Status:

RECRUITING

A Study on Efficacy and Safety of HST101 in Chinese Patients with Hypercholesterolemia

Lead Sponsor:

Hasten Biopharmaceutical Co., Ltd.

Conditions:

Hypercholesterolemia

Dyslipidemias

Eligibility:

All Genders

18+ years

Phase:

PHASE3

Brief Summary

This randomized study is to assess LDL-C reductions at Week 12 with monthly (Q4W \[≤31 days\]) dosing of HST101 (lerodalcibep) 300 mg administered subcutaneously (SC) compared to placebo in patients w...

Detailed Description

This is a multi-center, randomized, double-blind, placebo-controlled Phase 3 study. Participants who fulfill the inclusion and exclusion criteria will be enrolled at up to 35 study sites in mainland C...

Eligibility Criteria

Inclusion

  • Provision of written and signed informed consent form prior to any study-specific procedure;
  • Male or female participants ≥18 years of age at the screening visit;
  • Body weight ≥ 40 kg and body mass index (BMI) ≥18 and ≤35 kg/m2;
  • On a stable diet and lipid-lowering oral drugs (such as statins, ezetimibe or Hybutimibe, omega-3 compounds, fenofibrate, nicotinic acid, etc.) for at least 4 weeks prior to the first drug administration
  • LDL-C≥1.8 mmol/L (70 mg/dL) and TG≤4.52 mmol/L (400 mg/dL) at screening for ASCVD patients or those at very (ultra)-high risk for ASCVD, including patients with HeFH; LDL-C ≥ 2.6 mmol/L (100 mg/dL) and TG ≤ 4.52 mmol/L (400 mg/dL) at screening for patients at high-risk for ASCVD including patients with HeFH;
  • Patients on a PCSK9 mAb at a dose of 75 mg, 140 mg, or 150 mg Q2W must undergo a washout period of ≥6 weeks after the last dose; for those on 300 mg or 420 mg Q4W, the washout period is ≥10 weeks following last dose;
  • Female of childbearing potential must have a negative pregnancy test at the last screening visit and consent to use highly effective contraceptives during the trial and 3 months after the last dose of investigational drug.

Exclusion

  • Documented history of homozygous familial hypercholesterolemia (HoFH);
  • Estimated glomerular filtration rate (eGFR)\<30 mL/min/1.73m2;
  • Active liver disease or hepatic dysfunction, history of liver transplant, and/or ALT or AST \>2.5 × ULN at screening;
  • Poorly controlled thyroid disorder including hypothyroidism or hyperthyroidism;
  • Poorly controlled Type 1 or Type 2 diabetes mellitus defined as fasting blood glucose ≥11.0 mmol/L (200 mg/dL) and glycosylated hemoglobin (HbA1c) ≥ 9%;
  • Serious arrhythmia, MI, unstable angina pectoris, PCI, CABG, implantable cardioverter defibrillator, aortic valve surgery or stroke within 3 months prior to the first dose;
  • Planned cardiac surgery or revascularization during the study period;
  • New York Heart Association (NYHA) Class III-IV heart failure;
  • Pregnant or lactating women;
  • Poorly controlled hypertension (SBP≥160 mmHg or DBP≥100 mmHg in a sitting position)
  • Unexplained creatine kinase (CK) \> 5 x ULN (retested once is needed if suspected to be related to excessive exercise or abnormal activity);
  • LDL apheresis or plasma exchange within 2 months prior to the first dose;
  • HIV, Treponema pallidum, or HCV antibody test positive, or HBV-DNA \>ULN at screening;
  • History of prescription drug abuse, illicit drug use or alcohol abuse within 6 months prior to screening;
  • History of any major drug allergy, including allergy to protein biologics;
  • Participate another clinical trial within 30 days or less than 5 half-lifes (drug) before screening, whichever is longer

Key Trial Info

Start Date :

November 16 2024

Trial Type :

INTERVENTIONAL

Allocation :

ESTIMATED

End Date :

May 1 2026

Estimated Enrollment :

210 Patients enrolled

Trial Details

Trial ID

NCT06568471

Start Date

November 16 2024

End Date

May 1 2026

Last Update

February 6 2025

Active Locations (18)

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Page 1 of 5 (18 locations)

1

Beijing Anzhen Hospital of Capital Medical University

Beijing, Beijing Municipality, China

2

Beijing Luhe Hospital, Capital Medical Univeristy

Beijing, Beijing Municipality, China

3

Beijing Tsinghua Changgeng Hospital

Beijing, Beijing Municipality, China

4

Fuwai Hospital, CAMS & PUMC

Beijing, Beijing Municipality, China