Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
ID06863272

Phase 1/2 Study of Ifinatamab Deruxtecan Alone or with Other Treatments for Metastatic Castration-Resistant Prostate Cancer

Led by Merck Sharp & Dohme LLC · Updated on 2026-05-29

360

Participants Needed

80

Research Sites

N/A

Total Duration

On this page

Sponsors

M

Merck Sharp & Dohme LLC

Lead Sponsor

D

Daiichi Sankyo

Collaborating Sponsor

AI-Summary

What this Trial Is About

Researchers are evaluating the safety and effectiveness of ifinatamab deruxtecan (I-DXd), alone or combined with other treatments, for people with metastatic castration-resistant prostate cancer (mCRPC). This study aims to find a safe dose of I-DXd in combination with other therapies and to monitor prostate specific antigen (PSA) levels during treatment. It is a phase 1/2, open-label study under the MK-2400-U01 master protocol. Participants may receive one of several treatments: docetaxel given intravenously every three weeks for up to 10 cycles; I-DXd alone administered intravenously every three weeks until side effects, disease progression, death, or withdrawal; I-DXd combined with MK-5684 taken orally; or I-DXd combined with an androgen receptor pathway inhibitor (either abiraterone acetate or enzalutamide) taken orally. The study includes a dose escalation phase followed by longer treatment periods. During the study, participants will be monitored for treatment side effects, PSA response, and other outcomes such as disease progression and survival over several years. Researchers will track adverse events, dose-limiting toxicities, and reasons for stopping treatment. The total follow-up may last up to about 54 months, with regular assessments including safety, efficacy, and quality of life measures.

CONDITIONS

Brief Title

A Clinical Study of Ifinatamab Deruxtecan Based Treatment Combinations or as Monotherapy to Treat Metastatic Castrate Resistant Prostate Cancer (mCRPC) (MK-2400-01A/IDeate-Prostate02)

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Histologically or cytologically confirmed adenocarcinoma of the prostate without small cell histology
  • Evidence of metastatic prostate cancer progression during androgen deprivation therapy within 6 months before screening
  • Current metastatic disease
  • Prior treatment with 1 or 2 androgen receptor pathway inhibitors with progression during or after treatment
  • Stable bone resorptive therapy for 4 or more weeks before randomization if applicable
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 to 1 within 10 days before randomization
  • Prior treatment with poly-ADP-ribose polymerase inhibitors if indicated or ineligible for such treatment
Not Eligible

You will not qualify if you...

  • History of interstitial lung disease or pneumonitis requiring steroids, or current or suspected ILD/pneumonitis
  • Severe pulmonary compromise from other lung illnesses
  • Uncontrolled or significant cardiovascular disease
  • History of pituitary dysfunction
  • Poorly controlled diabetes mellitus
  • History or current adrenal insufficiency (e.g., Addison's disease)
  • Prior treatment with taxane-based chemotherapy for mCRPC
  • Chronic steroid use over 10 mg daily prednisone equivalent except for certain inhaled or topical steroids
  • Radiotherapy within 2 weeks before study start or radiation-related toxicities requiring corticosteroids
  • Active malignancy requiring treatment within past 3 years
  • Active central nervous system metastases or carcinomatous meningitis
  • Active autoimmune disease requiring systemic treatment in past 2 years
  • History of allogeneic tissue or solid organ transplant

AI-Screening

AI-Powered Screening

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 screening and enrollment visit

Treatment

Duration - Varies by treatment; up to several months depending on cycles or until discontinuation criteria are met

Participants receive assigned drug treatments including docetaxel every 3 weeks for up to 10 cycles, or Ifinatamab Deruxtecan alone or combined with MK-5684 or androgen receptor pathway inhibitors until unacceptable toxicity, disease progression, death, or withdrawal.

Visits every 3 weeks corresponding with treatment cycles

Trial Site Locations

Total: 80 locations

1

UCLA Hematology & Oncology ( Site 0003)

Los Angeles, California, United States, 90095

Actively Recruiting

2

University of California-Irvine Medical Center ( Site 0016)

Orange, California, United States, 92868

Actively Recruiting

3

UCSF Medical Center at Mission Bay ( Site 0034)

San Francisco, California, United States, 94158

Actively Recruiting

4

MedStar Georgetown Cancer Institute at MedStar Washington Hospital Center ( Site 0026)

Washington D.C., District of Columbia, United States, 20010

Actively Recruiting

5

Memorial Sloan Kettering Cancer Center ( Site 0006)

New York, New York, United States, 10065

Actively Recruiting

6

UPMC Hillman Cancer Center ( Site 0014)

Pittsburgh, Pennsylvania, United States, 15232

Actively Recruiting

7

The West Clinic, PLLC dba West Cancer Center ( Site 0005)

Germantown, Tennessee, United States, 38138

Actively Recruiting

8

Fred Hutchinson Cancer Center ( Site 0013)

Seattle, Washington, United States, 98109

Actively Recruiting

9

Instituto Alexander Fleming ( Site 0202)

Ciudad Autónoma de Buenos Aires, Buenos Aires, Argentina, C1426ANZ

Actively Recruiting

10

Fundación CORI para la Investigación y Prevención del Cáncer ( Site 0200)

