Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT05598151

Dose Escalation and Expansion Study of HM97662 in Advanced or Metastatic Solid Tumors

Led by Hanmi Pharmaceutical Company Limited · Updated on 2025-04-30

170

Participants Needed

10

Research Sites

281 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This is a Phase1 study to assess the safety, PK, PD and efficacy of HM97662, EZH1/2 dual inhibitor, in solid tumors. The study is comprised of Dose-Escalation Part followed by randomized Dose-Ranging Part and Dose-Expansion Part. Dose-Escalation Part is planned with a 3+3 Dose-Escalation design and is to establish the MTD or RD for randomized Dose-Ranging Part. Dose-Ranging Part is designed mainly to further evaluate safety and preliminary efficacy of HM97662 monotherapy in subjects with specific genomic alterations to more precisely determine the potential RP2D that are to be tested in a Dose-Expansion Part. Dose-Expansion Part is designed to assess the potential efficacy of HM97662 monotherapy when administered at the RP2D to subjects in indication-specific expansion cohorts.

CONDITIONS

Official Title

Dose Escalation and Expansion Study of HM97662 in Advanced or Metastatic Solid Tumors

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Histologically and/or cytologically confirmed advanced or metastatic solid tumor who have failed or are intolerant to standard therapy.
  • Patients in the dose-escalation part must have evaluable or measurable disease at baseline.
  • Patients in the randomized dose-ranging and dose-expansion parts must have at least one measurable lesion at baseline by CT or MRI per RECIST v1.1.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  • Life expectancy of at least 3 months before starting HM97662.
  • Adequate kidney function.
  • Adequate blood cell counts.
  • Adequate liver function.
  • Males or females aged 18 years or older (or country's legal age of majority if higher) at informed consent.
  • For dose-ranging part, documented alteration in at least one gene of the SWI/SNF complex in tumor tissue (archival or newly obtained).
Not Eligible

You will not qualify if you...

  • Prior exposure to valemetostat or other EZH1/2 dual inhibitors.
  • Known brain metastases that are untreated, symptomatic, or require therapy to control symptoms.
  • Currently taking medications that are strong CYP3A inhibitors or strong/moderate CYP3A inducers.
  • Clinically significant toxicities from prior treatments that have not resolved to Grade 1 or lower per CTCAE v5.0 or are clinically unstable.
  • Major surgery within 4 weeks before first dose of study drug.
  • Females who are pregnant or breastfeeding.
  • Patients who have had an organ transplant.

AI-Screening

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Trial Site Locations

Total: 10 locations

1

Cancer Research SA

Adelaide, Australia

Actively Recruiting

2

Grampians Health

Ballarat, Australia

Actively Recruiting

3

Monash Medical Centre

Clayton, Australia

Actively Recruiting

4

Peninsula and Southeast Oncology

Frankston, Australia

Actively Recruiting

5

National Cancer Center

Goyang-si, Gyeonggi-do, South Korea

Not Yet Recruiting

6

Asan Medical Center

Seoul, South Korea

Actively Recruiting

7

Samsung Medical Center

Seoul, South Korea

Not Yet Recruiting

8

Seoul National University Bundang Hospital

Seoul, South Korea

Actively Recruiting

9

Seoul National University Hospital

Seoul, South Korea

Actively Recruiting

10

The Catholic University of Korea, Seoul ST. Mary's Hospital

Seoul, South Korea

Actively Recruiting

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Research Team

J

Jiyeon Yoon

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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