Status:

TERMINATED

NUV-868 as Monotherapy and in Combination With Olaparib or Enzalutamide in Adult Patients With Advanced Solid Tumors

Lead Sponsor:

Nuvation Bio Inc.

Conditions:

Advanced Solid Tumor

Ovarian Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

NUV-868-01 is a first-in human, open- label, Phase 1/2 dose escalation and expansion study in patients with advanced solid tumors. The Phase 1 and 1b portions include patients with advanced solid tumo...

Detailed Description

This study was initially planned as a Phase 1/2 study; however, the study stopped early prior to the start of Phase 2.

Eligibility Criteria

Inclusion

  • Key Inclusion Criteria For All Phases and Cohorts:
  • Recovered from toxicity to prior anticancer therapy
  • Adequate bone marrow and organ function
  • No known active or symptomatic central nervous system (CNS) disease
  • Cohort-Specific Inclusion Criteria: In addition to the inclusion criteria listed above, the following criteria apply for enrollment into specific cohorts.
  • Phase 1 (NUV-868 Monotherapy)
  • Patients with advanced solid tumors that have progressed during or after treatment with approved therapies or for which there is no standard effective therapy available
  • Life expectancy of \> 3 months
  • Eastern Cooperative Oncology Group Performance Status ≤ 2
  • Measurable or non-measurable disease
  • Phase 1b (NUV-868 in Combination With Enzalutamide or Olaparib)
  • Life expectancy of \> 3 months
  • Eastern Cooperative Oncology Group Performance Status ≤ 2
  • (Select cohorts only) Measurable disease
  • Patient must be able to read and write sufficiently to document food intake and study drug dosing on the Dosing Diary or must have a caregiver who is willing and able to complete the Dosing Diary with the patient.
  • One of the following tumor types:
  • Ovarian: Platinum-resistant OR platinum-refractory high grade serous ovarian, fallopian, or primary peritoneal cancer in the relapsed setting
  • Pancreatic: Pancreatic ductal adenocarcinoma (PDAC) with progression on or after treatment with at least one line of systemic chemotherapy in the advanced setting
  • Prostate: Histologically confirmed, metastatic adenocarcinoma of the prostate (adenocarcinoma/high grade carcinoma with neuroendocrine features is allowed) with progression on or after treatment with at least one NHT in the metastatic setting
  • Breast: Triple-negative breast cancer (TNBC) with progression on or after treatment with at least one line of systemic chemotherapy in the advanced setting
  • Other advanced tumors (only Phase 1b dose escalation, NUV-868 + olaparib): the study Medical Monitor must approve enrollment.
  • For all tumor types: Patients will be allowed in the study regardless of their BRCA/HRR status.
  • Phase 2
  • Life expectancy of \> 6 months
  • (Select cohorts only): At least one measurable lesion defined by standard criteria
  • Eastern Cooperative Oncology Group Performance Status ≤ 1
  • One of the following tumor types:
  • Ovarian: Platinum-resistant or platinum- refractory high grade serous ovarian, fallopian, or primary peritoneal cancer in the relapsed setting
  • Pancreatic: Progression on or after treatment with at least one line of systemic chemotherapy in the advanced setting
  • Prostate: Histologically confirmed, metastatic adenocarcinoma of the prostate (adenocarcinoma/high grade carcinoma with neuroendocrine features is allowed) with progression on or after treatment with at least one NHT in the metastatic setting
  • Breast: TNBC with progression on or after treatment with at least one line of systemic chemotherapy in the advanced setting
  • Key Exclusion Criteria For All Phases and Cohorts:
  • Have received chemotherapy, hormonal therapy (except for ongoing luteinizing hormone-releasing hormone \[LHRH\] analogs in male patients and premenopausal women), radiation, or biological anticancer therapy within 14 days prior to the first dose of NUV-868.
  • Received treatment with an investigational agent for any indication within 14 days for non-myelosuppressive agent, or within 21 days or \< 5 half-lives (whichever is longer) for myelosuppressive agent, prior to the first dose of study treatment.
  • Requires medications that are known to be strong (or moderate for olaparib) inducers and/or strong (or moderate for olaparib) inhibitors of CYP3A4/5 enzymes.
  • Female patients who are pregnant of breastfeeding.

Exclusion

    Key Trial Info

    Start Date :

    March 29 2022

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    July 15 2024

    Estimated Enrollment :

    82 Patients enrolled

    Trial Details

    Trial ID

    NCT05252390

    Start Date

    March 29 2022

    End Date

    July 15 2024

    Last Update

    November 6 2025

    Active Locations (22)

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    Page 1 of 6 (22 locations)

    1

    The University of Arizona Cancer Center

    Tucson, Arizona, United States, 85724

    2

    Ellison Institute of Technology

    Los Angeles, California, United States, 90064

    3

    Rocky Mountain Cancer Centers, LLP

    Aurora, Colorado, United States, 80012

    4

    Rocky Mountain Cancer Centers, LLP

    Lone Tree, Colorado, United States, 80124