Status:

ACTIVE_NOT_RECRUITING

TACTIVE-U: A Study to Learn About the Study Medicine (Vepdegestrant) When Given With Other Medicines in People With Advanced or Metastatic Breast Cancer. (Sub-Study C)

Lead Sponsor:

Pfizer

Collaborating Sponsors:

Arvinas Estrogen Receptor, Inc.

Carrick Therapeutics Limited

Conditions:

Breast Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE1

PHASE2

Brief Summary

The purpose of this study is to learn about the safety and effects of the study medicine called vepdegestrant. The safety and effects of vepdegestrant will be see when given with other medicines. Vepd...

Detailed Description

C4891024 is a prospective, open-label, multicenter, Phase 1b/2 sub-study to evaluate the safety, antitumor activity, and PK of ARV-471 with samuraciclib in the treatment of participants with A/MBC. Th...

Eligibility Criteria

Inclusion

  • Histological or cytological diagnosis of breast cancer. At time of enrollment this must not be amendable to surgical resection with curative intent (≥1% ER+ stained cells as per local practice on the most recent tumor biopsy HER2- tumor by IHC or in-situ hybridization per ASCO/CAP).
  • prior anticancer therapies: up to 2 lines of prior therapies for advanced/metastatic disease; 1 line of any CDK4/6 inhibitor-based regimen is required (in any setting eg adjuvant, metastatic)
  • at least 1 measurable lesion as defined by RECIST v1.1.
  • ECOG PS ≤1.

Exclusion

  • visceral crisis at risk of life-threatening complications in the short term
  • known history of drug-induced pneumonitis or other significant symptomatic deterioration of lung functions.
  • newly diagnosed brain metastases, or symptomatic CNS metastases, carcinomatous meningitis, or leptomeningeal disease. Participants with a history of CNS metastases or cord compression are eligible if they have been definitively treated, clinically stable and discontinued anti-seizure medications and corticosteroids for at least 28 days prior to enrollment in the of study.
  • history of any other tumor malignancies within the past 3 years, except for the following: (1) adequately treated basal or squamous cell carcinoma of the skin; (2) curatively treated in situ carcinoma of the cervix.
  • inflammatory breast cancer
  • impaired cardiovascular function or clinically significant cardiovascular diseases
  • concurrent administration of medications, food, or herb supplements that are strong inhibitors/inducers of CYP3A, strong CYP2D6 inhibitors and drugs known to predispose to Torsade de Pointes or QT interval prolongation.
  • renal impairment, not adequate liver function and/or bone marrow function
  • known active infection

Key Trial Info

Start Date :

January 10 2024

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

April 30 2026

Estimated Enrollment :

11 Patients enrolled

Trial Details

Trial ID

NCT06125522

Start Date

January 10 2024

End Date

April 30 2026

Last Update

October 31 2025

Active Locations (21)

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Page 1 of 6 (21 locations)

1

Highlands Oncology Group

Fayetteville, Arkansas, United States, 72703

2

Highlands Oncology Group

Rogers, Arkansas, United States, 72758

3

Highlands Oncology Group

Springdale, Arkansas, United States, 72762

4

Clinical and Translational Research Unit (CTRU)

Palo Alto, California, United States, 94304