Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
MALE
ID06785636

Phase 1b/2a Open-Label Study of Pocenbrodib Alone or with Abiraterone Acetate, Olaparib, or 177Lu-PSMA-617 in Men with Metastatic Castration-Resistant Prostate Cancer

Led by Pathos AI, Inc. · Updated on 2026-04-24

252

Participants Needed

18

Research Sites

43 weeks

Total Duration

On this page

Sponsors

P

Pathos AI, Inc.

Lead Sponsor

D

Duke University

Collaborating Sponsor

AI-Summary

What this Trial Is About

Researchers are evaluating the safety, pharmacokinetics, preliminary antitumor activity, and pharmacodynamics of pocenbrodib, alone or combined with abiraterone acetate, olaparib, or 177Lu-PSMA-617, in men with metastatic castration-resistant prostate cancer (mCRPC) who have progressed after prior therapies including at least one potent anti-androgen treatment. This Phase 1b/2a open-label study aims to find an appropriate dose and assess early treatment effects in this population. The Phase 1b part tests five increasing doses of pocenbrodib monotherapy (50, 100, 150, 200, and 250 mg) given once daily for 5 days followed by 2 days off. Participants start at the lowest dose with careful safety monitoring before moving to higher doses. If safety and minimum efficacy are demonstrated, Phase 2a begins, enrolling four groups: pocenbrodib alone, or combined with abiraterone acetate, olaparib, or 177Lu-PSMA-617. These groups run simultaneously but are evaluated separately. Participants will have regular assessments including imaging and prostate-specific antigen (PSA) tests to measure treatment response and progression. Safety and dose-limiting toxicities are closely tracked over 28-day cycles. Pharmacokinetic measures like plasma drug concentrations and half-life will be recorded. The study period extends up to about 32 months, with outcomes such as tumor response, progression-free survival, and overall survival monitored to understand the treatment's effects.

CONDITIONS

Brief Title

Open-Label Study of Pocenbrodib Alone and in Combination With Abiraterone Acetate, Olaparib, or 177Lu-PSMA-617

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • 18 years of age or older
  • Histologic confirmation of prostate adenocarcinoma
  • Metastatic disease confirmed by imaging within 56 days before screening
Not Eligible

You will not qualify if you...

  • Evidence of small cell or neuroendocrine prostate cancer on recent biopsy
  • Liver metastases confirmed by biopsy or lesions larger than 1 cm on imaging
  • Treatment with chemotherapy, investigational agents, or certain antiandrogen drugs within 14 days before screening or five half-lives, whichever is shorter
  • Serious medical, psychiatric, psychological, familial, or geographical conditions that may interfere with participation or increase treatment risk

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Run-in Period

Duration - Multiple 28-day cycles during Phase 1b

Participants receive escalating doses of pocenbrodib monotherapy to determine safety and appropriate dosing.

Visits occur at the end of each 28-day cycle for safety and pharmacokinetic assessments

Treatment

Duration - Up to approximately 6 months or until disease progression or unacceptable toxicity

Participants receive pocenbrodib alone or in combination with abiraterone acetate, olaparib, or 177Lu-PSMA-617 depending on cohort assignment, with dosing schedules of 5 days on followed by 2 days off each week.

Regular visits throughout treatment for dosing, safety, and efficacy evaluations

Follow-up

Duration - Up to approximately 32 months from first dose

Participants are monitored for overall survival and long term safety after treatment ends.

Periodic visits for survival and safety assessments

Trial Site Locations

Total: 18 locations

1

MemorialCare Orange Coast Medical Center

Fountain Valley, California, United States, 92708

Actively Recruiting

2

Cancer and Blood Research Center

Los Alamitos, California, United States, 90720

Actively Recruiting

3

University of Colorado Health

Aurora, Colorado, United States, 80045

Actively Recruiting

4

Mount Sinai Medical Center

Miami, Florida, United States, 33140

Actively Recruiting

5

Emory University Hospital

Atlanta, Georgia, United States, 30322

Actively Recruiting

6

University of Chicago

Chicago, Illinois, United States, 60637

Actively Recruiting

7

Community Health Network

Indianapolis, Indiana, United States, 46250

Actively Recruiting

8

Ochsner

Jefferson, Louisiana, United States, 70121

Actively Recruiting

9

Johns Hopkins Hospital

Baltimore, Maryland, United States, 21287

Actively Recruiting

10

Karmanos Cancer Institute

Detroit, Michigan, United States, 48201

Actively Recruiting

11

Siteman Cancer Center

St Louis, Missouri, United States, 63108

Actively Recruiting

12

Nebraska Cancer Specialists

Omaha, Nebraska, United States, 68130

Actively Recruiting

13

Duke University medical center

Durham, North Carolina, United States, 27710

Actively Recruiting

14

The Ohio State University

Columbus, Ohio, United States, 43210

Actively Recruiting

15

Taylor Cancer Research Center

Maumee, Ohio, United States, 43537

Actively Recruiting

16

University of Texas Southwestern Medical Center

Dallas, Texas, United States, 75390

Actively Recruiting

17

Oncology Consultants, P.A

Houston, Texas, United States, 77030

Actively Recruiting

18

NEXT Oncology - Virginia

Fairfax, Virginia, United States, 22031

Actively Recruiting

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Research Team

S

Steve Kye, MD. MPH

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

2

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