Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT07222267

An Investigational Study of BG-75202 Alone and in Combination With Other Therapeutic Agents in Adults With Advanced Solid Tumors

Led by BeOne Medicines · Updated on 2026-05-11

86

Participants Needed

25

Research Sites

578 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics (PK), pharmacodynamics, and preliminary antitumor activity of BG-75202 (KAT6A/B inhibitor) alone and in combination with other therapies in participants with breast cancer and other advanced solid tumors.

CONDITIONS

Official Title

An Investigational Study of BG-75202 Alone and in Combination With Other Therapeutic Agents in Adults With Advanced Solid Tumors

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Participants with confirmed advanced, metastatic breast cancer or other solid tumors who have no effective standard therapies left or cannot tolerate them (Part 1A).
  • Participants with advanced breast cancer with 1 to 3 prior systemic therapy lines in the metastatic setting, with no more than 2 lines of chemotherapy (Parts 1B and 2A).
  • Participants with advanced breast cancer in areas without approved or available CDK4/6 inhibitors as first-line treatment, who have not received CDK4/6 inhibitors or systemic treatment for advanced disease (Parts 2B and 2C).
  • Participants with breast cancer must have confirmed advanced breast cancer per ASCO/CAP guidelines.
  • Female participants with metastatic breast cancer must be postmenopausal or receiving ovarian function suppression treatment.
  • Measurable disease by RECIST v 1.1 criteria.
  • Stable ECOG Performance Status of 0 or 1.
  • Adequate organ function.
Not Eligible

You will not qualify if you...

  • Prior treatment with KAT6A/B or KAT7 inhibitors or degraders.
  • Active leptomeningeal disease or uncontrolled, untreated brain metastases.
  • Any other malignancy within 3 years before screening except the cancer under study or treated local recurrence unlikely to need intervention during the study.
  • Additional protocol-defined criteria may apply.

AI-Screening

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Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 25 locations

1

University of Alabama At Birmingham Hospital

Birmingham, Alabama, United States, 35294-0004

Actively Recruiting

2

Yale Cancer Center

New Haven, Connecticut, United States, 06510

Actively Recruiting

3

Washington University in St Louis

St Louis, Missouri, United States, 63110-1010

Actively Recruiting

4

Next Oncology Austin

Austin, Texas, United States, 78758

Actively Recruiting

5

The University of Texas Md Anderson Cancer Center

Houston, Texas, United States, 77030-4009

Actively Recruiting

6

Blacktown Cancer and Haematology Centre

Blacktown, New South Wales, Australia, NSW 2148

Actively Recruiting

7

Chris Obrien Lifehouse

Camperdown, New South Wales, Australia, NSW 2050

Actively Recruiting

8

Cancer Research South Australia

Adelaide, South Australia, Australia, SA 5000

Actively Recruiting

9

Peter Maccallum Cancer Centre

Melbourne, Victoria, Australia, VIC 3000

Actively Recruiting

10

Cancer Hospital Chinese Academy of Medical Sciences

Beijing, Beijing Municipality, China, 100021

Actively Recruiting

11

Beijing Cancer Hospital

Beijing, Beijing Municipality, China, 100142

Actively Recruiting

12

Sun Yat Sen University Cancer Center Huangpu Branch

Guangzhou, Guangdong, China, 510555

Actively Recruiting

13

Harbin Medical University Cancer Hospital

Harbin, Heilongjiang, China, 150000

Actively Recruiting

14

Jiangsu Province Hospital Longjiang Branch

Nanjing, Jiangsu, China, 210036

Actively Recruiting

15

Fudan University Shanghai Cancer Centerpudong

Shanghai, Shanghai Municipality, China, 201321

Actively Recruiting

16

Tianjin Medical University Cancer Institute and Hospital

Tianjin, Tianjin Municipality, China, 300060

Actively Recruiting

17

Istituto Europeo Di Oncologia

Milan, Italy, 20141

Actively Recruiting

18

Istituto Nazionale Tumori Fondazione G Pascale

Naples, Italy, 80131

Actively Recruiting

19

Fondazione Policlinico Universitario Agostino Gemelli

Roma, Italy, 00168

Actively Recruiting

20

Istituto Clinico Humanitas

Rozzano, Italy, 20089

Actively Recruiting

21

Hospital Universitario Vall Dhebron

Barcelona, Spain, 08035

Actively Recruiting

22

Next Oncology Barcelona

Barcelona, Spain, 8023

Actively Recruiting

23

Hospital Universitario 12 de Octubre

Madrid, Spain, 28041

Actively Recruiting

24

Hospital Clinico San Carlos

Madrid, Spain, 28240

Actively Recruiting

25

Hospital Universitario Virgen de La Victoria

Málaga, Spain, 29010

Actively Recruiting

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Research Team

S

Study Director

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

5

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