Status:

COMPLETED

Pharmacokinetics and Pharmacodynamics of Different PTG-300 Regimens in Healthy Volunteers

Lead Sponsor:

Protagonist Therapeutics, Inc.

Conditions:

Healthy Volunteers

Eligibility:

MALE

18-65 years

Phase:

PHASE1

Brief Summary

To estimate the bioavailability of PTG-300 following subcutaneous and intramuscular administration in healthy volunteers.

Detailed Description

This is a single center, open-label study in healthy males. Subjects will be screened for eligibility within 28 days of dosing. Twelve subjects will receive single doses of the following treatments i...

Eligibility Criteria

Inclusion

  • Healthy male volunteers, age 18 to 65 years, inclusive.
  • Subjects must have a Body Mass Index (BMI) between 18 and 32 kg/m2 inclusive.
  • Subjects must have clinical laboratory values within normal range as specified by the testing laboratory, unless deemed not clinically significant by the Investigator.
  • Agree to use a barrier method of contraception from Day -2 to 90 days after the last dose of study drug.
  • Subjects must have the ability and willingness to attend the necessary visits to the study center.

Exclusion

  • History of clinically significant endocrine, neurological, gastrointestinal, cardiovascular, haematological, hepatic, immunological, renal, respiratory, or genitourinary abnormalities or diseases.
  • History of malignancy, with the exception of adequately treated non-melanomatous skin carcinoma.
  • Mentally or legally incapacitated, has significant emotional problems at the time of Screening Visit or expected during the conduct of the study, or has a history of a clinically significant psychiatric disorder that would impact the subjects ability to participate in the trial according to the Investigator.
  • Fever (body temperature \>38°C) or symptomatic viral or bacterial infection within 2 weeks prior to screening; evidence of intestinal infection within 30 days prior to screening.
  • History of severe allergic or anaphylactic reactions.
  • A supine blood pressure outside the range of 90 to 139 mm Hg systolic and 50 to 89 mm Hg diastolic, OR heart rate (HR) \>100 beats per minute at Screening and at Day -1.
  • Laboratory values that are outside the normal range and considered clinically significant by the Investigator.
  • Positive test for hepatitis C antibody, hepatitis B surface antigen or human immunodeficiency virus (HIV) antibody at Screening.
  • Subjects considered at high risk of iron deficiency according to the Investigator.
  • Subjects with iron deficiency as defined by a ferritin or transferrin saturation below the normal range
  • Clinically significant abnormality on ECG performed at the Screening Visit or prior to administration of the initial dose of study drug.
  • Corrected QT (QTcF) greater than 450 msec at Screening.
  • Subjects with a positive toxicology screening panel.
  • Subjects with a history of substance abuse or dependency or history of recreational IV drug use (by self-declaration).
  • Consumption of \>14 alcohol units per week (where 1 unit = 284 mL of beer, 25 mL of 40% spirit, or a 125 mL glass of wine).
  • Unable to refrain from or anticipates the use of any medications, including prescription and non-prescription drugs and herbal remedies (such as St. John's Wort \[Hypericum perforatum\]), beginning 14 days (or 5 half lives, whichever is longer) before administration of the initial dose of study drug and continuing throughout the study until the final study visit.

Key Trial Info

Start Date :

September 14 2020

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

June 30 2021

Estimated Enrollment :

12 Patients enrolled

Trial Details

Trial ID

NCT04516382

Start Date

September 14 2020

End Date

June 30 2021

Last Update

September 16 2021

Active Locations (1)

Enter a location and click search to find clinical trials sorted by distance.

Page 1 of 1 (1 locations)

1

Protagonist Clinical Center

Melbourne, Australia