Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT05274048

Neratinib and Fam-Trastuzumab Deruxtecan in Advanced Gastro-esophageal Cancer Patients

Led by Fox Chase Cancer Center · Updated on 2025-10-29

18

Participants Needed

3

Research Sites

257 weeks

Total Duration

On this page

Sponsors

F

Fox Chase Cancer Center

Lead Sponsor

N

National Comprehensive Cancer Network

Collaborating Sponsor

AI-Summary

What this Trial Is About

This is Phase 1 dose finding trial with potential dose expansion to evaluate the safety, toxicity, recommended phase 2 dose (RP2D), and maximum tolerated dose (MTD) of Neratinib plus TDxD using a standard 3+3 dose escalation design in patients with metastatic or unresectable gastro-esophageal cancer that are HER2-overexpressing (IHC 3+ or IHC2+/ISH+) and any other gastrointestinal cancer with HER2 expression with IHC3+. Patients must have progressed or been intolerant of at least one prior line of chemotherapy + HER2 directed therapy.

CONDITIONS

Official Title

Neratinib and Fam-Trastuzumab Deruxtecan in Advanced Gastro-esophageal Cancer Patients

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Diagnosed with unresectable or metastatic gastrointestinal cancer confirmed by biopsy
  • Have measurable or evaluable disease by RECIST 1.1 criteria
  • Tumors must overexpress HER2: IHC 3+ or IHC 2+/ISH+ for gastroesophageal cancer, or IHC 3+ for other GI cancers
  • Received at least one prior HER2 directed therapy for metastatic/unresectable gastroesophageal cancer, completed at least 2 weeks before treatment start
  • Prior or concurrent malignancies are allowed if they do not interfere with safety or efficacy assessment
  • Age over 18 years
  • ECOG performance status between 0 and 2
  • Normal organ and marrow function as defined by specific blood count and chemistry thresholds
  • Left Ventricular Ejection Fraction of 45% or higher
  • Females of childbearing potential and males with partners of childbearing potential must agree to effective contraception during and after treatment
  • Able and willing to swallow oral tablets
  • Able to understand and willing to sign informed consent and HIPAA documents
Not Eligible

You will not qualify if you...

  • Received chemotherapy or radiotherapy within 2 weeks before treatment start or not recovered from prior treatment side effects
  • Receiving other investigational agents or previously treated with TDxD
  • Immunotherapy or investigational treatments not discontinued for more than 21 days before treatment
  • Have untreated brain metastases; treated brain metastases must be stable for at least 4 weeks
  • Have ongoing diarrhea of more than 4 bowel movements per day despite care in the past 2 weeks
  • History or suspicion of interstitial lung disease or pneumonitis, or significant lung disease requiring oxygen support
  • History of allergic reactions to similar drugs used in the study
  • Taking medications that strongly affect Neratinib or TDxD metabolism
  • Uncontrolled illness including infections, heart failure, unstable angina, arrhythmia, or psychiatric/social conditions limiting compliance
  • QTcF interval prolongation above specified thresholds
  • Immune deficiency including uncontrolled HIV with low CD4 count or untreated hepatitis B
  • Pregnant or breastfeeding

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 3 locations

1

Stanford Cancer Center

Palo Alto, California, United States, 94304

Actively Recruiting

2

Roswell Park Comprehensive Cancer Center

Buffalo, New York, United States, 14263

Actively Recruiting

3

Fox Chase Cancer Center

Philadelphia, Pennsylvania, United States, 19111

Actively Recruiting

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Research Team

N

Namrata Vijavergia, MD

CONTACT

T

Tanu Singh

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

1

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Neratinib and Fam-Trastuzumab Deruxtecan in Advanced Gastro-esophageal Cancer Patients | DecenTrialz