Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
NCT04421820

BOLD-100 in Combination With FOLFOX for the Treatment of Advanced Solid Tumours

Led by Bold Therapeutics, Inc. · Updated on 2026-05-04

220

Participants Needed

18

Research Sites

313 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

BOLD-100 is an intravenously administered sterile solution containing the ruthenium-based small molecule. BOLD-100 has been shown to preferentially decrease the expression of GRP78 in tumour cells and ER stressed cells when compared to normal cells. BOLD-100 will be combined with cytotoxic FOLFOX chemotherapy in this study, with a dose escalation cohort to ensure tolerability and safety, followed by a cohort expansion phase.

CONDITIONS

Official Title

BOLD-100 in Combination With FOLFOX for the Treatment of Advanced Solid Tumours

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Be 18 years or older
  • Be male or non-pregnant female and agree to follow contraceptive requirements
  • Have histologically or cytologically confirmed metastatic or unresectable gastrointestinal tumors
  • For Arm VII, have received only 1 prior metastatic therapy line
  • Have measurable disease by RECIST v1.1
  • Have expected survival of at least 16 weeks
  • Be ambulatory with ECOG performance score of 0 or 1
  • Have adequate organ function
  • Be on stable doses of medications affecting liver or kidney drug processing
  • Be fully informed about the illness and study and sign consent
  • For Arm VII, have BRAF wild-type tumor status
Not Eligible

You will not qualify if you...

  • Neuropathy greater than grade 2
  • Previous intolerance or severe reaction to fluorouracil or oxaliplatin
  • Stroke within 6 months before starting treatment
  • History or presence of central nervous system metastases or leptomeningeal tumors
  • Serious medical conditions that could worsen with treatment or limit compliance
  • History of serious heart disease
  • Bleeding in lungs, brain, or significant gastrointestinal bleeding within 6 months before treatment
  • Any other cancer within 3 years before starting treatment
  • Active gastrointestinal disease with malabsorption
  • Non-healing wounds, fractures, ulcers, or symptomatic peripheral vascular disease
  • Radiation therapy or surgery within 4 weeks before treatment start
  • Weight loss over 10% in past 3 months before treatment
  • HIV infection on combination anti-retroviral therapy
  • Use of other investigational or anti-cancer therapy within 4 weeks before treatment
  • Currently breastfeeding
  • Dihydropyrimidine Dehydrogenase (DPD) deficiency
  • Current or prior use of strong DPD inhibitors
  • For Arm VII, prior exposure to BOLD-100
  • For Arm VII, tumors with microsatellite instability-high (MSI-H)
  • For Arm VII, concurrent monoclonal antibody therapy for metastatic colorectal cancer (anti-EGFR, anti-VEGF, or anti-HER2)

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 18 locations

1

University of California, Los Angeles

Santa Monica, California, United States, 90095

Completed

2

Moffitt Cancer Center

Tampa, Florida, United States, 33612

Completed

3

Cross Cancer Institue

Edmonton, Alberta, Canada

Actively Recruiting

4

Juravinski Cancer Centre

Hamilton, Ontario, Canada

Actively Recruiting

5

The Ottawa Hospital Cancer Centre

Ottawa, Ontario, Canada

Actively Recruiting

6

Princess Margaret Cancer Centre

Toronto, Ontario, Canada

Actively Recruiting

7

Jewish General Hospital

Montreal, Quebec, Canada

Actively Recruiting

8

McGill University Health Centre Glen Site

Montreal, Quebec, Canada

Actively Recruiting

9

Universitatsklinikum Bonn

Bonn, Germany

Actively Recruiting

10

University Hospital of Ulm

Ulm, Germany

Actively Recruiting

11

Mater Miserecordiae University Hospital

Dublin, Ireland

Actively Recruiting

12

St. James Hospital

Dublin, Ireland

Actively Recruiting

13

St. Vincent's University Hospital

Dublin, Ireland

Actively Recruiting

14

National Cancer Center

Goyang, South Korea

Actively Recruiting

15

Kangbuk Samsung Hospital

Seoul, South Korea

Actively Recruiting

16

Samsung Medical Center

Seoul, South Korea

Actively Recruiting

17

Seoul National University Hospital

Seoul, South Korea

Actively Recruiting

18

Severance Hospital - Yonsei University

Seoul, South Korea

Actively Recruiting

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Research Team

M

Michelle Jones

CONTACT

J

Jim Pankovich

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

9

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