Status:

COMPLETED

PK/PD Study of 2 Agalsidase Formulations in Single Dose of 1 mg/kg Administered to Healthy Volunteers as IV Infusion

Lead Sponsor:

Bio Sidus SA

Conditions:

Fabry Disease

Eligibility:

MALE

18-40 years

Phase:

PHASE1

Brief Summary

Pharmacokinetic/Pharmacodynamic Study of 2 agalsidase beta Formulations in Single Dose Administered to Healthy Volunteers as intravenous infusion, at a concentration of 1 mg/kg

Detailed Description

Volunteers will receive either one or the other agalsidase beta formulation. Drug will be administered as an intravenous 5h infusion. Plasma samples will be taken at different time points, from before...

Eligibility Criteria

Inclusion

  • Male subjects between the ages of 18 and 40
  • Body mass index (BMI) between 19 and 25 kg/m².
  • Volunteers whose complementary exams (ECG, chest X-ray, blood and urine, PCR for COVID-19), performed prior to their inclusion are within the normal range and/or are not clinically significant according to the investigator's judgement.
  • Subjects with systolic blood pressure higher than 110 mmHg and lower than 139 mmHg, diastolic blood pressure higher than 70 mmHg and lower than 89 mmHg with a heart rate higher than 50 and lower than 90 beats per minute after being seated for 5 minutes and, then, standing up (extreme values are included)
  • Volunteers who are well disposed to the study and have signed the approved informed consent prior to the start of the study

Exclusion

  • History of clinically significant allergies (except for untreated asymptomatic seasonal allergies)
  • A drop of ≥ 20 mmHg of systolic blood pressure or ≥ 10 mmHg of diastolic blood pressure within the first 3 minutes after the postural change
  • Volunteers who are receiving other drugs (prescription or over-the-counter) or who have within the 2 weeks prior to the study
  • Volunteers with history of autoimmune diseases.
  • Chronic disorders of the CNS, psychological and/or psychiatric disorders: bipolar disorder, severe depression, insomnia, changes in personality
  • Active or chronic infections
  • Having received live or inactivated viral or bacterial vaccines, within the fifteen days prior to visits 1 or 2
  • For COVID vaccines, a 15 day window period prior to visits #1 or #2 must be respected. This period was taken from the recommendations published by the National Ministry of Health on May 29th 2021. The volunteer will be able to receive the vaccine 35 days after receiving the investigational product.
  • Known allergies to any of the components of the formulations
  • Active smoker, of more than 10 cigarettes/day
  • Current clinical evidence of severe digestive disorders, surgeries of the gastrointestinal tract (except for appendectomy)
  • Current clinical evidence of kidney disease
  • Current clinical evidence of liver disorders
  • Current clinical evidence of respiratory and cardiac disease
  • Presence of diabetes mellitus, thyroid dysfunction or other endocrine disorders
  • Evidence of active gastroduodenal disease
  • History of peripheral thrombotic phenomena
  • Underlying neurological disease
  • Presence of a current progressive chronic disease
  • History of drug or alcohol abuse or addiction within the last three years
  • Participation in a clinical study within the last three months
  • Use of any drug within the fourteen days prior to the start of the study that, according to the principal investigator's judgement may interfere with the biodistribution of the medicinal product.
  • Subjects who have donated or suffered from blood loss within the twelve weeks prior to the start of the study, or intends to donate blood within the following three months after the completion of the study.
  • Excessive drinker of tea, cocoa, mate, coffee and/or caffeinated drinks (\>5 cups/day) or of wine (\>0.5 L/day) or alcohol (\>50 ml/day)
  • Significant abnormalities in the electrocardiogram
  • Positive PCR test for COVID-19
  • Positive serology for HIV, hepatitis B or hepatitis C
  • Abnormal clinical laboratory test results (that according to the principal investigator's judgement are considered clinically significant)
  • Uncooperative volunteers

Key Trial Info

Start Date :

October 23 2021

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

April 17 2022

Estimated Enrollment :

24 Patients enrolled

Trial Details

Trial ID

NCT05343715

Start Date

October 23 2021

End Date

April 17 2022

Last Update

October 15 2025

Active Locations (1)

Enter a location and click search to find clinical trials sorted by distance.

Page 1 of 1 (1 locations)

1

Sanatorio Nuestra Señora del Pilar

Ciudadela, Buenos Aires, Argentina, 1702