La Rioja, Argentina, F5300COE

Actively Recruiting

11

Macquarie University-MQ Health Clinical Trials Unit ( Site 0801)

Macquarie University, New South Wales, Australia, 2109

Actively Recruiting

12

Liga Norte Riograndense Contra o Câncer ( Site 0271)

Natal, Rio Grande do Norte, Brazil, 59062-000

Actively Recruiting

13

Irmandade da Santa Casa de Misericórdia de Porto Alegre ( Site 0270)

Porto Alegre, Rio Grande do Sul, Brazil, 90020-090

Actively Recruiting

14

Hospital Moinhos de Vento ( Site 0278)

Porto Alegre, Rio Grande do Sul, Brazil, 90035-001

Actively Recruiting

15

Hospital Universitário São Francisco de Assis - Bragança Paulista ( Site 0268)

Bragança Paulista, São Paulo, Brazil, 12916-542

Actively Recruiting

16

Hospital das Clínicas da Faculdade de Medicina de Ribeirão Preto da Universidade de São Paulo (USP) ( Site 0273)

Ribeirão Preto, São Paulo, Brazil, 14048900

Actively Recruiting

17

Fundação Faculdade Regional de Medicina de São José do Rio Preto ( Site 0263)

São José do Rio Preto, São Paulo, Brazil, 15090-000

Actively Recruiting

18

Hospital Alemao Oswaldo Cruz ( Site 0279)

São Paulo, São Paulo, Brazil, 01327-001

Actively Recruiting

19

IPITEC ( Site 0275)

São Paulo, Brazil, 01221-020

Actively Recruiting

20

IBCC - Instituto Brasileiro de Controle do Câncer ( Site 0269)

São Paulo, Brazil, 03102-006

Actively Recruiting

21

BC Cancer - Vancouver Center ( Site 0103)

Vancouver, British Columbia, Canada, V5Z 4E6

Actively Recruiting

22

Sunnybrook Research Institute ( Site 0109)

Toronto, Ontario, Canada, M4N 3M5

Actively Recruiting

23

Princess Margaret Cancer Centre ( Site 0102)

Toronto, Ontario, Canada, M5G 2M9

Actively Recruiting

24

Jewish General Hospital ( Site 0108)

Montreal, Quebec, Canada, H3T 1E2

Actively Recruiting

25

CIUSSS de l Estrie - CHUS - Centre Hosp. Univ. Sherbrooke ( Site 0107)

Sherbrooke, Quebec, Canada, J1H 5N4

Actively Recruiting

26

Clinica Universidad Catolica del Maule ( Site 0236)

Talca, Maule Region, Chile, 3465584

Actively Recruiting

27

FALP ( Site 0232)

Santiago, Region M. de Santiago, Chile, 7500921

Actively Recruiting

28

Centro de Oncología de Precisión ( Site 0241)

Santiago, Region M. de Santiago, Chile, 7560908

Actively Recruiting

29

Bradfordhill ( Site 0231)

Santiago, Region M. de Santiago, Chile, 8420383

Actively Recruiting

30

ONCOCENTRO APYS ( Site 0234)

Viña del Mar, Valparaiso, Chile, 2520598

Actively Recruiting

31

Institut Bergonié - Centre Régional de Lutte Contre Le Cancer de Bordeaux et Sud Ouest ( Site 0498)

Bordeaux, Gironde, France, 33000

Actively Recruiting

32

Centre Oscar Lambret ( Site 0495)

Lille, Nord, France, 59000

Actively Recruiting

33

Institut De Cancerologie De L Ouest ( Site 0494)

Saint-Herblain, Pays de la Loire Region, France, 44800

Actively Recruiting

34

Centre Hospitalier de la Côte Basque ( Site 0496)

Bayonne, Pyrenees-Atlantiques, France, 64100

Actively Recruiting

35

centre hospitalier lyon sud ( Site 0497)

Pierre-Bénite, Rhone, France, 69310

Actively Recruiting

36

NCT ( Site 0528)

Heidelberg, Baden-Wurttemberg, Germany, 69120

Actively Recruiting

37

Universitaetsklinikum Jena ( Site 0525)

Jena, Thuringia, Germany, 07747

Actively Recruiting

38

Universitaetsklinikum Hamburg-Eppendorf ( Site 0524)

Hamburg, Germany, 20246

Actively Recruiting

39

St Vincent's University Hospital ( Site 0463)

Dublin, Dublin, Ireland, D04 T6F4

Actively Recruiting

40

Beaumont Hospital, Dublin ( Site 0465)

Dublin, Ireland, D09 V2N0

Actively Recruiting

41

Tallaght University Hospital ( Site 0462)

Dublin, Ireland, D24 NR0A

Actively Recruiting

42

Rambam Health Care Campus ( Site 0400)

Haifa, Israel, 3109601

Actively Recruiting

43

Hadassah Medical Center ( Site 0404)

Jerusalem, Israel, 9112001

Actively Recruiting

44

Rabin Medical Center ( Site 0402)

Petah Tikva, Israel, 4941492

Actively Recruiting

45

Sheba Medical Center ( Site 0401)

