Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
MALE
NCT07002320

Investigating SX-682 in Combination With Apalutamide in Metastatic Castration-resistant Prostate Cancer

Led by Institute of Cancer Research, United Kingdom · Updated on 2026-04-15

78

Participants Needed

4

Research Sites

231 weeks

Total Duration

On this page

Sponsors

I

Institute of Cancer Research, United Kingdom

Lead Sponsor

P

Prostate Cancer UK

Collaborating Sponsor

AI-Summary

What this Trial Is About

ASpiRE will investigate the effect of the drug SX-682 in combination with Apalutamide in men suffering from metastatic castration-resistant prostate cancer (mCRPC).

CONDITIONS

Official Title

Investigating SX-682 in Combination With Apalutamide in Metastatic Castration-resistant Prostate Cancer

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Written informed consent and ability to cooperate with treatment
  • Age 18 years or older
  • Confirmed adenocarcinoma of the prostate with accessible tumor tissue for analysis
  • For phase 1 cohorts, biopsiable disease with consent for pre- and post-treatment biopsies
  • Diagnosis of metastatic castration-resistant prostate cancer
  • Documented resistance to at least one prior next generation antiandrogen therapy (enzalutamide, Apalutamide, or darolutamide) with minimum 12 weeks treatment
  • Documented prostate cancer progression by standard criteria including RECIST v1.1, PCWG3 bone scan, or PSA progression
  • PSA level of 10 ng/ml or higher
  • Prior castration by surgery or ongoing hormone therapy
  • Ongoing androgen deprivation with serum testosterone below 50 ng/dL
  • ECOG Performance Status of 2 or less
  • Willingness to use effective contraception during and 6 months after treatment
  • Ability to swallow study drug tablets
  • Steroid use discontinued if possible; up to 5 mg twice daily prednisolone allowed
  • Hematological and biochemical parameters within specified ranges measured within one week before starting trial
Not Eligible

You will not qualify if you...

  • Surgery, chemotherapy, or other anti-cancer therapy within 4 weeks before trial entry, except certain antiandrogen therapies
  • Participation in another interventional clinical trial within 4 weeks prior
  • Recent radiotherapy within 2 to 4 weeks before trial entry
  • Clinical or biochemical hyperaldosteronism or hypopituitarism
  • History of seizures or predisposing brain conditions
  • Malabsorption syndrome or conditions affecting drug absorption
  • Certain cardiac conditions including prolonged QTcF interval, arrhythmias, recent serious cardiac events, uncontrolled blood pressure
  • Significant liver disease or cirrhosis
  • Conditions contraindicating investigational drug use or causing high treatment risk
  • Other malignancies within 5 years except treated basal cell carcinoma
  • Unresolved significant toxicity from prior therapy
  • Inability to comply with study procedures
  • Predominantly small cell or neuroendocrine prostate cancer
  • Immunocompromised status
  • Active or uncontrolled autoimmune disease requiring corticosteroids
  • Recent thromboembolic disease within 12 months
  • Serious concurrent illness or infection
  • Known intolerance to Apalutamide, SX-682, or components
  • Symptoms or documented infection of COVID-19
  • Use of prohibited medications including certain antipsychotics, antidepressants, anticoagulants, and others
  • History of severe drug-induced skin reactions or pneumonitis requiring steroids

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 4 locations

1

Oncology Institute of Southern Switzerland

Bellinzona, Switzerland, CH6500

Not Yet Recruiting

2

Belfast Health and Social Care Trust

Belfast, United Kingdom, BT9 7AB

Actively Recruiting

3

Cambridge University Hospitals NHS Foundation Trust

Cambridge, United Kingdom, CB2 0QQ

Actively Recruiting

4

The Royal Marsden NHS Foundation Trust - Drug Development Unit

Sutton, United Kingdom, SM2 5PT

Actively Recruiting

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Research Team

A

Aasia Hussain, PhD

CONTACT

B

Bindumalini Rao Baikady, PhD

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

2

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Investigating SX-682 in Combination With Apalutamide in Metastatic Castration-resistant Prostate Cancer | DecenTrialz