Status:

ACTIVE_NOT_RECRUITING

Cabazitaxel in Combination With 177Lu-PSMA-617 in Metastatic Castration-resistant Prostate Cancer

Lead Sponsor:

Peter MacCallum Cancer Centre, Australia

Conditions:

Metastatic Castration-resistant Prostate Cancer

mCRPC

Eligibility:

MALE

18+ years

Phase:

PHASE1

PHASE2

Brief Summary

This clinical trial will evaluate the safety of Cabazitaxel in combination with 177Lu-PSMA-617 in metastatic castration-resistant prostate cancer.

Detailed Description

This prospective, single-centre, single-arm, open label, phase I/II trial will assess the safety, efficacy and anti-tumour activity of cabazitaxel in combination with 177Lu-PSMA-617 in patients with m...

Eligibility Criteria

Inclusion

  • Male patients aged 18 years or older at the time of informed consent.
  • Patient has provided written informed consent.
  • Histologically confirmed adenocarcinoma of the prostate without neuroendocrine or small cell differentiation.
  • Eastern Cooperative Oncology Group (ECOG) performance status of ≤ 1
  • Patients must have had prior treatment with docetaxel.
  • Patients must have progressed on a second-generation androgen receptor (AR)-targeted agent (e.g., enzalutamide, abiraterone, or apalutamide) in the castrate-resistant setting.
  • Patients must have progressive disease. The Prostate Cancer Clinical Trials Working Group 3 (PCWG3) defines this as any one of the following:
  • PSA progression: minimum of two rising PSA values from a baseline measurement with an interval of ≥ 1 week between each measurement
  • Soft tissue or visceral disease progression as per Response Evaluation Criteria in Solid Tumours version 1.1 (RECIST 1.1) criteria
  • Bone progression: ≥ 2 new lesions on bone scan
  • At least three weeks since the completion of surgery prior to registration.
  • Prior surgical orchiectomy or chemical castration maintained on luteinizing hormone-releasing hormone (LHRH) analogue (agonist or antagonist).
  • Serum testosterone levels ≤ 1.75nmol/L within 28 days prior to registration.
  • Imaging evidence of metastatic disease documented with either whole body bone scan (WBBS) or computed tomography (CT) scan performed within 28 days prior to registration.
  • Significant prostate-specific membrane antigen (PSMA) avidity on PSMA PET/CT, defined as a minimum uptake of SUVmax 15 at a site of disease.
  • Patients must have a life expectancy ≥ 12 weeks.
  • Assessed by a medical oncologist as suitable for treatment with cabazitaxel and 177Lu-PSMA-617.
  • Patients must have adequate bone marrow, hepatic and renal function documented within 28 days prior to registration, defined as:
  • Haemoglobin ≥ 90 g/L independent of transfusions (no red blood cell transfusion in last 28 days prior to registration)
  • Absolute neutrophil count (ANC) ≥ 1.5x10\^9/L
  • Platelets ≥ 150 x10\^9/L
  • Total bilirubin ≤ 1.5 x upper limit of normal (ULN) except for patients with known Gilbert's syndrome, where this applies for the unconjugated bilirubin component
  • Aspartate transaminase (AST) and alanine transaminase (ALT) ≤ 2.5 x ULN if there is no evidence of liver metastasis or ≤ 5 x ULN in the presence of liver metastases
  • Albumin ≥ 25 g/L
  • Adequate renal function: patients must have a creatinine clearance estimated of ≥ 40 mL/min using the Cockcroft-Gault equation
  • Sexually active patients are willing to use medically acceptable forms of barrier contraception.
  • Willing and able to comply with all study requirements, including all treatments and the timing and nature of all required assessments.

Exclusion

  • Superscan on WBBS or diffuse marrow disease on PSMA PET.
  • Site(s) of measurable disease that are FDG-positive with low PSMA expression (SUVmax \<10).
  • Prior treatment with cabazitaxel or 177Lu-PSMA-617.
  • Contraindications to the use of corticosteroid treatment.
  • Other malignancies within the previous 2-years other than basal cell or squamous cell carcinomas of skin or other cancers that are unlikely to recur within 24 months.
  • Presence of untreated brain metastases or leptomeningeal metastases.
  • Patients with symptomatic or impending cord compression unless appropriately treated beforehand and clinically stable for ≥ four weeks.
  • Concurrent illness, including severe infection that may jeopardise the ability of the patient to undergo the procedures outlined in this protocol with reasonable safety.
  • Persistent toxicities (CTCAE v5.0 \>/= Grade 2) caused by previous cancer therapy, excluding alopecia.
  • Known HIV or hepatitis B or C infection.
  • Radiotherapy or systemic anti-cancer therapies administered within 14 days prior to registration, excluding androgen deprivation therapy (ADT).

Key Trial Info

Start Date :

July 14 2022

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

December 1 2026

Estimated Enrollment :

35 Patients enrolled

Trial Details

Trial ID

NCT05340374

Start Date

July 14 2022

End Date

December 1 2026

Last Update

April 6 2025

Active Locations (2)

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Page 1 of 1 (2 locations)

1

St Vincent's Hospital

Sydney, New South Wales, Australia, 2000

2

Peter MacCallum Cancer Centre

Melbourne, Victoria, Australia, 3000