Status:

TERMINATED

Central Nervous System Effects Following Infusion of Diphenhydramine Using Pharmacokinetic and Pharmacodynamic Modeling

Lead Sponsor:

Dent Neuroscience Research Center

Conditions:

Central Nervous System Effects of Diphenhydramine

Pharmacokinetics of Diphenhydramine

Eligibility:

All Genders

35+ years

Phase:

PHASE4

Brief Summary

This study seeks to explore the magnitude and duration of central nervous system effects and pharmacokinetics after intravenous infusion of diphenhydramine.

Eligibility Criteria

Inclusion

  • Medically-stable volunteers of either gender between 35 and 50 years old or over the age of 65
  • No medication changes anticipated for the duration of the study except as defined in protocol

Exclusion

  • Insulin-dependent diabetes
  • Psychiatric or neurologic disease affecting cognition in a way that may interfere with study outcomes in the opinion of the investigator
  • Unstable Coronary Artery Disease (active angina, MI within 6 months, stent placement within 6 months, cardiac surgery within 6 months)
  • Estimated CrCl \< 30 mL/min using the Cockroft-Gault equation based on ideal body weight or total body weight
  • Any malignancy actively being treated or not in remission
  • Currently taking any CNS stimulant or depressant medications that may interfere with study outcomes in the opinion of the investigator unless using as defined in the protocol
  • Positive toxicology test for marijuana at screening visit or visit 2 or using marijuana not as defined in the protocol
  • Active or recent history of a substance use disorder within one year
  • Any medical condition that in the opinion of the investigator would disqualify the subject from participation in the study
  • Female subjects who are pregnant, planning to become pregnant, or breastfeeding on any study day
  • Female subjects of childbearing potential unwilling to use acceptable method of contraception during the study as defined in the protocol
  • Contraindication, known allergy, or suspected intolerability to study medication
  • Receipt of an antihistamine within 5 half-lives prior to the start of study visit 1 or study visit 2, as determined by the investigator
  • Positive toxicology test for a drug that is inconsistent with permitted medication use (defined in the protocol) as interpreted by the investigator
  • Participation in any other investigational drug study during the study or within 4 weeks prior to screening

Key Trial Info

Start Date :

March 15 2022

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

October 4 2022

Estimated Enrollment :

3 Patients enrolled

Trial Details

Trial ID

NCT05219604

Start Date

March 15 2022

End Date

October 4 2022

Last Update

February 14 2024

Active Locations (1)

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Page 1 of 1 (1 locations)

1

Dent Neurologic Institute

Amherst, New York, United States, 14226

Central Nervous System Effects Following Infusion of Diphenhydramine Using Pharmacokinetic and Pharmacodynamic Modeling | DecenTrialz