Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
ID03328078

Open-Label Dose Escalation and Expansion Trial of Emavusertib (CA-4948) in Adults with Relapsed or Refractory Primary Central Nervous System Lymphoma

Led by Curis, Inc. · Updated on 2026-04-16

152

Participants Needed

45

Research Sites

8 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating the safety, how the body processes the drugs (pharmacokinetics), and the anti-cancer effects of oral emavusertib alone or combined with ibrutinib in adults with relapsed or refractory blood cancers, specifically primary central nervous system lymphoma (PCNSL). This multi-center, open-label trial includes several parts to study these treatments in different patient groups, including those who have progressed after previous therapies and those new to certain treatments. The study is sponsored by Curis, Inc. and spans from initial dose-finding to assessing response rates and safety. The trial is conducted in four parts. Part A1 involved increasing doses of emavusertib alone to find a safe dose. Part A2 tested emavusertib combined with ibrutinib at specified doses. Part B includes two groups of participants with PCNSL who progressed on a Bruton tyrosine kinase inhibitor (BTKi), receiving emavusertib at either 100 mg or 200 mg twice daily plus ibrutinib daily in 28-day cycles. Part C involves three groups of participants with PCNSL new to BTKi treatment, randomly assigned to emavusertib alone, ibrutinib alone, or their combination, with treatment cycles of 28 days continuing as tolerated. Participants will take study drugs orally and undergo regular monitoring for safety and treatment effects. Researchers will evaluate side effects, determine maximum tolerated doses, and measure response rates and durations. Pharmacokinetic profiles of both drugs will be assessed over months. The trial includes assessments of tumor progression and survival, with follow-ups lasting up to several years. Participants' health status and response to treatment will be carefully tracked throughout the study.

CONDITIONS

Brief Title

CA-4948-101: Open-Label, Dose Escalation and Expansion Trial of Emavusertib (CA-4948) in Relapsed or Refractory Primary Central Nervous System Lymphoma (R/R PCNSL)

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Males and females aged 18 years or older
  • Life expectancy of at least 3 months
  • Eastern Cooperative Oncology Group (ECOG) Performance Status of 0, 1, or 2
  • Histopathologically confirmed diagnosis of primary central nervous system lymphoma (PCNSL), with typical imaging if biopsy not available
  • For parenchymal lesions, presence of at least one measurable target lesion between 10 mm and 40 mm on brain MRI or CT scan within 28 days prior to treatment
  • For leptomeningeal involvement, cerebrospinal fluid analysis with or without spine imaging within 28 days prior to treatment
Not Eligible

You will not qualify if you...

  • Participants with only intraocular PCNSL without brain lesion or cerebrospinal fluid involvement
  • Participants with T-cell lymphoma, systemic lymphoma, or non-CNS lymphoma metastatic to the CNS
  • Evidence of systemic lymphoma confirmed by PET or CT scan of chest, abdomen, and pelvis
  • Prior history of malignancies other than lymphoma (except certain skin or cervical/breast cancers) unless disease-free for 3 or more years
  • Active malignancy other than PCNSL requiring systemic therapy
  • Previous Bruton tyrosine kinase inhibitor (BTKi) treatment in Part C
  • History of severe rhabdomyolysis without full recovery
  • Need for urgent therapy due to uncontrolled tumor mass or edema
  • External beam radiation to the CNS within 28 days prior to treatment
  • Recent use of investigational drugs within 28 days or 5 half-lives before treatment
  • Allogeneic hematopoietic stem cell transplant within 60 days prior to treatment or ongoing graft-versus-host disease requiring immunosuppressive medication adjustments
  • Prior systemic anti-cancer treatments within 14 days or 5 half-lives before treatment (with exceptions for certain BTKi use in Part B only)
  • History of hypersensitivity or anaphylaxis to emavusertib, ibrutinib, or their components

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Treatment

Duration - Up to 66 months

Participants receive oral emavusertib alone or in combination with oral ibrutinib in repeated 28-day treatment cycles to evaluate safety, tolerability, and efficacy.

