Actively Recruiting

Phase 2
Phase 3
Age: 0Years - 100Years
All Genders
ID05948943

A Two-stage Double-blind, Randomized, Placebo-controlled Study to Assess the Efficacy, Safety and Pharmacokinetics of Alpelisib in Pediatric and Adult Patients With Lymphatic Malformations Associated With a PIK3CA Mutation

Led by Novartis Pharmaceuticals · Updated on 2026-06-02

232

Participants Needed

57

Research Sites

256 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating alpelisib film-coated tablets (FCT) in participants with lymphatic malformations (LyM) associated with a PIK3CA mutation. The study aims to assess how alpelisib affects radiological response and symptom severity compared to placebo. This phase II/III, multi-center trial includes both pediatric and adult participants with this genetic mutation. The study has two stages. Stage 1 is a 24-week open-label phase to select doses of alpelisib for adults (18 years and older) and children aged 6 to 17 years, followed by an extension. Participants are randomized to different doses based on age. Stage 2 is a 24-week randomized, double-blind, placebo-controlled phase to confirm efficacy and safety of the selected dose in adults and children 6 to 17 years old, followed by an open-label extension. Additionally, children aged 0 to 5 years participate in a 24-week open-label phase with dose 3 of alpelisib, with an extension if they enroll. Participants will undergo regular assessments including radiological evaluations, symptom severity scales, and quality of life questionnaires up to approximately 8 years. Safety and response are monitored throughout both stages. The primary outcome is the radiological response rate at Week 24 of Stage 2. Other measures include patient and investigator impressions of change, symptom and lesion assessments, and alpelisib blood levels. Participants are expected to take study medication orally and attend scheduled visits during the study period.

CONDITIONS

Brief Title

Alpelisib in Pediatric and Adult Patients With Lymphatic Malformations Associated With a PIK3CA Mutation.

Who Can Participate

Age: 0Years - 100Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Signed informed consent and assent when applicable
  • Willingness to remain at the clinical site and follow study schedules and restrictions
  • Physician-confirmed diagnosis of symptomatic lymphatic malformations not included under PROS criteria
  • Not a candidate for or unwilling to receive non-drug therapies like surgery, sclerotherapy, or embolization until after Week 24
  • Evidence of a somatic mutation in the PIK3CA gene before randomization
  • At least one measurable lymphatic malformation lesion confirmed before randomization
  • Ability to ingest study medication orally or via feeding tube as assessed within 7 days before treatment start
Not Eligible

You will not qualify if you...

  • Physician-confirmed diagnosis of PROS at the time of informed consent
  • Diagnosis of Central Conducting Lymphatic Anomaly, General Lymphatic Anomaly, Gorham-Stout disease, or Kaposiform lymphangiomatosis
  • History of Stevens-Johnson syndrome, erythema multiforme, or toxic epidermal necrolysis
  • Established type I diabetes or uncontrolled type II diabetes
  • Previous treatment with alpelisib or other PI3K inhibitors for more than 2 weeks
  • Other exclusion criteria may apply

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Stage 1 Treatment

Duration - 24 weeks

Participants aged 6 years and older receive alpelisib at assigned doses in an open-label fashion to determine optimal dosing over 24 weeks.

Visits during 24 weeks of treatment

Stage 2 Treatment

Duration - 24 weeks

Participants aged 6 years and older are randomized to receive alpelisib at the selected confirmatory dose or placebo for 24 weeks in a double-blind manner. Pediatric participants aged 0-5 years receive open-label alpelisib dosing for 24 weeks.

Visits during 24 weeks of treatment

Extension Phase

Duration - Duration varies based on participant continuation

Participants who complete Stage 1 or Stage 2 may continue receiving alpelisib in an open-label extension phase to further assess safety and efficacy.

