Status:

COMPLETED

Phase 1 First in Human Study of ZN-d5 as a Single Agent

Lead Sponsor:

K-Group Alpha, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc.

Conditions:

Acute Myeloid Leukemia

Non Hodgkin Lymphoma

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

Phase 1 dose escalation study of ZN-d5 in subjects with relapsed or refractory non-Hodgkin lymphoma (NHL) or acute myeloid leukemia (AML).

Detailed Description

This is an open-label multicenter Phase 1 dose escalation study evaluating the safety, tolerability, clinical activity, pharmacokinetics and pharmacodynamics of the novel BCL-2 inhibitor ZN-d5 in subj...

Eligibility Criteria

Inclusion

  • Key
  • NHL: relapsed or refractory NHL including DLBCL, FL, MZL, MCL, LCL, LPL and PTC
  • Subjects must have received at least 2 prior lines of therapy and have either failed or not be eligible for any available therapies expected to provide clinical benefit and have measurable disease.
  • AML: Primary, secondary, or treatment-related AML, relapsed or refractory to prior therapy, which may include failure of one cycle of induction therapy.
  • White blood cell count \< 25 × 109/L. Cytoreduction prior to treatment is acceptable.
  • Subjects may not be pregnant and must agree to use an effective method of contraception.
  • Eastern Cooperative Oncology Group performance status ≤ 2.
  • Estimated life expectancy of at least 12 weeks.
  • Adequate hematologic and organ function, including creatinine clearance ≥ 60 mL/min.
  • Key

Exclusion

  • Recent interventions including major surgery, radiation therapy, stem cell transplant.
  • Treatment with anti-neoplastic agents with 5 half-lives.
  • Significant unresolved toxicity from prior treatments including active GVHD.
  • Active central nervous system disease.
  • Clinically substantial myocardial impairment.
  • Prior therapy with venetoclax.

Key Trial Info

Start Date :

October 13 2020

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

December 12 2023

Estimated Enrollment :

39 Patients enrolled

Trial Details

Trial ID

NCT04500587

Start Date

October 13 2020

End Date

December 12 2023

Last Update

September 19 2024

Active Locations (14)

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Page 1 of 4 (14 locations)

1

Site 2708

Darlinghurst, New South Wales, Australia

2

Site 2704

Liverpool, New South Wales, Australia

3

Site 2710

Kurralta Park, South Australia, Australia

4

Site 2709

Hobart, Tasmania, Australia