Status:

COMPLETED

Multicenter, Double-blind, Placebo-controlled Study to Evaluate the Efficacy and Safety of Fluconazole in Hypercalcicuric Patients With Increased 1.25(OH) 2D Levels

Lead Sponsor:

Hospices Civils de Lyon

Conditions:

Nephrolithiasis

Nephrocalcinosis

Eligibility:

All Genders

10-60 years

Phase:

PHASE2

Brief Summary

Hypercalciuria is one of the most frequent metabolic disorders associated with nephrolithiasis and/or nephrocalcinosis leading to Chronic Kidney Disease (CKD) and bone complications in adults. Hyperc...

Eligibility Criteria

Inclusion

  • Patients who presented in their medical history nephrolithiasis and/or nephrocalcinosis
  • Patients who have at inclusion (V1), a local biological evaluation with:
  • 24-hour urine calcium \> 0.1 mmol/kg/day,
  • and 1,25(OH)2D levels ≥ 150 pmol/L,
  • and 25-OH-D levels ≥ 20 nmol/L,
  • and calcemia levels ≤ 2.65 mmol/L.
  • Children from 10 years
  • Adults until 60 years
  • Women of child-bearing potential (including sexually active adolescent females) must use highly effective methods of contraception (Annex 7 CTFG recommendations) during the study period. Likewise, partners of male patients of child-bearing potential must use highly effective methods of contraception. Male patients must use condoms.
  • Patients insured or beneficiary of a health insurance plan
  • Evidence of signed and dated informed consent document(s) indicating that the subject and/or his parents/legal guardian has/have been informed of all pertinent aspects of the trial.

Exclusion

  • Patient who already received fluconazole or ketoconazole during the last 6 months before inclusion
  • Patient weight below than 28 kg
  • Patient with BMI \>35
  • Women menopaused
  • Patients who cannot stop hydrochlorothiazide or other diuretics during the screening and study period
  • Patients who cannot stop vitamin D supplementation and/or calcium supplementation (drugs, enriched waters, etc.) during the study period
  • Hypersensibility to fluconazole and/or other derivative azoles and/or excipients
  • Due to the presence of lactose excipient, patients presenting rare hereditary abnormalities of galactose intolerance, of Lapp lactase deficit or of glucose-galactose malabsorption
  • Patients who need co-administration with other drugs known to prolong the QT interval and metabolized by cytochrome P450 (CYP) 3A4 (pimozide, quinidine and erythromycin; the exhaustive list of drugs known to prolong the QTc is available on: https://crediblemeds.org).
  • Patients with iatrogenic hypercalciuria (vitamin D intoxication, immobilization)
  • Relating to the risk of QT interval prolongation:
  • congenital Long QT syndrome;
  • familial history of sudden cardiac death before 50 years of age;
  • cardiopathy: ischemia or myocardial infarction, congestive cardiac insufficiency, left ventricle hypertrophy, cardiomyopathy, conduction trouble within 6 months preceding the inclusion;
  • arrhythmia history (in particular ventricular arrhythmia, auricular fibrillation or recent rhythm recovery after an auricular fibrillation);
  • electrolytic instabilities: hypokalemia, hypomagnesemia, hypocalcemia ;
  • bradycardia (\< 50 beats per minute) ;
  • acute neurological events (i.e. intracranial hemorrhage or sub-arachnoid, cerebrovascular accident, intracranial trauma) within 6 months preceding the inclusion;
  • adult patients with a QT interval/corrected QT interval \> 470ms for women and \> 450ms for men at the ECG performed at the inclusion visit (V1). For children from 10 years, the QT interval/corrected QT interval should be \> 460ms for girls and \> 450ms for boys.
  • Children with a history of cardiac pathology
  • Patients with an estimated glomerular filtration rate \< 60 mL/min/1.73m²
  • Patients with a liver disease or an abnormality in the initial liver lab test
  • Patients with enuresis
  • Patients with another cause of identified lithiasis
  • Patients suffering from granulomatosis pathology such as sarcoidosis
  • Patient with hyperparathyroidism
  • Women who are pregnant or breast feeding, or who have a project of pregnancy before the end of the study
  • Patients with a project of travelling in a sunny area during the study period
  • Immunodeficient patients
  • Patients with other diseases or disorders that could preclude assessment
  • Patient who is participating in another research study that may interfere with the results or conclusions of this study
  • Patients under judicial protection.

Key Trial Info

Start Date :

January 13 2021

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

July 1 2024

Estimated Enrollment :

56 Patients enrolled

Trial Details

Trial ID

NCT04495608

Start Date

January 13 2021

End Date

July 1 2024

Last Update

July 12 2024

Active Locations (11)

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Page 1 of 3 (11 locations)

1

Service de Néphrologie Rhumatologie Dermatologie Pédiatrique

Bron, France, Bron

2

CHU de Dijon

Dijon, France

3

Hôpital Edouard Herriot

Lyon, France

4

APHM - CHU Conception

Marseille, France