase:

PHASE1

Brief Summary

This is a study to evaluate the safety, tolerability, and pharmacokinetics of single oral doses of TS-142 compared to placebo and of a single repeated dose compared to placebo in healthy volunteers. T...

Eligibility Criteria

Inclusion

  • Healthy adult male and female participants between 18 and 55 years of age, inclusive
  • Body weight ≥ 45 kg at screening and admission visits.
  • Body Mass Index (BMI) ≥ 18 and ≤ 30 kg/m\^2 at screening visit.

Exclusion

  • Clinically significant abnormal values for hematology, clinical chemistry or urinalysis at the screening and/or admission visits.
  • Clinically significant abnormal physical examination (including neurological assessments), vital signs, or 12-lead ECGs at the screening and/or admission visits.
  • QTcF \>450 msec for male participants or QTcF \>470 msec for female participants at the screening and/or admission visits.
  • Significant history or presence of hepatic, renal, cardiovascular, pulmonary, gastrointestinal, hematological, neurological, immunologic, ophthalmologic, metabolic or oncological disease.
  • History or present diagnosis of sleep disorders.
  • Currently experiencing sleep disturbance related to postmenopausal symptoms at the screening and/or admission visits.
  • History or presence of suicidal behavior, defined as participants who have answered 'YES' to any of the C-SSRS suicidal behavior questions at the screening and/or admission visits.
  • Positive urine screen for alcohol or controlled substances at the screening or admission visits.
  • Recent history (within the previous 6 months) of alcohol or drug abuse.
  • Regular alcohol consumption of \> 2 units/day or 10 units/week during the last 3 months prior to screening. One unit is equivalent to 8 g of alcohol: a half pint (240 mL) of beer, a glass (125 mL) of wine, or 25 mL of spirits.
  • Current use, or use of tobacco or tobacco-containing products (cigarettes, pipes, e-cigarettes, nicotine patches, etc.) during the month prior to screening, or positive urine cotinine screen (\>400 ng/mL) at the screening and/or admission visits.
  • History of and/or current evidence of serologic positive results for hepatitis B surface antigen (HBsAg), hepatitis C antibodies, or human immunodeficiency virus (HIV) antibodies 1 and 2.
  • Donation of one or more units of blood, plasma (including platelet donations), or acute loss of an equivalent amount of blood within 60 days prior to screening visit (one unit= 450 mL).
  • Exposure to any investigational product within 60 days prior to screening.
  • Use of any prescription or over-the-counter medication, herbal medication, vitamins, or mineral supplements within 14 days prior to administration of the study drug.
  • Participants who regularly consume \>500 mg of caffeine on a daily basis.
  • Is known to be allergic to the study drug or any components of the study drug.
  • Participated in strenuous exercise within 48 hours prior to study start (initial dosing) and/or is unwilling to avoid strenuous exercise at any time throughout the study.
  • Participants who work night shifts or need to work night shifts during the trial.

Key Trial Info

Start Date :

September 14 2020

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

January 21 2021

Estimated Enrollment :

28 Patients enrolled

Trial Details

Trial ID

NCT04464239

Start Date

September 14 2020

End Date

January 21 2021

Last Update

February 10 2021

Active Locations (1)

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Page 1 of 1 (1 locations)

1

PPD Phase I unit

Austin, Texas, United States, 78744