Actively Recruiting

Phase 1
Age: 18Years - 70Years
All Genders
NCT03973268

Mechanism of Action Underlying Ketamine's Antidepressant Effects: The AMPA Throughput Theory in Patients With Treatment-Resistant Major Depression

Led by National Institute of Mental Health (NIMH) · Updated on 2026-02-24

70

Participants Needed

1

Research Sites

366 weeks

Total Duration

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AI-Summary

What this Trial Is About

Background: Most drugs that treat mood disorders take a long time to work. Ketamine works within hours. A dose can last for a week or more. Certain receptors in the brain might help ketamine work. A drug that blocks these receptors might affect how it works. Objective: To see if the antidepressant response of ketamine is linked to AMPA receptors. Eligibility: Adults ages 18-70 with major depression disorder without psychotic features Design: Participants will be screened under protocol 01-M-0254. They will have blood tests and a physical exam. Participants will stay at the NIH Clinical Center for 5 weeks. Phase 1 lasts 4 weeks. For 2 weeks, participants will taper off their psychiatric medicine. Then they will have the following tests: * Blood draws * Psychological tests * MRI: Participants will lie in a machine that takes pictures of their brain. * MEG: Participants will lie down and do tasks. A cone lowered on their head will record brain activity. * Optional sleep tests: Electrodes on the scalp and body and belts around the body will monitor participants while they sleep. * Optional TMS: Participants will do tasks while a wire coil is held on their scalp. An electrical current will pass through the coil that affects brain activity. For phase 2, on day 0 participants will take the study drug or a placebo orally. While having a MEG, they will get ketamine infused into a vein in one arm while blood is drawn from a vein in the other arm. On day 1, participants will again take the study drug or a placebo orally. On days 3-7, they will repeat many of the phase 1 tests. Days 8 and 9 are optional and include an open label ketamine treatment and many of the phase 1 tests.

CONDITIONS

Official Title

Mechanism of Action Underlying Ketamine's Antidepressant Effects: The AMPA Throughput Theory in Patients With Treatment-Resistant Major Depression

Who Can Participate

Age: 18Years - 70Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Age between 18 and 70 years
  • Ability to understand and agree to all tests and sign informed consent
  • Completed screening under protocol 01-M-0254
  • Diagnosis of major depressive disorder without psychotic features based on clinical assessment
  • Initial Montgomery-Asberg Depression Rating Scale (MADRS) score of 22 or higher and Young Mania Rating Scale (YMRS) score below 12
  • Lack of response to at least two adequate antidepressant treatments, including current episode
  • Current major depressive episode lasting at least four weeks
  • Agree to be hospitalized during study participation
  • For open-label ketamine treatment, completion of Phase II and use of effective birth control or sexual abstinence if able to become pregnant
Not Eligible

You will not qualify if you...

  • Current psychotic features or diagnosis of schizophrenia or other psychotic disorders
  • Substance abuse or dependence within past 3 months (except caffeine or nicotine) and negative drug/alcohol tests at screening
  • Serious unstable medical illnesses including liver, kidney, heart, lung, endocrine, neurological, immune, or blood disorders
  • Pregnancy, nursing, or physical ability to become pregnant without effective birth control during study
  • History of seizures, epilepsy, stroke, brain surgery, head injury, or structural brain lesions
  • Medical conditions likely to alter brain structure or function, even if controlled
  • Significant abnormal lab tests
  • Hearing loss that could worsen with imaging procedures
  • Positive HIV test
  • Weight over 119 kg
  • Use of psychiatric or non-psychiatric medications prior to Phase II (must be tapered during Phase I)
  • Use of opioid medications in past 3 months
  • Use of reversible monoamine oxidase inhibitors (MAOI) prior to Phase II
  • Use of fluoxetine or aripiprazole at screening
  • Unwillingness to stop structured psychotherapy during Phases I and II
  • Presence of metallic implants
  • Claustrophobia or inability to lie still for imaging
  • Serious suicidal or homicidal risk or history of aggressive behavior
  • Current NIMH staff or immediate family member
  • For open-label treatment, serious adverse reactions to ketamine or positive drug test before treatment
  • Pregnancy or nursing during open-label treatment

AI-Screening

AI-Powered Screening

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Trial Site Locations

Total: 1 location

1

National Institutes of Health Clinical Center

Bethesda, Maryland, United States, 20892

Actively Recruiting

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Research Team

Y

Yamila I Carmona

CONTACT

C

Carlos A Zarate, M.D.

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

TRIPLE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

BASIC_SCIENCE

Number of Arms

3

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