Actively Recruiting

Phase 2
Age: 18Years +
All Genders
ID06995677

A Phase 2 Multicenter, Open-Label Study Evaluating the Efficacy and Safety of TYRA-300 in Participants With FGFR3 Altered Low Grade, Intermediate Risk Non-Muscle Invasive Bladder Cancer (SURF302)

Led by Tyra Biosciences, Inc · Updated on 2026-05-20

90

Participants Needed

40

Research Sites

30 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating the efficacy and safety of TYRA-300 in adults with low-grade, intermediate-risk non-muscle invasive bladder cancer (NMIBC) that has specific FGFR3 gene alterations. This Phase 2 multicenter study focuses on patients who have residual visible tumors and meet certain risk criteria, aiming to better understand treatment effects in this particular group. Participants receive self-administered oral tablets of TYRA-300 daily at doses of 50mg, 60mg, or a dose to be determined. The study is randomized and open-label, with three experimental dose cohorts. Treatment continues while monitoring for tumor response and safety over time. During the study, participants will undergo assessments including bladder mapping, tumor evaluations, and laboratory tests to monitor organ function and treatment effects. Researchers will measure tumor response at 3 months, duration of response, time to recurrence, recurrence-free survival, progression-free survival, and safety outcomes up to 2 years. Participants will be followed and monitored regularly throughout the study period.

CONDITIONS

Brief Title

Efficacy and Safety of TYRA-300 in Participants With FGFR3 Altered Low Grade, Intermediate Risk Non-Muscle Invasive Bladder Cancer

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Participants age 18 years and older who can give informed consent and comply with study procedures
  • Able to understand and provide written informed consent
  • Histologically confirmed low-grade non-muscle invasive bladder cancer (Ta or T1) within 6 weeks prior to randomization
  • Residual visible tumor between 3 mm and 12 mm as a marker lesion
  • Intermediate risk NMIBC as defined by recurrence within 1 year, solitary tumor larger than 3 cm, multifocal tumor, or T1 low grade
  • Documented activating FGFR3 mutation or fusion
  • Underwent bladder mapping and identification of visible marker lesion(s) within 6 weeks prior to randomization
  • No evidence of urothelial carcinoma of upper urinary tract or prostatic urethra within 6 months
  • No prior BCG administration within 1 year before consent
  • No intravesical chemotherapy within 8 weeks prior to first treatment day
  • ECOG performance status 0-1
  • Pathology consistent with at least 80% urothelial carcinoma if mixed histology
  • Adequate bone marrow, liver, and renal function as specified
  • Ability to swallow tablets
  • Willingness to use effective contraception during and after treatment as required
  • HIV positive participants must have undetectable viral load and stable antiretroviral therapy
  • Participants with chronic hepatitis B or C must meet specific viral load and treatment criteria
Not Eligible

You will not qualify if you...

  • Presence of tumor in ureter or prostatic urethra
  • History or current muscle invasive bladder cancer
  • History or current lymph node positive or metastatic bladder cancer
  • Pure squamous cell carcinoma, adenocarcinoma, or undifferentiated carcinoma of bladder
  • Currently receiving systemic cancer therapy or prohibited therapies
  • Prior pelvic radiotherapy
  • Prior FGFR inhibitor treatment
  • Systemic immunotherapy within 6 months prior to randomization
  • Treatment with investigational agents within 30 days or 5 half-lives prior to randomization
  • Prior intravesical agent treatment within 8 weeks before first treatment day
  • Ongoing toxicity from previous therapy
  • Major surgery within 4 weeks prior to first treatment day
  • Conditions impairing compliance or increasing risk, such as uncontrolled diabetes
  • Pregnant or breastfeeding females, or males planning to father a child during or shortly after treatment
  • Impaired wound healing capacity
  • Serum phosphate above normal limits
  • Eye conditions increasing risk of toxicity or current retinal disorders
  • Uncontrolled cardiovascular disease
  • Gastrointestinal disorders affecting oral drug absorption
  • Known active HIV or hepatitis B or C infection
  • Second primary malignancy within 3 years excluding certain skin and surveillance cancers
  • Allergy to TYRA-300 or its components
  • Use of strong CYP3A4 inhibitors or inducers
  • History of prolonged QT syndrome or QTcF interval over 470 ms

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Treatment

Duration - Up to 24 months

Participants receive daily oral doses of TYRA-300 as monotherapy for their bladder cancer.

Visits occur regularly during treatment to assess safety and response

Follow-up

Duration - Up to 24 months after treatment

Participants are monitored for recurrence, progression, and long-term safety after treatment ends.