Visits as scheduled during extension

Trial Site Locations

Total: 57 locations

1

UCSF Benioff Children s Hospital

Oakland, California, United States, 94609

Actively Recruiting

2

Lucile Packard Childrens Hosp

Palo Alto, California, United States, 94304

Actively Recruiting

3

Childrens National Medical Center

Washington D.C., District of Columbia, United States, 20010-2970

Actively Recruiting

4

Nemours Childrens Clinic

Jacksonville, Florida, United States, 32207

Actively Recruiting

5

Childrens Hosp Boston Dept of Heme

Boston, Massachusetts, United States, 02115

Actively Recruiting

6

WA Uni School Of Med

St Louis, Missouri, United States, 63110

Actively Recruiting

7

Cinn Children Hosp Medical Center

Cincinnati, Ohio, United States, 45229-3039

Actively Recruiting

8

Univ Hospital Of Cleveland

Cleveland, Ohio, United States, 44106

Actively Recruiting

9

Cleveland Clinic Foundation

Cleveland, Ohio, United States, 44195

Actively Recruiting

10

Nationwide Children s Hospital

Columbus, Ohio, United States, 43205

Actively Recruiting

11

Oregon Health Science University

Portland, Oregon, United States, 97239

Actively Recruiting

12

CHOP Abramson Pediatric Resch Ctr

Philadelphia, Pennsylvania, United States, 19104

Actively Recruiting

13

Childrens Hosp Pittsburgh UPMC

Pittsburgh, Pennsylvania, United States, 15224

Actively Recruiting

14

Baylor College Of Medicine

Houston, Texas, United States, 77030

Actively Recruiting

15

U of TX Health Science Ct

Houston, Texas, United States, 77030

Actively Recruiting

16

Childrens Hospital and Regional Medical Center

Seattle, Washington, United States, 98105

Actively Recruiting

17

Novartis Investigative Site

CABA, Buenos Aires, Argentina, C1181ACH

Actively Recruiting

18

Novartis Investigative Site

CABA, Buenos Aires, Argentina, C1425BEA

Actively Recruiting

19

Novartis Investigative Site

Capital Federal, Argentina, C1023AAB

Actively Recruiting

20

Novartis Investigative Site

Sydney, New South Wales, Australia, 2010

Actively Recruiting

21

Novartis Investigative Site

Sydney, New South Wales, Australia, 2031

Actively Recruiting

22

Novartis Investigative Site

Brisbane, Queensland, Australia, 4101

Actively Recruiting

23

Novartis Investigative Site

Brussels, Belgium, 1200

Actively Recruiting

24

Novartis Investigative Site

Angers, France, 49933

Actively Recruiting

25

Novartis Investigative Site

Bordeaux, France, 33076

Actively Recruiting

26

Novartis Investigative Site

Bron, France, 69677

Actively Recruiting

27

Novartis Investigative Site

Caen, France, 14033

Actively Recruiting

28

Novartis Investigative Site

Dijon, France, 21000

Actively Recruiting

29

Novartis Investigative Site

Lille, France, 59000

Actively Recruiting

30

Novartis Investigative Site

Marseille, France, 13885

Actively Recruiting

31

Novartis Investigative Site

Montpellier, France, 34295

Actively Recruiting

32

Novartis Investigative Site

Paris, France, 75010

Actively Recruiting

33

Novartis Investigative Site

Paris, France, 75015

Actively Recruiting

34

Novartis Investigative Site

Toulouse, France, 31054

Actively Recruiting

35

Novartis Investigative Site

Tours, France, 37044

Actively Recruiting

36

Novartis Investigative Site

Freiburg im Breisgau, Baden-Wurttemberg, Germany, 79106

Actively Recruiting

37

Novartis Investigative Site

Mannheim, Baden-Wurttemberg, Germany, 68305

Withdrawn

38

Novartis Investigative Site

Cologne, North Rhine-Westphalia, Germany, 50937

Actively Recruiting

39

Novartis Investigative Site

Leipzig, Saxony, Germany, 04103

Actively Recruiting

40

Novartis Investigative Site

Berlin, Germany, 13353

Actively Recruiting

41

Novartis Investigative Site

Ulm, Germany, 89081

Actively Recruiting

42

Novartis Investigative Site

Bologna, BO, Italy, 40138

Actively Recruiting

43

Novartis Investigative Site

Milan, MI, Italy, 20122

Actively Recruiting

44

Novartis Investigative Site

Roma, RM, Italy, 00165

Actively Recruiting

45

Novartis Investigative Site

Roma, RM, Italy, 00168

Actively Recruiting

46

Novartis Investigative Site

Torino, TO, Italy, 10126

Actively Recruiting

47

Novartis Investigative Site

Naples, Italy, 80122

Actively Recruiting

48

Novartis Investigative Site

Nijmegen, Gelderland, Netherlands, 6500HB

Actively Recruiting

49

Novartis Investigative Site

Rotterdam, South Holland, Netherlands, 3015 GD

Actively Recruiting

50

Novartis Investigative Site

Palma, Balearic Islands, Spain, 07120

Actively Recruiting

51

Novartis Investigative Site

Esplugues, Barcelona, Spain, 08950

Actively Recruiting

52

Novartis Investigative Site

L'Hospitalet de Llobregat, Barcelona, Spain, 08907

Actively Recruiting

53

Novartis Investigative Site

A Coruña, Spain, 15006

Actively Recruiting

54

Novartis Investigative Site

Barcelona, Spain, 08035

Actively Recruiting

55

Novartis Investigative Site

Madrid, Spain, 28009

Actively Recruiting

56

Novartis Investigative Site

Madrid, Spain, 28046

Actively Recruiting

57

Novartis Investigative Site

Lausanne, Switzerland, 1011

Actively Recruiting

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Research Team

N

Novartis Pharmaceuticals

N

Novartis Pharmaceuticals

How is the study designed?

Study Type

INTERVENTIONAL

Masking

QUADRUPLE

Allocation

RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

9

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