Status:

ACTIVE_NOT_RECRUITING

A Single Arm Phase 2 Study to Evaluate Efficacy and Safety of Trastuzumab Deruxtecan for Patients With HER2 Mutant NSCLC

Lead Sponsor:

AstraZeneca

Collaborating Sponsors:

Daiichi Sankyo

Conditions:

HER2-mutant Non-Small Cell Lung Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

The purpose of this study is to evaluate the efficacy and safety of T-DXd in participants with HER2 mutant metastatic non-squamous NSCLC.

Eligibility Criteria

Inclusion

  • Pathologically documented metastatic non-squamous NSCLC.
  • Has relapsed from or is refractory to at least one-line of anticancer treatment.
  • Documented HER2 exon 19 or 20 mutation from central FFPE tumour tissue testing.
  • WHO or ECOG performance status of 0 or 1.
  • Presence of at least one measurable lesion assessed by the investigator based on RECIST 1.1.
  • LVEF ≥ 50% within 28 days before enrolment.

Exclusion

  • Mixed small cell lung cancer, squamous histology NSCLC, and sarcomatoid histology variant NSCLC.
  • Corrected QT interval (QTcF) prolongation to \> 470 ms (females) or \> 450 ms (males), based on average of the screening triplicate 12-lead ECG.
  • History of (non-infectious) ILD/pneumonitis that required steroids, has current ILD/pneumonitis, or where suspected ILD/pneumonitis cannot be ruled out by imaging at screening.
  • Has unresolved toxicities from previous anticancer therapy, defined as toxicities (excluding alopecia) not yet resolved to Grade ≤1 or baseline. Participants with clinically stable chronic Grade 2 toxicity not reasonably expected to be exacerbated by study intervention may be included only after consultation with the AstraZeneca study physician or designee.
  • Has been previously treated with HER2-targeted therapies, except for pan-HER class TKIs or has received prior treatment with an ADC which consists of an exatecan derivative that is a topoisomerase I inhibitor.

Key Trial Info

Start Date :

July 13 2022

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

March 16 2026

Estimated Enrollment :

72 Patients enrolled

Trial Details

Trial ID

NCT05246514

Start Date

July 13 2022

End Date

March 16 2026

Last Update

August 28 2025

Active Locations (28)

Enter a location and click search to find clinical trials sorted by distance.

Page 1 of 7 (28 locations)

1

Research Site

Baoding, China, 071000

2

Research Site

Beijing, China, 100142

3

Research Site

Beijing, China, 100191

4

Research Site

Changchun, China, 130000