Actively Recruiting

Phase 1
Age: 18Years - 80Years
All Genders
NCT06225856

An Open-Label, Multicenter, Phase I Study to Evaluate the Safety, Pharmacokinetics and Preliminary Efficacy of YY201 in Patients With Advanced Solid Tumors and Hematological Malignancies

Led by Shanghai Yuyao Biotech Co., Ltd. · Updated on 2024-01-31

96

Participants Needed

1

Research Sites

165 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This is a multicenter, open-label, phase I clinical study of YY201 in the patients with relapsed/refractory lymphomas and relapsed/refractory large granular lymphocytic leukemia who failed or cannot tolerate standard treatment.

CONDITIONS

Official Title

An Open-Label, Multicenter, Phase I Study to Evaluate the Safety, Pharmacokinetics and Preliminary Efficacy of YY201 in Patients With Advanced Solid Tumors and Hematological Malignancies

Who Can Participate

Age: 18Years - 80Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Patients must understand and sign informed consent and be able to follow all study procedures.
  • Aged between 18 and 80 years, male or female.
  • Patients with advanced solid tumors or relapsed/refractory hematologic malignancies who have failed or cannot tolerate standard treatments.
  • For advanced solid tumors in the dose-escalation phase, at least one tumor lesion evaluable by RECIST v1.1.
  • For dose-expansion phase, measurable tumor lesions per RECIST v1.1, with specific criteria for previously irradiated tumors.
  • Enrollment in dose-expansion phase limited to advanced solid tumors sensitive to STAT3 therapy, peripheral T-cell lymphoma with STAT3 mutation refractory or relapsed after therapy, and relapsed/refractory acute myeloid leukemia sensitive to STAT3 therapy excluding certain subtypes.
  • ECOG performance status of 1 or less.
  • For advanced primary liver cancer, Child-Pugh liver function grade A or better grade B (7 or less).
  • Adequate bone marrow, liver, kidney, and coagulation function according to specified laboratory thresholds.
  • Agreed to provide tumor tissue samples in dose-expansion phase.
  • Expected survival of at least 3 months.
  • Women of childbearing potential must have a negative pregnancy test within 7 days before first dose and agree to use effective contraception during and 30 days after treatment.
Not Eligible

You will not qualify if you...

  • Previous adverse reactions from anti-cancer therapy have not recovered to CTCAE grade 1 or less, except for certain non-safety-risk toxicities.
  • Symptomatic central nervous system metastases or CNS involvement for AML patients.
  • Recent chemotherapy, radiation, biological, endocrine, or immune therapies within 4 weeks before first dose, with some exceptions.
  • Use of other investigational drugs within 4 weeks before first dose.
  • Prior use of STAT3 inhibitors for anti-tumor treatment.
  • Major organ surgery within 4 weeks before first dose or planned elective surgery during the trial.
  • Uncontrolled malignant pleural, ascites, or pericardial effusions.
  • Inability to swallow oral medication or conditions affecting gastrointestinal absorption.
  • Use of strong CYP3A4 inducers or inhibitors within 1 week before first dose or planned during study.
  • Active gastrointestinal diseases or bleeding conditions.
  • Recent thromboembolic events within 12 months.
  • Significant cardiovascular disease including recent heart attack, severe angina, heart failure, low ejection fraction, or prolonged QTc.
  • Active or previous autoimmune diseases with potential recurrence, excluding stable thyroid disease and type I diabetes.
  • Prior immunotherapy with severe immune-related adverse events.
  • Significant electrolyte abnormalities.
  • Active infections requiring treatment or fever above 38.5°C before dosing.
  • Active tuberculosis, HIV infection, or active hepatitis B or C infections.
  • Recent hematopoietic stem cell transplant or ongoing immunosuppressive therapy or graft-versus-host disease requiring drug control.
  • Pregnant or breastfeeding women.
  • Men wishing to father children.
  • Known alcohol or drug dependence.
  • Inability to comply with study procedures.
  • Any other clinically significant disease or abnormality that may affect safety or study results.

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 1 location

1

Shanghai East Hospital

Shanghai, Shanghai Municipality, China

Actively Recruiting

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Research Team

Y

Ye Guo

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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An Open-Label, Multicenter, Phase I Study to Evaluate the Safety, Pharmacokinetics and Preliminary Efficacy of YY201 in Patients With Advanced Solid Tumors and Hematological Malignancies | DecenTrialz