Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
ID05919264

A Phase 1/2 Study of FOG-001 in Participants With Locally Advanced or Metastatic Solid Tumors

Led by Parabilis Medicines, Inc. · Updated on 2026-05-28

595

Participants Needed

33

Research Sites

21 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating FOG-001 for safety, tolerability, pharmacokinetics, pharmacodynamics, and anti-tumor activity in people with locally advanced or metastatic solid tumors that likely or known to have mutations activating the Wnt pathway. This first-in-human, phase 1/2, multicenter study includes dose escalation and expansion phases to assess FOG-001 alone and in combination with other cancer drugs. FOG-001 is given either intravenously or subcutaneously in continuous 28-day cycles. Some participants receive FOG-001 alone, while others receive it combined with mFOLFOX-6, Nivolumab, Trifluridine/tipiracil, or Bevacizumab according to prescribing information. Multiple study parts include treatment of various cancers such as colorectal, hepatocellular carcinoma, desmoid tumors, and prostate cancer, based on specific mutation status. Participants will undergo safety evaluations including monitoring for adverse events and dose-limiting toxicities over approximately 10 months. Tumor response is assessed regularly using imaging criteria, along with specific measurements like PSA30 for prostate cancer. Pharmacokinetic and pharmacodynamic tests are done during early cycles. The study involves frequent visits for treatment administration, scans, lab tests, biopsies, and clinical assessments to track treatment effects and safety throughout the study period.

CONDITIONS

Brief Title

FOG-001 in Locally Advanced or Metastatic Solid Tumors

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • Adequate organ and marrow function
  • Diagnosis of treatment-refractory advanced/metastatic solid tumor with documented WNT-pathway activating mutations or non-MSI-H/non-dMMR colorectal cancer (CRC) for dose escalation cohorts
  • At least one lesion suitable for core needle biopsy for certain dose escalation cohorts
  • Histologically, cytologically, or radiographically confirmed hepatocellular carcinoma (HCC) with documented WPAM in APC or CTNNB1 for select cohorts
  • Diagnosis of desmoid tumor (aggressive fibromatosis) for certain cohorts
  • Diagnosis of locally advanced or metastatic non-MSI-H or non-dMMR CRC with specific mutation status for combination therapy cohorts
  • Diagnosis of advanced or metastatic solid tumors with documented WPAM or equivalent evidence for dose expansion cohorts
Not Eligible

You will not qualify if you...

  • Known history of bone metastasis except for patients with metastatic castration-resistant prostate cancer
  • Vertebral compression fracture or non-traumatic bone fracture within past 12 months without antiresorptive therapy
  • Osteoporosis defined as T-score ≤ -2.5 at lumbar spine, femoral neck, or total hip by DXA scan
  • Uncontrolled inflammatory bowel disease (ulcerative colitis or Crohn's disease)
  • Unstable or inadequate cardiac function
  • Known meningeal carcinomatosis, leptomeningeal carcinomatosis, spinal cord compression, or symptomatic or unstable brain metastases
  • Pregnant, lactating, or planning to become pregnant

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person) for screening and enrollment

Treatment

Duration - Repeated 28-day cycles until disease progression or discontinuation

Participants receive FOG-001 and may receive other anticancer agents according to assigned doses in continuous 28-day cycles to evaluate safety, tolerability, and antitumor activity.

Visits every 28 days for treatment administration with additional assessments every 63 days

Follow-up

Duration - Up to approximately 10 months on average after treatment

Participants are monitored for safety and disease status after treatment completion.

Visits approximately every 63 days for response and safety assessments

Trial Site Locations

Total: 33 locations

1

Mayo Clinic

Phoenix, Arizona, United States, 85054

Actively Recruiting

2

Honor Health

Scottsdale, Arizona, United States, 85258

Actively Recruiting

3

Arizona Cancer Center at University of Arizona

Tucson, Arizona, United States, 85719

Actively Recruiting

4

University of California, Los Angeles (UCLA)

Los Angeles, California, United States, 90095

Actively Recruiting

5

Stanford Cancer Institute, Stanford University

Palo Alto, California, United States, 94304

Actively Recruiting

6

University of California San Francisco, Helen Diller Family Comprehensive Cancer Center

San Francisco, California, United States, 94158

Actively Recruiting

7

Sarcoma Oncology Center

Santa Monica, California, United States, 90403

Actively Recruiting

8

University of Colorado

Aurora, Colorado, United States, 80045

Actively Recruiting

9

Yale University School of Medicine

New Haven, Connecticut, United States, 06520

Actively Recruiting

10

Johns Hopkins University, Sibley Memorial Hospital

Washington D.C., District of Columbia, United States, 20016

Actively Recruiting

11

Mayo Clinic

Jacksonville, Florida, United States, 32224

Actively Recruiting

12

Florida Cancer Specialists

Lake Mary, Florida, United States, 32746

Terminated

13

Johns Hopkins University, The Sidney Kimmel Comprehensive Cancer Center

Baltimore, Maryland, United States, 21287

Actively Recruiting

14

Massachusetts General Hospital

Boston, Massachusetts, United States, 02114

Actively Recruiting

15

Dana Farber Cancer Institute

Boston, Massachusetts, United States, 02215

Actively Recruiting

16

M Health Fairview University of Minnesota Medical Center

Minneapolis, Minnesota, United States, 55455

Actively Recruiting

17

Mayo Clinic

Rochester, Minnesota, United States, 55905

Actively Recruiting

18

Washington University School of Medicine

St Louis, Missouri, United States, 63110

Actively Recruiting

19

Memorial Sloan Kettering Cancer Center

New York, New York, United States, 10065

Actively Recruiting

20

Duke University

Durham, North Carolina, United States, 27705

Actively Recruiting

21

University Hospitals Cleveland Medical Center, Seidman Cancer Center

Cleveland, Ohio, United States, 44106

Actively Recruiting

22

Cleveland Clinic

Cleveland, Ohio, United States, 44195

Actively Recruiting

23

Oregon Health and Science University

Portland, Oregon, United States, 97239

Actively Recruiting

24

University of Pennsylvania, Perelman School of Medicine

Philadelphia, Pennsylvania, United States, 19104

Actively Recruiting

25

University of Pittsburgh Medical Center, Hillman Cancer Center

Pittsburgh, Pennsylvania, United States, 15232

Actively Recruiting

26

Sarah Cannon Research Institute

Nashville, Tennessee, United States, 37203

Actively Recruiting

27

Vanderbilt Ingram Cancer Center

Nashville, Tennessee, United States, 37232

Actively Recruiting

28

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States, 77030

Actively Recruiting

29

South Texas Accelerated Research Therapeutics, LLC

San Antonio, Texas, United States, 78229

Actively Recruiting

30

University of Virginia

Charlottesville, Virginia, United States, 22908

Actively Recruiting

31

University of Wisconsin, Carbone Cancer Center

Madison, Wisconsin, United States, 53705

Actively Recruiting

32

Integrated Clinical Oncology Network (ICON)

South Brisbane, Queensland, Australia, 4101

Actively Recruiting

33

Peter MacCallum Cancer Centre

Melbourne, Victoria, Australia, 3000

Actively Recruiting

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Research Team

C

Clinical Trial Inquiries

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

18

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