Status:

ACTIVE_NOT_RECRUITING

A Relative Bioavailability and Food Effect Study of TYRA-300-B01 Capsule and Tablet Formulations in Healthy Adult Participants

Lead Sponsor:

Tyra Biosciences, Inc

Conditions:

Healthy

Eligibility:

All Genders

26-55 years

Phase:

PHASE1

Brief Summary

The purpose of this study is to evaluate the relative bioavailability of capsule and tablet formulations of TYRA-300-B01, and to evaluate the safety, tolerability, and food effect of TYRA-300-B01 tabl...

Detailed Description

This is a Phase 1, multi-cohort trial studying TYRA-300-B01, a novel, potent fibroblast growth factor receptor (FGFR) 3-selective tyrosine kinase inhibitor, in healthy, adult participants. The purpose...

Eligibility Criteria

Inclusion

  • Males or females of non-childbearing potential, between 18 and 55 years of age
  • In good health, determined by no clinically significant findings from medical history, 12-lead electrocardiogram (ECG), vital signs, and clinical laboratory assessments
  • Body mass index (BMI) 18 to 32 kg/m\^2 (inclusive)
  • Cohorts 1 and 2 ethnicity requirements: none
  • Cohort 3 ethnicity requirements: first- or second-generation Japanese participants

Exclusion

  • Significant history of any hematological, renal, endocrine, pulmonary, gastrointestinal, cardiovascular, hepatic, psychiatric, neurologic, immunologic, musculoskeletal disease, or allergic disease (as determined by the Investigator)
  • Any ocular condition likely to increase the risk of eye toxicity
  • Gastrointestinal disorders that will affect oral administration or absorption of TYRA-300-B01
  • Females of child-bearing potential and males who plan to father a child while enrolled in this study

Key Trial Info

Start Date :

October 16 2023

Trial Type :

INTERVENTIONAL

Allocation :

ESTIMATED

End Date :

July 1 2025

Estimated Enrollment :

60 Patients enrolled

Trial Details

Trial ID

NCT06006702

Start Date

October 16 2023

End Date

July 1 2025

Last Update

March 26 2025

Active Locations (1)

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Nucleus Network

Melbourne, Victoria, Australia, 3004