Actively Recruiting

Phase 2
Age: 18Years +
All Genders
NCT04945148

Oxidative Phosphorylation Targeting In Malignant Glioma Using Metformin Plus Radiotherapy Temozolomide

Led by Hopital Foch · Updated on 2025-11-21

640

Participants Needed

7

Research Sites

207 weeks

Total Duration

On this page

Sponsors

H

Hopital Foch

Lead Sponsor

N

National Cancer Institute, France

Collaborating Sponsor

AI-Summary

What this Trial Is About

Tailored approaches targeting crucial oncogenes and pathways have shown successful results in a number of cancer types and offer exciting perspective in neuro-oncology. IDH (Isocitrate dehydrogenase) wild-type (IDHwt) glioblastoma (GBM) (10%) present a unique and homogenous energetic metabolism which is specifically dependent on the oxidative phosphorylation (OXPHOS) rather than on the aerobic glycolysis. OXPHOS+ IDHwt GBMs overexpress mitochondrial markers and can be specifically inhibited by mitochondrial inhibitors in vitro and in vivo. Metformin is an oral inhibitor of mitochondrial complex I and is a widely used drug in diabetic and non-diabetic patients, safe and well tolerated in association with radiotherapy and chemotherapy. Basing on drastic effect, the investigators have observed in vivo (reduction of \>50% of tumor growth) and hypothesize that metformin could be specifically efficient to treat up-front patients affected by OXPHOS+ GBM, in association with the standard first-line treatment with radiotherapy and temozolomide (RT-TMZ). The investigators set up a dedicated molecular analysis including RNA assay and expression of OXPHOS markers for formalin-fixed paraffin-embedded tumors (FFPE), which allows to detect OXPHOS+ GBM at diagnosis. Here a phase II, open label, non-randomized multicenter trial including five French neurooncology centers (H. Foch-Suresnes, Pitié-Salpêtrière-Paris, Saint Louis-Paris, Lyon, Marseille) and one in Italy (Istituto Besta, Milan) is proposed. Newly diagnosed IDH wild-type GBM patients with the OXPHOS+ signature will be eligible for inclusion in this trial. The investigators expect to screen 640 patients and to include 64 patients over a period of 24 months with 24 months of follow-up.

CONDITIONS

Official Title

Oxidative Phosphorylation Targeting In Malignant Glioma Using Metformin Plus Radiotherapy Temozolomide

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Signed informed consent obtained before any study procedures
  • Willingness and ability to comply with study treatment, visits, and follow-up
  • Newly diagnosed, histologically confirmed supratentorial IDH wild-type glioblastoma (Grade 4 malignant glioma)
  • Tumor shows OXPHOS+ subtype by central laboratory testing
  • No prior treatment for glioblastoma except surgery
  • Recovery from surgery without major ongoing safety issues
  • On stable or no corticosteroid treatment (dexamethasone ≤ 6 mg or equivalent)
  • Eastern Cooperative Oncology Group performance status 0-2
  • Able to receive combined radiotherapy and chemotherapy per Stupp protocol
  • Adequate bone marrow and liver function
  • Creatinine clearance ≥ 30 mL/min (dose adjustment for 30-50 mL/min)
  • Able to start radiotherapy within 7 weeks after diagnosis
  • Life expectancy of at least 16 weeks
  • Affiliated with appropriate health insurance
  • Age 18 years or older
  • Women of childbearing potential with negative pregnancy test within 7 days before study drug
  • Women of childbearing potential agree to contraception during treatment and for 30 days after last dose
  • Sexually active males agree to contraception during treatment and for 6 months after last dose
  • White blood cells ≥ 2000/μL
  • Neutrophils ≥ 1500/μL
  • Platelets ≥ 100,000/μL
  • Hemoglobin ≥ 9.0 g/dL
  • Serum creatinine ≤ 1.5 times upper limit of normal or creatinine clearance ≥ 30 mL/min
  • AST ≤ 3.0 times upper limit of normal
  • ALT ≤ 3.0 times upper limit of normal
  • Total bilirubin ≤ 1.5 times upper limit of normal (or ≤ 3.0 for Gilbert Syndrome patients)
Not Eligible

You will not qualify if you...

  • Prior glioblastoma treatment other than surgery, including Gliadel wafer
  • Second primary cancer except treated non-melanoma skin cancer, treated in-situ cervical cancer, or other treated solid tumors with no disease for ≥ 5 years
  • Known metastatic extracranial or leptomeningeal disease
  • IDH mutant glioblastoma
  • Secondary glioblastoma from prior lower-grade glioma
  • Serious or uncontrolled medical disorder increasing study risk or interfering with treatment
  • Unable to swallow oral medication or gastrointestinal disorders affecting absorption
  • Pregnant or breastfeeding women
  • Immunocompromised patients, including HIV positive on antiviral therapy
  • Active hepatitis B or C infection
  • Known allergy to metformin, temozolomide, or their components
  • Severe renal insufficiency (creatinine clearance < 30 mL/min)
  • Other central nervous system disorders unrelated to cancer unless controlled or non-interfering
  • Unable or unwilling to have contrast-enhanced brain MRI
  • Acute medical conditions impairing kidney function such as dehydration or severe infection
  • Diseases causing tissue hypoxia like heart failure, respiratory failure, or recent heart attack
  • Past diabetic precoma or acute metabolic acidosis
  • Alcohol intoxication or alcoholism
  • Persons under legal protection regimes
  • Prisoners or involuntarily incarcerated individuals
  • Patients compulsorily detained for psychiatric or infectious disease treatment

AI-Screening

AI-Powered Screening

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Trial Site Locations

Total: 7 locations

1

Foch Hospital

Suresnes, Hauts de Seine, France, 92150

Actively Recruiting

2

Hôpital Neurologique Pierre Wertheimer

Bron, Lyon, France, 69500

Actively Recruiting

3

Timone Hospital

Marseille, Marseille, France, 13354

Actively Recruiting

4

Saint Louis Hospital

Paris, Paris, France, 75010

Actively Recruiting

5

Pitié Salpêtrière Hospital

Paris, PARIS, France, 75013

Actively Recruiting

6

Istituto Nazionale Carlo Besta

Milan, Milano, Italy, 20131

Not Yet Recruiting

7

Spidali Riuniti Di Livorno

Livorno, Toscana Nord Ouest, Italy, 57100

Not Yet Recruiting

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Research Team

A

Anna Luisa DI STEFANO, MD

CONTACT

E

Elisabeth HULIER-AMMAR, PhD

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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