Actively Recruiting

Phase 2
Age: 18Years +
MALE
NCT05766371

Pembrolizumab Plus 177Lu-PSMA-617 in Patients With Castration Resistant Prostate Cancer

Led by University of California, San Francisco · Updated on 2026-04-17

48

Participants Needed

1

Research Sites

389 weeks

Total Duration

On this page

Sponsors

U

University of California, San Francisco

Lead Sponsor

M

Merck Sharp & Dohme LLC

Collaborating Sponsor

AI-Summary

What this Trial Is About

This is a single-center, open-label, study of Prostate-Specific Membrane Antigen (PSMA)-targeted radionuclide therapy with 177Lu-PSMA-617 in combination with pembrolizumab in participants with metastatic castrate-resistant prostate cancer (mCRPC) who have previously progressed on at least one prior androgen pathway inhibitor (e.g., abiraterone, enzalutamide, apalutamide).

CONDITIONS

Official Title

Pembrolizumab Plus 177Lu-PSMA-617 in Patients With Castration Resistant Prostate Cancer

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Histologically confirmed metastatic castration-resistant prostate cancer progressing per PCWG3 criteria
  • Male participants aged 18 years or older
  • Castrate serum testosterone level below 50 ng/dL; if no bilateral orchiectomy, must continue LHRH analogue treatment
  • Prior progression on at least one second-generation androgen signaling inhibitor (e.g., abiraterone, enzalutamide, apalutamide, darolutamide)
  • Recovery to Grade �3=1 for prior anti-cancer treatment side effects (except alopecia and Grade �2 neuropathy)
  • Prior radiotherapy allowed if last treatment was over 2 weeks before study start and patient has recovered with no corticosteroid need or pneumonitis
  • At least one PSMA PET avid lesion with uptake above liver background
  • ECOG performance status of 0 or 1 (Karnofsky �3= 70%)
  • Adequate bone marrow, liver, and kidney function as specified
  • Use of effective contraception during treatment and for 6 months after
  • Consent to follow radioprotection precautions
  • Willingness to undergo tumor biopsy if accessible
  • Previously treated brain metastases allowed if treatment was over 28 days ago, no new lesions on MRI, and stable without steroids
  • Prior or concurrent malignancies allowed if not interfering with study
  • Ability and willingness to sign informed consent
Not Eligible

You will not qualify if you...

  • De novo small cell neuroendocrine prostate cancer
  • Soft tissue lesions larger than specified that are negative on PSMA PET
  • Systemic anti-cancer therapy within 14 days before study start (except LHRH analogues)
  • Untreated brain metastases
  • Prior PSMA-directed treatment
  • Previous therapy with anti-PD-1, anti-PD-L1, anti-PD-L2, or other T-cell receptor agents
  • Participation in other investigational studies within 4 weeks before study start
  • More than 2 prior lines of taxane chemotherapy
  • Severe hypersensitivity to pembrolizumab or its components
  • Active autoimmune disease requiring systemic treatment within 2 years
  • Diagnosis of immunodeficiency or recent immunosuppressive therapy
  • History of significant pneumonitis or interstitial lung disease
  • Receipt of live vaccine within 30 days before study start
  • Inability to give valid informed consent due to age, medical, or psychiatric conditions
  • Significant cardiovascular disease as detailed
  • Recent major surgery or radiation involving large bone marrow area
  • Active infection requiring IV antibiotics
  • Active or untreated Hepatitis B or C infections except controlled cases
  • Active tuberculosis
  • Psychiatric or substance abuse disorders interfering with study participation
  • Bleeding disorders that prevent safe biopsy
  • Any condition impairing ability to comply with study procedures

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 1 location

1

University of California, San Francisco

San Francisco, California, United States, 94143

Actively Recruiting

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Research Team

U

UCSF Genitourinary Medical Oncology Recruitment

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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Pembrolizumab Plus 177Lu-PSMA-617 in Patients With Castration Resistant Prostate Cancer | DecenTrialz