Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT07543744

A Comparative Study of Pharmacokinetics, Safety, and Immunogenicity of RPH-030 and Vectibix® in Patients With Metastatic Colorectal Cancer With Wild-type RAS as First-line Therapy in Combination With FOLFIRI

Led by R-Pharm · Updated on 2026-04-22

180

Participants Needed

26

Research Sites

171 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The primary objective of this study is to demonstrate equivalence of pharmacokinetic properties, and comparability of safety and immunogenicity parameters of RPH-030 and Vectibix® following a single (first) intravenous administration to patients with mCRC with wild-type RAS genes as 1-line therapy in combination with FOLFIRI. The additional objective is to perform a pilot evaluation of the efficacy of RPH-030 and Vectibix® following a single (first) intravenous administration to patients with mCRC with wild-type RAS genes as 1-line therapy in combination with FOLFIRI.

CONDITIONS

Official Title

A Comparative Study of Pharmacokinetics, Safety, and Immunogenicity of RPH-030 and Vectibix® in Patients With Metastatic Colorectal Cancer With Wild-type RAS as First-line Therapy in Combination With FOLFIRI

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Signed informed consent form
  • Histologically confirmed metastatic colorectal adenocarcinoma
  • Consent to screening biopsy if archival tissue unavailable
  • Candidates for first-line therapy with metastatic colorectal cancer
  • Wild-type RAS gene status
  • ECOG performance status 0-1
  • At least one measurable lesion per RECIST 1.1 (excluding single bone lesions)
  • Recovery from prior therapy toxicities to Grade 1 or less (except non-impacting chronic events)
  • Serum magnesium ≥ 0.66 mmol/L, calcium ≥ 2.15 mmol/L, potassium ≥ 3.5 mmol/L at randomization
  • Life expectancy of at least 13 weeks
  • Agreement to use effective contraception or abstinence if of childbearing potential
  • Ability to comply with study procedures
  • For pharmacokinetic study participants: body weight between 50-100 kg at consent
Not Eligible

You will not qualify if you...

  • Prior systemic antitumor therapy except neoadjuvant/adjuvant fluoropyrimidine chemotherapy
  • Previous anti-EGFR antibody or EGFR tyrosine kinase inhibitor therapy
  • Concurrent immunotherapy, hormonal cancer therapy, or unapproved cancer treatments
  • Major surgery within 28 days or recent radiotherapy with toxicity within 14 days before randomization
  • Presence of BRAF gene mutation
  • Severe comorbidities or life-threatening complications
  • Paralytic ileus, gastrointestinal obstruction, or uncontrolled diarrhea
  • Progressive or symptomatic central nervous system metastases requiring steroids or anticonvulsants
  • Serious cardiac conditions or uncontrolled hypertension
  • Severe respiratory failure or uncontrolled systemic diseases
  • Gilbert's syndrome
  • Hematologic abnormalities (neutrophils <1.5 x10^9/L, platelets <100 x10^9/L, hemoglobin <90 g/L)
  • Renal impairment (creatinine >1.5x ULN or GFR <45 mL/min)
  • Hepatic impairment (elevated bilirubin, AST/ALT, or ALP)
  • Feasibility for radical resection of metastases
  • History of other recent malignancies requiring treatment
  • Conditions limiting protocol compliance such as dementia or substance abuse
  • Participation in other clinical trials recently or previously in this trial
  • Acute infections within 28 days before randomization
  • Positive tests for hepatitis B, C, HIV, or syphilis
  • Inability to receive intravenous administration
  • Contraindication to intravenous contrast
  • Chronic corticosteroid use above specified doses
  • Hypersensitivity to study drugs or monoclonal antibody therapies
  • Pregnancy or breastfeeding
  • Excessive alcohol consumption or history of addiction
  • Other significant comorbidities affecting participation or study results
  • Inability to perform required blood sampling for pharmacokinetic analysis

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 26 locations

1

State Budgetary Healthcare Institution of the Arkhangelsk Region "Arkhangelsk Oncology Dispensary"

Arkhangelsk, Russia, 163045

Actively Recruiting

2

Moscow City Oncology Hospital No. 62 (MGOB 62)