Repeated visits every 28 days during treatment cycles

Trial Site Locations

Total: 45 locations

1

St. Joseph's Hospital and Medical Center

Phoenix, Arizona, United States, 85013

Actively Recruiting

2

Mayo Clinic

Phoenix, Arizona, United States, 85054

Completed

3

City of Hope

Duarte, California, United States, 91010

Actively Recruiting

4

Providence St. John's Health Center

Santa Monica, California, United States, 90404

Actively Recruiting

5

UCLA Department of Medicine - Hematology/Oncology

Santa Monica, California, United States, 90404

Withdrawn

6

Smilow Cancer Hospital at Yale-New Haven

New Haven, Connecticut, United States, 06510

Completed

7

Mayo Clinic

Jacksonville, Florida, United States, 32224

Actively Recruiting

8

Northwestern Memorial Hospital

Chicago, Illinois, United States, 60611

Actively Recruiting

9

Dana Farber Cancer Institute

Boston, Massachusetts, United States, 02215

Actively Recruiting

10

Mayo Clinic

Rochester, Minnesota, United States, 55905

Actively Recruiting

11

Fred and Pamela Buffett Cancer Center

Omaha, Nebraska, United States, 68198

Actively Recruiting

12

Hackensack University Medical Center

Hackensack, New Jersey, United States, 07601

Completed

13

Roswell Park Comprehensive Cancer Center

Buffalo, New York, United States, 14263

Actively Recruiting

14

Mt Sinai

New York, New York, United States, 10029

Actively Recruiting

15

Columbia University Irving Medical Center

New York, New York, United States, 10032

Withdrawn

16

Memorial Sloan Kettering Cancer Center

New York, New York, United States, 10065

Actively Recruiting

17

Duke University Medical Center, Duke Cancer Center

Durham, North Carolina, United States, 27710

Actively Recruiting

18

Cleveland Clinic

Cleveland, Ohio, United States, 44195

Actively Recruiting

19

Providence Neurological Specialties West

Portland, Oregon, United States, 97225

Actively Recruiting

20

Hospital of the University of Pennsylvania

Philadelphia, Pennsylvania, United States, 19104

Completed

21

UPMC Hilman Cancer Center

Pittsburgh, Pennsylvania, United States, 15232

Actively Recruiting

22

University of Tennessee Medical Center

Knoxville, Tennessee, United States, 37920

Completed

23

UT Southwestern Medical Center

Dallas, Texas, United States, 75235

Active, Not Recruiting

24

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States, 77030

Actively Recruiting

25

Huntsman Cancer Institute, University of Utah

Salt Lake City, Utah, United States, 84112

Actively Recruiting

26

Swedish Cancer Institute

Seattle, Washington, United States, 98104

Completed

27

University of Washington Medical Center

Seattle, Washington, United States, 98195

Actively Recruiting

28

Všeobecná fakultní nemocnice v Praze

Prague, Czechia

Actively Recruiting

29

Institut Bergonie

Bordeaux, France

Actively Recruiting

30

Hopital de la Timone

Marseille, France

Actively Recruiting

31

Hospital Pitie Salpetriere

Paris, France

Actively Recruiting

32

Institut Curie Hospital

Paris, France

Actively Recruiting

33

Hematology Department Soroka UMC / Heanatology Department

Beersheba, Israel

Actively Recruiting

34

Rambam Medical Center

Haifa, Israel

Actively Recruiting

35

Hadassah Medical Center / Ein-Carem

Jerusalem, Israel

Actively Recruiting

36

Università di Torino Croce e Carle

Cuneo, Italy

Actively Recruiting

37

SODc Ematologia Azienda Ospedaliera Universitaria Careggi

Florence, Italy

Actively Recruiting

38

IRST - Istituto Scientifico Romagnolo per lo Studio e la Cura dei Tumori

Meldola, Italy

Actively Recruiting

39

IRCCS San Raffaele Scientific Institute

Milan, Italy

Actively Recruiting

40

Uniwersyteckie Centrum Kliniczne Osrodek Badan Klinicznych Wczesnych Faz

Gdansk, Poland

Actively Recruiting

41

Oddzial Kliniczny Hematologii

Krakow, Poland

Withdrawn

42

NarodowyInstytutu Onkologii im. Marii Sklodowskiej-Curie-Panstwowy Instytutu Badawczy

Warsaw, Poland

Actively Recruiting

43

University Hospital Vall d'Hebron

Barcelona, Spain

Actively Recruiting

44

MD Anderson Cancer Center Madrid

Madrid, Spain

Actively Recruiting

45

Hospital Universitario Virgen del Rocio

Seville, Spain

Actively Recruiting

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Research Team

A

Ahmed Hamdy, MD

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

4

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