Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT06439836

Pembrolizumab Plus CA-4948 for the Treatment of Patients With Progressive Metastatic Urothelial Cancer Despite Prior Immunotherapy

Led by National Cancer Institute (NCI) · Updated on 2026-05-13

27

Participants Needed

11

Research Sites

108 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This phase I trial tests the safety, side effects, best dose, and effectiveness of emavusertib (CA-4948) in combination with pembrolizumab in treating patients with urothelial cancer that has spread from where it first started to other places in the body (metastatic) and that has a resistance to PD-1/PD-L1 immune checkpoint inhibitors. CA-4948, a kinase inhibitor, may stop the growth of tumor cells by blocking some of the enzymes needed for cell growth. Immunotherapy with monoclonal antibodies, such as pembrolizumab, may help the body's immune system attack the tumor, and may interfere with the ability of tumor cells to grow and spread. Giving CA-4948 in combination with pembrolizumab may be safe, tolerable and/or effective in treating patients with metastatic urothelial cancer that is resistant to PD-1/PD-L1 immune checkpoint inhibitors.

CONDITIONS

Official Title

Pembrolizumab Plus CA-4948 for the Treatment of Patients With Progressive Metastatic Urothelial Cancer Despite Prior Immunotherapy

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Patients must have histologically confirmed metastatic or unresectable urothelial cancer
  • Age 18 years or older
  • Eastern Cooperative Oncology Group (ECOG) performance status 0 to 2 within 28 days prior to registration
  • Leukocyte count of at least 3,000/mcL
  • Absolute neutrophil count (ANC) of at least 1,500/mcL
  • Platelet count of at least 100,000/mcL
  • Hemoglobin level of at least 9 g/dL without recent red blood cell transfusion
  • Creatine phosphokinase less than or equal to grade 2
  • Creatinine less than 1.5 times institutional upper limit of normal or creatinine clearance of at least 30 mL/min
  • Total bilirubin less than or equal to 1.5 times institutional upper limit of normal
  • AST and ALT less than or equal to 3 times upper limit of normal
  • INR or prothrombin time less than or equal to 1.5 times upper limit of normal unless on therapeutic anticoagulants
  • aPTT less than or equal to 1.5 times upper limit of normal unless on therapeutic anticoagulants
  • Ability to provide tumor tissue samples or undergo biopsy
  • Measurable metastatic or unresectable disease
  • Prior treatment with a PD-1 or PD-L1 inhibitor
  • Prior treatment with platinum-based chemotherapy or enfortumab vedotin
  • Primary resistance to PD-1/PD-L1 blockade as defined by specific treatment and progression criteria
  • Negative pregnancy test for females of childbearing potential and agreement to use contraception
  • Agreement to use contraception for males of childbearing potential
  • HIV-infected patients on effective therapy with undetectable viral load within 6 months
  • Patients vaccinated for COVID-19 and influenza allowed
  • Patients with stable, previously treated brain metastases allowed
  • Patients with prior or concurrent malignancy not interfering with study allowed
  • Willingness and ability to swallow pills
  • Ability to understand and sign informed consent
Not Eligible

You will not qualify if you...

  • Patients with unresolved toxicities greater than grade 1 from prior cancer therapy except certain neuropathy or alopecia
  • Diagnosis of immunodeficiency or use of high-dose systemic steroids or immunosuppressive therapy within 7 days prior to study drug
  • Grade 3 or higher immune-related adverse events from prior PD-1/PD-L1 therapy
  • History of allergic reactions to CA-4948 or pembrolizumab analogs
  • Uncontrolled illnesses including lung disease, heart failure, unstable angina, or arrhythmia
  • Receiving other investigational agents
  • Presence of carcinomatous meningitis
  • Malabsorption syndrome or conditions interfering with intestinal absorption
  • Active autoimmune disease requiring systemic treatment in past 2 years
  • History or current pneumonitis requiring steroids
  • Conditions or lab abnormalities that could interfere with study participation
  • Receipt of live vaccine within 30 days before treatment
  • Pregnant or breastfeeding women
  • Known active hepatitis B or C infection
  • History of active tuberculosis

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 11 locations

1

City of Hope Comprehensive Cancer Center

Duarte, California, United States, 91010

Actively Recruiting

2

UCI Health - Chao Family Comprehensive Cancer Center and Ambulatory Care

Irvine, California, United States, 92612

Actively Recruiting

3

UC San Diego Moores Cancer Center

La Jolla, California, United States, 92093

Actively Recruiting

4

UC Irvine Health/Chao Family Comprehensive Cancer Center

Orange, California, United States, 92868

Actively Recruiting

5

University of Miami Miller School of Medicine-Sylvester Cancer Center

Miami, Florida, United States, 33136

Actively Recruiting

6

Emory University Hospital Midtown

Atlanta, Georgia, United States, 30308

Actively Recruiting

7

Emory University Hospital/Winship Cancer Institute

Atlanta, Georgia, United States, 30322

Actively Recruiting

8

Emory Saint Joseph's Hospital

Atlanta, Georgia, United States, 30342

Actively Recruiting

9

Mount Sinai Hospital

New York, New York, United States, 10029

Actively Recruiting

10

NYP/Weill Cornell Medical Center

New York, New York, United States, 10065

Actively Recruiting

11

UT Southwestern/Simmons Cancer Center-Dallas

Dallas, Texas, United States, 75390

Actively Recruiting

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How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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