Actively Recruiting

Phase 2
Age: 2Years - 100Years
All Genders
ID06997588

Study Assessing the Efficacy, Safety and Pharmacokinetics of Alpelisib in Pediatric and Adult Patients With PIK3CA-related Overgrowth Spectrum (PROS)

Led by Novartis Pharmaceuticals · Updated on 2026-06-02

104

Participants Needed

32

Research Sites

112 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating the effectiveness, safety, and tolerability of daily oral alpelisib in both children and adults with PIK3CA-related overgrowth spectrum (PROS), a condition characterized by abnormal tissue growth due to PIK3CA gene mutations. This Phase II study aims to provide important data on how alpelisib affects PROS symptoms and progression. The study includes a screening period of up to 42 days where eligibility is determined, including a whole body MRI to assess lesions related to PROS. The core treatment period lasts 48 weeks, with adults receiving 250 mg of alpelisib once daily, children aged 6 to under 18 years receiving 125 mg daily, and children aged 2 to under 6 years receiving 50 mg daily. Following this, participants may enter extension periods lasting up to two more years, continuing treatment under the same dosing rules. Those still benefiting at study end may access alpelisib post-trial. Participants will have regular assessments including MRI scans to measure lesion size and presence of new lesions, evaluations of pain and symptom severity, and blood tests to measure alpelisib levels. These assessments occur at multiple time points throughout the trial and extensions, up to approximately three years. The main outcome measured is the proportion of participants showing a confirmed objective response by week 48, with safety and long-term effects closely monitored.

CONDITIONS

Brief Title

EPIK-P4: A Phase II Single-arm Study to Assess the Efficacy, Safety and Pharmacokinetics of Alpelisib (BYL719) in Pediatric and Adult Patients With PIK3CA-related Overgrowth Spectrum (PROS)

Who Can Participate

Age: 2Years - 100Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Male or female participants aged 2 years or older at the time of informed consent/assent
  • Diagnosis of PROS with symptomatic and progressive overgrowth, including syndromic disease or isolated features (except isolated macrodactyly, macrocephaly, or epidermal nevus)
  • Documented somatic mutation in the PIK3CA gene confirmed by DNA-based test
  • Karnofsky or Lansky performance status index of 50 or higher
  • PGI-S score of mild, moderate, severe, or very severe at screening
  • Adequate bone marrow and organ function
  • At least one measurable PROS-related lesion of 2 cm or larger associated with symptoms or functional limitations
Not Eligible

You will not qualify if you...

  • Participants with only isolated macrodactyly, epidermal nevus/nevi, and macroencephaly without other PROS-related lesions
  • Previous treatment with alpelisib or other PI3K inhibitors, except brief attempts under 2 weeks stopped at least 4 weeks before study
  • Major surgery within 3 months prior to consent
  • Radiation treatment for PROS within 12 months prior to consent
  • Significant PROS-related thrombotic event within 30 days before consent or recent vascular procedures within 6 weeks
  • Significant bleeding from PROS lesion within 30 days before treatment start
  • Clinically significant worsening of PROS-related lab abnormalities or symptoms during screening phase
  • Other inclusion/exclusion criteria may apply

AI-Screening

AI-Powered Screening

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Your Study Journey

Screening

Duration - Up to 6 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person) including a whole body MRI scan

Treatment

Duration - 48 weeks for the core period, followed by up to 2 years in extension periods

Participants receive alpelisib to assess its efficacy, safety, and pharmacokinetics in treating PROS. Dosing varies by age group and continues during the core and extension periods.

Multiple visits for treatment and assessments up to approximately 3 years

Trial Site Locations

Total: 32 locations

1

Washington University

St Louis, Missouri, United States, 63110

Actively Recruiting

2

Cinn Children Hosp Medical Center

Cincinnati, Ohio, United States, 45229-3039

Actively Recruiting

3

Childrens Hosp Pittsburgh UPMC

Pittsburgh, Pennsylvania, United States, 15224

Actively Recruiting

4

Baylor College Of Medicine

Houston, Texas, United States, 77030

Actively Recruiting

5

Novartis Investigative Site

Sydney, New South Wales, Australia, 2010

Actively Recruiting

6

Novartis Investigative Site

Sydney, New South Wales, Australia, 2031

Actively Recruiting

7

Novartis Investigative Site

North Adelaide, South Australia, Australia, 5066

Actively Recruiting

8

Novartis Investigative Site

Salzburg, Austria, 5020

Actively Recruiting

9

Novartis Investigative Site

Vienna, Austria, A 1090

Actively Recruiting

10

Novartis Investigative Site

Ghent, Belgium, 9000

Actively Recruiting

11

Novartis Investigative Site

Angers, France, 49933

Actively Recruiting

12

Novartis Investigative Site

Bron, France, 69677

Actively Recruiting

13

Novartis Investigative Site

Dijon, France, 21000

Actively Recruiting

14

Novartis Investigative Site

Montpellier, France, 34295

Actively Recruiting

15

Novartis Investigative Site

Paris, France, 75015

Actively Recruiting

16

Novartis Investigative Site

Toulouse, France, 31400

Actively Recruiting

17

Novartis Investigative Site

Tours, France, 37044

Actively Recruiting

18

Novartis Investigative Site

Freiburg im Breisgau, Baden-Wurttemberg, Germany, 79106

Actively Recruiting

19

Novartis Investigative Site

Düsseldorf, North Rhine-Westphalia, Germany, 40225

Actively Recruiting

20

Novartis Investigative Site

Leipzig, Saxony, Germany, 04103

Actively Recruiting

21

Novartis Investigative Site

Halle, Saxony-Anhalt, Germany, 06120

Actively Recruiting

22

Novartis Investigative Site

Berlin, Germany, 13353

Actively Recruiting

23

Novartis Investigative Site

Stuttgart, Germany, 70374

Actively Recruiting

24

Novartis Investigative Site

Roma, RM, Italy, 00168

Actively Recruiting

25

Novartis Investigative Site

Torino, TO, Italy, 10126

Actively Recruiting

26

Novartis Investigative Site

Trieste, TS, Italy, 34137

Actively Recruiting

27

Novartis Investigative Site

Esplugues, Barcelona, Spain, 08950

Actively Recruiting

28

Novartis Investigative Site

A Coruña, Spain, 15006

Actively Recruiting

29

Novartis Investigative Site

Barcelona, Spain, 08035

Actively Recruiting

30

Novartis Investigative Site

Madrid, Spain, 28046

Actively Recruiting

31

Novartis Investigative Site

Lausanne, Switzerland, 1011

Actively Recruiting

32

Novartis Investigative Site

Liverpool, United Kingdom, L12 2AP

Actively Recruiting

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Research Team

N

Novartis Pharmaceuticals

N

Novartis Pharmaceuticals

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

2

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