Ramat Gan, Israel, 5265601

Actively Recruiting

46

Sourasky Medical Center ( Site 0403)

Tel Aviv, Israel, 6423906

Actively Recruiting

47

AOU San Luigi Gonzaga di Orbassano ( Site 0434)

Orbassano, Torino, Italy, 10143

Actively Recruiting

48

Azienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia ( Site 0432)

Brescia, Italy, 25123

Actively Recruiting

49

Fondazione IRCCS Istituto Nazionale Dei Tumori ( Site 0431)

Milan, Italy, 20133

Actively Recruiting

50

A.O.U. Federico II di Napoli ( Site 0435)

Naples, Italy, 80131

Actively Recruiting

51

Fondazione Policlinico Universitario Agostino Gemelli ( Site 0433)

Roma, Italy, 00168

Actively Recruiting

52

Ziekenhuis Gelderse Vallei ( Site 0683)

Ede, Gelderland, Netherlands, 6716 RP

Actively Recruiting

53

UMC St. Radboud ( Site 0679)

Nijmegen, Gelderland, Netherlands, 6525 GA

Actively Recruiting

54

Nij Smellinghe ( Site 0684)

Drachten, Provincie Friesland, Netherlands, 9202 NN

Actively Recruiting

55

Auckland City Hospital ( Site 0831)

Auckland, New Zealand, 1023

Actively Recruiting

56

Uniwersytecki Szpital Kliniczny w Poznaniu ( Site 0590)

Poznan, Greater Poland Voivodeship, Poland, 60-355

Actively Recruiting

57

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie - Panstwowy Instytut Badawczy w Warszawie ( Site 0586)

Warsaw, Masovian Voivodeship, Poland, 02-781

Actively Recruiting

58

Uniwersyteckie Centrum Kliniczne ( Site 0588)

Gdansk, Pomeranian Voivodeship, Poland, 80-214

Actively Recruiting

59

Szpital Wojewódzki im. M.Kopernika Oddział Onk. Klinicznej z Pododdziałem Chemioterapii Jednodniowej ( Site 0587)

Koszalin, West Pomeranian Voivodeship, Poland, 75-581

Actively Recruiting

60

Asan Medical Center ( Site 0925)

Songpagu, Seoul, South Korea, 05505

Actively Recruiting

61

Severance Hospital Yonsei University Health System ( Site 0924)

Seoul, South Korea, 03722

Active, Not Recruiting

62

Samsung Medical Center ( Site 0926)

Seoul, South Korea, 06351

Actively Recruiting

63

ICO L Hospitalet ( Site 0617)

L Hospitalet Del Llobregat, Barcelona, Spain, 08908

Actively Recruiting

64

Hospital Universitario Ramon y Cajal ( Site 0620)

Madrid, Spain, 28034

Actively Recruiting

65

Hospital Clinico San Carlos ( Site 0618)

Madrid, Spain, 28040

Actively Recruiting

66

Hospital Universitario 12 de Octubre ( Site 0622)

Madrid, Spain, 28041

Actively Recruiting

67

Hospital Universitario Virgen del Rocio ( Site 0619)

Seville, Spain, 41013

Actively Recruiting

68

Taichung Veterans General Hospital ( Site 0902)

Taichung, Taiwan, 40705

Actively Recruiting

69

Taipei Veterans General Hospital ( Site 0901)

Taipei, Taiwan, 11217

Actively Recruiting

70

Baskent University Dr. Turgut Noyan Research and Training Center ( Site 0650)

Adana, Turkey (Türkiye), 01250

Actively Recruiting

71

Hacettepe Universitesi Tip Fakultesi ( Site 0648)

Ankara, Turkey (Türkiye), 06230

Actively Recruiting

72

Ankara Universitesi Tip Fakultesi Hastanesi ( Site 0653)

Ankara, Turkey (Türkiye), 06620

Actively Recruiting

73

Ankara Bilkent Şehir Hastanesi ( Site 0654)

Ankara, Turkey (Türkiye), 06800

Actively Recruiting

74

Koç Üniversitesi Hastanesi ( Site 0656)

Istanbul, Turkey (Türkiye), 34010

Actively Recruiting

75

Istanbul Universitesi Cerrahpasa ( Site 0649)

Istanbul, Turkey (Türkiye), 34098

Actively Recruiting

76

Recep Tayyip Erdogan University Training and Research Hospital ( Site 0655)

Rize, Turkey (Türkiye), 53020

Actively Recruiting

77

Addenbrooke's Hospital ( Site 0747)

Cambridge, Cambridgeshire, United Kingdom, CB2 2QQ

Actively Recruiting

78

St Bartholomew's Hospital ( Site 0749)

London, London, City of, United Kingdom, EC1A 7BE

Actively Recruiting

79

Royal Free Hospital ( Site 0743)

London, London, City of, United Kingdom, NW3 2QG

Actively Recruiting

80

Royal Marsden Hospital (Sutton) ( Site 0741)

London, Surrey, United Kingdom, SM3 5PT

Actively Recruiting

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Research Team

T

Toll Free Number

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

4

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