Istra, Russia, 143515

Actively Recruiting

3

Regional Budgetary Healthcare Institution "Ivanovo Regional Oncology Dispensary"

Ivanovo, Russia, 153051

Actively Recruiting

4

State Budgetary Healthcare Institution of Kaluga Region "Kaluga Regional Clinical Oncology Dispensary"

Kaluga, Russia, 248007

Actively Recruiting

5

State Autonomous Healthcare Institution "Republican Clinical Oncology Dispensary of the Ministry of Health of the Republic of Tatarstan named after Professor M.Z. Sigal"

Kazan', Russia, 420029

Actively Recruiting

6

State Budgetary Healthcare Institution "Kuzbass Clinical Oncology Dispensary named after M.S. Rappoport" (SBHI "KCOD")

Kemerovo, Russia, 650036

Actively Recruiting

7

State Budgetary Healthcare Organisation "Clinical Oncology Dispensary No. 1" under the Ministry of Healthcare of Krasnodar region

Krasnodar, Russia, 350040

Actively Recruiting

8

Regional Budgetary Healthcare Institution "Kursk Oncology Research and Clinical Center named after G.E. Ostroverkhov"

Kursk, Russia, 305524

Actively Recruiting

9

State Budgetary Healthcare Institution "Leningrad Regional Clinical Hospital"

Kuz'molovskiy, Russia, 191104

Actively Recruiting

10

The Loginov Moscow Clinical Scientific Center (MCSC)

Moscow, Russia, 111123

Actively Recruiting

11

N.N. Blokhin National Medical Research Center of Oncology (Blokhin NRC of Oncology)

Moscow, Russia, 115522

Actively Recruiting

12

Oncology Center No. 1 of the City Clinical Hospital named after S.S. Yudin of the Moscow Healthcare Department

Moscow, Russia, 117152

Actively Recruiting

13

I.M. Sechenov First Moscow State Medical University (Sechenov University)

Moscow, Russia, 119435

Actively Recruiting

14

Branch of the Limited Liability Company "Hadassah Medical Ltd." (LLC Branch "Hadassah Medical")

Moscow, Russia, 121205

Actively Recruiting

15

Federal State Autonomous Institution "National Medical Research Center 'Medical and Rehabilitation Center'" of the Ministry of Health of the Russian Federation

Moscow, Russia, 125367

Actively Recruiting

16

Research Lab LLC

Moscow, Russia, 127521

Actively Recruiting

17

Joint-Stock Company "Medsi Group of Companies"

Moscow, Russia, 143442

Actively Recruiting

18

Limited Liability Company Medical and Sanitary Unit "Clinician-Pretor Clinic"

Novosibirsk, Russia, 630091

Actively Recruiting

19

Federal State Budgetary Healthcare Institution "Clinical Hospital No. 8 of the Federal Medical-Biological Agency of Russia"

Obninsk, Russia, 249032

Actively Recruiting

20

Federal State Budgetary Institution "National Medical Research Center of Radiology" of the Ministry of Health of the Russian Federation, Branch: P.A. Herzen Moscow Research Oncology Institute

Obninsk, Russia, 249036

Actively Recruiting

21

Omsk Region Budgetary Healthcare Institution "Clinical Oncology Dispensary"

Omsk, Russia, 644013

Actively Recruiting

22

Private Healthcare Institution "Clinical Hospital "RZD-Medicine" of Saint-Petersburg"

Saint Petersburg, Russia, 195271

Actively Recruiting

23

City Clinical Oncology Dispensary (Saint Petersburg)

Saint Petersburg, Russia, 198255

Actively Recruiting

24

State Health Institution "Tula Regional Clinical Oncology Dispensary"

Tula, Russia, 300039

Actively Recruiting

25

State Budgetary Healthcare Institution "Volgograd Regional Clinical Oncology Dispensary"

Volgograd, Russia, 400138

Actively Recruiting

26

State Institution of Healthcare of Yaroslavl Region "Regional Oncology Hospital"

Yaroslavl, Russia, 150054

Actively Recruiting

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Research Team

A

Andrey Osherov

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

DOUBLE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

2

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