Periodic visits for safety and efficacy assessments

Trial Site Locations

Total: 40 locations

1

Urology Centers of Alabama

Homewood, Alabama, United States, 35209

Actively Recruiting

2

Arkansas Urology

Little Rock, Arkansas, United States, 72211

Actively Recruiting

3

Tri Valley Urology - Murrieta

Murrieta, California, United States, 92562

Actively Recruiting

4

Om Research LLC

San Diego, California, United States, 92123

Actively Recruiting

5

Associated Urological Specialists

Chicago Ridge, Illinois, United States, 60415

Actively Recruiting

6

Duly Health and Care

Lisle, Illinois, United States, 60532

Actively Recruiting

7

Urology of Indiana

Greenwood, Indiana, United States, 46143

Actively Recruiting

8

First Urology

Jeffersonville, Indiana, United States, 47130

Actively Recruiting

9

University of Kansas Medical Center (KUMC)

Kansas City, Kansas, United States, 66160

Actively Recruiting

10

Johns Hopkins University

Baltimore, Maryland, United States, 21205

Actively Recruiting

11

Greater Boston Urology

Plymouth, Massachusetts, United States, 02360

Actively Recruiting

12

Atlantic Health System

Morristown, New Jersey, United States, 07960

Actively Recruiting

13

New Jersey Urology, LLC (Summit Health - Washington Township)

Voorhees Township, New Jersey, United States, 08043

Actively Recruiting

14

Memorial Sloan Kettering Cancer Center - Sidney Kimmel Center for Prostate and Urologic Cancers

New York, New York, United States, 10065

Actively Recruiting

15

Associated Medical Professionals of NY

Syracuse, New York, United States, 13210

Actively Recruiting

16

The Bronx Veterans Medical Research Foundation, Inc.

The Bronx, New York, United States, 10468

Actively Recruiting

17

Duke Cancer Institute

Durham, North Carolina, United States, 27705

Actively Recruiting

18

Associate Urologist of North Carolina

Raleigh, North Carolina, United States, 27612

Actively Recruiting

19

Oregon Urology Institute

Springfield, Ohio, United States, 97477

Actively Recruiting

20

MidLantic Urology

Bala-Cynwyd, Pennsylvania, United States, 19004

Actively Recruiting

21

Keystone Urology Specialists

Lancaster, Pennsylvania, United States, 17604

Actively Recruiting

22

Carolina Urologic Research Center

Myrtle Beach, South Carolina, United States, 29572

Actively Recruiting

23

Lowcounty Urology Clinics, P.A.

North Charleston, South Carolina, United States, 29406

Actively Recruiting

24

Conrad Pearson-Memphis

Germantown, Tennessee, United States, 38138

Actively Recruiting

25

Urology Associates PC

Nashville, Tennessee, United States, 37209

Actively Recruiting

26

Urology Austin

Austin, Texas, United States, 78759

Actively Recruiting

27

Baylor College of Medicine

Houston, Texas, United States, 77030

Actively Recruiting

28

Urology San Antonio

San Antonio, Texas, United States, 78229

Actively Recruiting

29

Epworth Freemasons-Victoria Parade

Richmond, Victoria, Australia, 3121

Actively Recruiting

30

Istituti Fisioterapici Ospitalieri (IFO)

Rome, Italy, Italy

Actively Recruiting

31

Istituto Europeo di Oncologia

Milan, Italy, 20141

Actively Recruiting

32

Azienda Ospedaliero Universitaria Pisana - Ospedale Santa Chiara

Pisa, Italy, 56126

Actively Recruiting

33

ASL Napoli 2 Nord - Ospedale Santa Maria delle Grazie

Pozzuoli, Italy, 80078

Actively Recruiting

34

Centro Médico Teknon

Barcelona, Spain, Spain, 08003

Actively Recruiting

35

Hospital Clínico San Carlos

Madrid, Spain, Spain, 28040

Active, Not Recruiting

36

Hospital Universitario 12 de Oc

Madrid, Spain, Spain, 28041

Actively Recruiting

37

Hospital Quirón Barcelona

Barcelona, Spain, 08908

Actively Recruiting

38

MD Anderson Cancer Center - Madrid

Madrid, Spain, 28003

Actively Recruiting

39

Hospital Universitario Ramón y Cajal

Madrid, Spain, 28034

Actively Recruiting

40

Hospital Universitario Marqués de Valdecilla

Santander, Spain, 39008

Actively Recruiting

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Research Team

G

Grace Indyk

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

3

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