Status:

RECRUITING

Regorafenib Combined With TAS-102 Versus Regorafenib Monotherapy in Third or Later Line Therapy of mCRC

Lead Sponsor:

Fudan University

Conditions:

Metastatic Colorectal Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

The purpose of this study is to evaluate the clinical benefit of regorafenib combined with TAS-102 compared with regorafenib monotherapy in patients with metastatic colorectal cancer who have failed a...

Detailed Description

Based on the current diagnostic and treatment guidelines, regorafenib and TAS-102 monotherapy are both standard third-line treatment options for patients with metastatic colorectal cancer (mCRC), yet ...

Eligibility Criteria

Inclusion

  • A total of 101 patients with metastatic colorectal cancer who meet the inclusion criteria and do not meet the exclusion criteria for receiving third-line or later-line therapy will be randomly assigned to receive corresponding treatment in a 1:1 ratio.
  • The subjects must meet all of the following criteria to be eligible for this study:
  • Patients with histologically confirmed recurrent/metastatic colorectal adenocarcinoma.
  • Patients who have failed at least one prior standard first- or second-line therapy, including fluoropyrimidine-based therapy, oxaliplatin, irinotecan, and bevacizumab. Treatment failure is defined as either radiographic evidence of disease progression or unacceptable toxicity during treatment or within three months following completion of therapy.
  • (Note: a. each line of therapy should include at least one or more chemotherapy agents administered for at least one cycle; b. adjuvant/neoadjuvant therapy is allowed. If relapse or metastasis occurs during or within six months after completion of adjuvant/neoadjuvant therapy, it is considered a failure of first-line chemotherapy for progressive disease. c. For patients with RAS/RAF wild-type tumors, the use of an EGFR inhibitor is not required.)
  • At least one measurable lesion, with the longest diameter ≥10 mm on spiral CT or ≥20 mm on conventional CT (RECIST 1.1 criteria).
  • ECOG performance status of 0-2.
  • Life expectancy of ≥12 weeks.
  • Adequate bone marrow, hepatic, and renal function measured within the screening period prior to randomization: absolute neutrophil count (ANC) ≥1.5 × 109 /L, hemoglobin ≥ 8.0 g/dL, platelet count ≥ 75 × 109 /L, total bilirubin \<1.5 × ULN, ALT and AST \<2.5 × ULN (≤5 × ULN for patients with liver involvement), serum creatinine ≤1.5 × ULN, and creatinine clearance ≥50 mL/min.
  • Women of childbearing potential must use effective contraception.
  • Voluntarily participating in this study, signing the informed consent form, understanding the purpose of the study and the necessary procedures, and willing to participate in this study.

Exclusion

  • Patients who meet any of the following criteria will be excluded from the study:
  • Proteinuria ≥2+ on dipstick or 24-hour urinary protein ≥1.0 g/24 h.
  • Abnormal coagulation function (PT\>16s, APTT\>43s, TT\>21s, Fbg\<2g/L), bleeding tendency, or receiving thrombolysis or anticoagulation therapy.
  • Patients at risk of gastrointestinal bleeding, including those with active digestive ulcers and fecal occult blood (++) and those with histories of black stools or hematemesis within three months.
  • Receiving systemic antitumor therapy, including chemotherapy, signal transduction inhibitors, or immune therapies, within three weeks prior to screening.
  • Patients with uncontrolled hypertension (systolic blood pressure \>140 mmHg, diastolic blood pressure \>90 mmHg) despite antihypertensive medication, grade I or higher coronary heart disease, grade I or higher arrhythmia (including QTc interval prolongation with ≥450 ms for men and ≥470 ms for women), or grade I or higher heart failure.
  • Patients with a history of thrombotic or embolic events requiring treatment within the preceding six months.
  • Patients who have received radiation therapy targeting the selected target lesion.
  • Symptomatic brain or meningeal metastasis.
  • Uncontrolled pleural or peritoneal effusion.
  • Receiving kidney dialysis.
  • Serious or uncontrolled infection.
  • Pregnant or lactating women or women of childbearing potential without adequate contraception.
  • Multiple factors affecting oral drug administration (dysphagia, chronic diarrhea, and bowel obstruction).
  • Patients who have been treated with small molecule tyrosine kinase inhibitors containing VEGFR (such as apatinib, fruquintinib, anlotinib, and lenvatinib).
  • Patients who have been treated with TAS-102.
  • Participation in another clinical study within four weeks prior to screening.
  • Patients with comorbidities that could seriously endanger patients' safety or affect their completion of the study.

Key Trial Info

Start Date :

July 1 2023

Trial Type :

INTERVENTIONAL

Allocation :

ESTIMATED

End Date :

July 4 2026

Estimated Enrollment :

101 Patients enrolled

Trial Details

Trial ID

NCT05970705

Start Date

July 1 2023

End Date

July 4 2026

Last Update

August 1 2023

Active Locations (1)

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1

Fudan University Shanghai Cancer Center

Shanghai, Shanghai Municipality, China, 200032