Status:

RECRUITING

Safety, Tolerability, Pharmacokinetics, and Preliminary Efficacy of BTX-9341 in Advanced and/or Metastatic Breast Cancer

Lead Sponsor:

Biotheryx, Inc.

Conditions:

Breast Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

The purpose of this study is to test BTX-9341 alone or in combination with fulvestrant (a currently marketed medication for breast cancer) in participants with advanced and/or metastatic hormone recep...

Detailed Description

This first-in-human (FIH), Phase 1 study of BTX-9341 is multicenter, nonrandomized, and open-label to evaluate the safety, tolerability, pharmacokinetics (PK), and preliminary efficacy of BTX-9341 in ...

Eligibility Criteria

Inclusion

  • Metastatic and/or locally advanced HR+/HER2- breast cancer (dose escalation: measurable disease and/or at least 1 lytic or mixed \[lytic + sclerotic\] bone lesion that can be assessed by CT or MRI or non-measurable disease \[including bone lesions\]; dose expansion: measurable disease)
  • Dose escalation: (a) received not more than 1 chemotherapy in the metastatic/advanced setting; (b) no limit to the lines of endocrine therapy (monotherapy or combination therapy) in the metastatic setting; (c) received CDK4/6 inhibitor therapy
  • Dose expansion: (a) received not more than 1 chemotherapy in metastatic/advanced setting; (b) received not more than 2 lines of endocrine therapy (monotherapy or combination therapy) and must have been on prior endocrine therapy for at least 6 months before progression; (c) received at most 2 lines of CDK4/6 inhibitor therapy (1 in the adjuvant setting and 1 in the metastatic setting) and must have been on prior CDK4/6 inhibitor therapy for at least 6 months
  • Acceptable hematologic function
  • ANC ≥ 1500 per mL. Note: Use of growth-factors to maintain the ANC criterion is prohibited.
  • Platelet count ≥ 100,000 per mL. Note: Use of transfusions or thrombopoietic agents to achieve the baseline platelet count criterion is prohibited.
  • Hemoglobin ≥ 9.0 g/dL. Note: Packed red blood cell transfusion is allowed up to 14 days prior to trial entry.
  • Acceptable liver function
  • Bilirubin ≤ 2.0 × institutional upper limit of normal (ULN) (or \< 3.0 × institutional ULN if Gilbert's disease is present)
  • Alanine transaminase (ALT)/aspartate aminotransferase (AST) ≤ 3.0 × institutional ULN (≤ 5.0 × institutional ULN if liver metastases present)
  • Alkaline phosphatase ≤ 2.5 × institutional ULN (≤ 5.0 × institutional ULN if bone or liver metastases present)
  • Able and willing to sign informed consent
  • Meets all study requirements in the opinion of the Investigator

Exclusion

  • RB1 (retinoblastoma) gene mutation
  • Symptomatic visceral disease
  • Clinical evidence or history of central nervous system metastasis
  • Abnormalities in coagulation, such as bleeding diathesis, or treatment with anticoagulants precluding injections of fulvestrant or luteinizing hormone-releasing hormone (LHRH) agonist

Key Trial Info

Start Date :

July 3 2024

Trial Type :

INTERVENTIONAL

Allocation :

ESTIMATED

End Date :

December 31 2027

Estimated Enrollment :

82 Patients enrolled

Trial Details

Trial ID

NCT06515470

Start Date

July 3 2024

End Date

December 31 2027

Last Update

June 6 2025

Active Locations (6)

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Page 1 of 2 (6 locations)

1

Biotheryx Investigative Site

Rochester, Minnesota, United States, 55905

2

Biotheryx Investigative Site

Omaha, Nebraska, United States, 68130

3

Biotheryx Investigative Site

Houston, Texas, United States, 77030

4

Biotheryx Investigative Site

San Antonio, Texas, United States, 78229