Status:

COMPLETED

Safety, PK, PD, Clinical Activity of KT-333 in Adult Patients With Refractory Lymphoma, Large Granular Lymphocytic Leukemia, Solid Tumors

Lead Sponsor:

Kymera Therapeutics, Inc.

Conditions:

Non Hodgkin Lymphoma (NHL)

Peripheral T-cell Lymphoma (PTCL)

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

This Phase 1a/1b study will evaluate the safety, tolerability and the pharmacokinetics/pharmacodynamics (PK/PD) of KT-333 in Adult patients with Relapsed or Refractory (R/R) Lymphomas, Large Granular ...

Detailed Description

This is an open-label Phase 1a (dose escalation)/1b (dose expansion) first-in-human study of KT-333 in adult patients. Patients with relapsed/refractory (R/R) lymphomas, LGL-L, T-PLL, and solid tumors...

Eligibility Criteria

Inclusion

  • Phase 1a Only: Cytologically or pathologically confirmed Lymphomas (including Hodgkin's, B-cell, T-cell, Small Lymphocytic, or Natural-Killer (NK)-cell Lymphomas and LGL-L), T-PLL and solid tumors with the exception of chronic lymphocytic leukemia (CLL) Note: Patients with indolent non-Hodgkin's lymphoma (NHL) and small lymphocytic lymphoma (SLL) are only eligible if not require immediate cytoreductive therapy or if there are no available treatments with potential benefit.
  • Phase 1b Only: Histologically or pathologically confirmed PTCL, CTCL, LGL-L \[T-cell LGL-L or Chronic Lymphoproliferative Disorder of NK-cells (CLPD-NK)\], or solid tumors.
  • Fresh or archival formalin fixed paraffin embedded (FFPE) tumor tissue or 15 slides preferably collected within 6 months or 2 years prior to first dose of the study drug (for lymphoma and solid tumor patients respectively).
  • Phase 1a only: Lymphoma and Solid Tumor: Relapsed and/or refractory disease to at least 2 prior systemic standard of care treatments or for whom standard therapies are not available.
  • Phase 1a: LGL-L/T-PLL only: Relapsed and/or refractory disease to at least 1 prior systemic standard of care treatment or for whom standard therapies are not available.
  • Phase 1b only: All disease types: Relapsed and/or refractory disease to at least 1 prior systemic standard of care treatments or for whom standard therapies are not available.
  • LGL-L patients only (hematology specific criteria):
  • One of the following:
  • Severe neutropenia \< 500/mm3, or,
  • Symptomatic anemia and/or,
  • Transfusion-dependent anemia.
  • ANC ≥ 200/μL at Screening and C1D1 (pre dose)
  • Platelet count ≥ 100,000/μL (assessed ≥ 7 days following last platelet transfusion in patients with thrombocytopenia requiring platelets).
  • LGL-L Patients Only (baseline disease characteristics):
  • CD3+CD8+ cell population \>650/mm3;
  • CD3+CD8+CD57+ population \>500/mm3;
  • Presence of a clonal T-cell receptor (within 1 month of diagnosis);
  • Note: patients with T-LGLL may be included with PI approval even if CD3+CD8+ cell population is\<650/mm3 or CD3+CD8+CD57+ population is \<500/mm3, though +TCR is required;
  • NK LGL is also permitted, provided there is a clonal NK-cell population noted with\>500 cells/mm3
  • PTCL and solid tumors Only: Measurable disease at Screening. Solid tumor patients with non-measurable disease are allowed in Phase1a
  • T-PLL: Measurable disease per Lugano and/or atypical T lymphocytes quantifiable by flow cytometry or morphology in the peripheral blood or bone marrow.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0-2 at Screening and C1D1 (pre-dose).
  • Adequate bone marrow function at Screening and C1D1 (pre-dose) for all patients except those with LGL-L Adequate liver/kidney organ function at Screening and C1D1 (pre-dose) for all patients.
  • Women of childbearing potential (WOCBP) must agree to use highly effective contraceptive methods for the duration of study treatment and 6 months after the last dose of KT333.

Exclusion

  • Known active uncontrolled or symptomatic central nervous system (CNS) metastases, carcinomatous meningitis, or leptomeningeal disease as indicated by clinical symptoms, cerebral edema, and/or progressive growth.
  • Note: Patients with solid tumors are eligible if their CNS metastases or cord compression have been treated (e.g., radiotherapy, stereotactic surgery) and they are clinically stable, off steroids for at least 4 weeks before first dose of study drug and have no evidence of progression at time of study enrollment.
  • Note: Patients with lymphomas are eligible if their CNS metastases or cord compression have been treated effectively (i.e. achieved CR) and there is no clinical or radiographic evidence of active lymphoma.
  • Diagnosis of Chronic Lymphocytic Leukemia (CLL).
  • History of or active concurrent malignancy other than lymphoma or solid tumors unless the patient has been disease-free for ≥ 2 years.
  • Patient has not recovered from any clinically significant adverse events (AEs) of previous treatments to pretreatment baseline or Grade 1 prior to first dose of study drug.
  • Ongoing unstable cardiovascular function.
  • Autologous hematopoietic stem cell transplant less than 3 months prior to first dose of study drug.
  • Prior allogenic hematopoietic or bone marrow transplant.

Key Trial Info

Start Date :

May 19 2022

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

March 3 2025

Estimated Enrollment :

56 Patients enrolled

Trial Details

Trial ID

NCT05225584

Start Date

May 19 2022

End Date

March 3 2025

Last Update

March 19 2025

Active Locations (13)

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Page 1 of 4 (13 locations)

1

UC Irvine Health-Chao Family Comprehensive Cancer Center

Orange, California, United States, 92868-3201

2

Norton Cancer Institute

Louisville, Kentucky, United States, 40207

3

Henry Ford Hospital

Detroit, Michigan, United States, 48202

4

Hackensack University Medical Center, John Theurer Cancer Center

Hackensack, New Jersey, United States, 07601